erythrosine and daunorubicin

erythrosine has been researched along with daunorubicin in 35 studies

Research

Studies (35)

TimeframeStudies, this research(%)All Research%
pre-19905 (14.29)18.7374
1990's12 (34.29)18.2507
2000's13 (37.14)29.6817
2010's5 (14.29)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bauduin, P; Couvreur, P; Guiot, P; Kante, B; Roland, M; Speiser, P1
Duncan, R; Kopecek, J; Subr, V1
Chorváth, B; Sedlák, J1
Ekberg, M; Larsson, R; Nygren, P; Slater, L1
Hamburger AW Nora, RE; Joneckis, CC; Nora, RE; Ordóñez, JV; Ross, DD; Sisk, AM; Wu, RK1
Diener, E; Diner, UE; Sinha, A; Vergidis, R; Xie, S1
Bottiroli, G; Croce, AC; Prosperi, E; Supino, R1
El Egakey, MA; Speiser, P1
Broxterman, HJ; Feller, N; Pinedo, HM; Währer, DC1
Broxterman, HJ; Feller, N; Kuiper, CM; Lankelma, J; Pinedo, HM; Ruhdal, JK; Scheper, RJ1
Ichimura, K; Kashiwagura, T; Kawahara, K; Koike, M; Matsui, W; Takeguchi, N1
Fridborg, H; Killander, A; Kristensen, J; Larsson, R; Liliemark, J; Nygren, P; Oberg, G; Simonsson, B1
Bagrij, T; Twentyman, PR; Versantvoort, CH; Wright, KA1
Fujita, T; Fukuzumi, M; Muranishi, S; Nishimaki, A; Yamada, H; Yamamoto, A1
Ford, PJ; Germann, UA; Harding, MW; Mason, VS; Shlyakhter, D1
Berger, W; Elbling, L; Hauptmann, E; Kokoschka, EM; Micksche, M; Vetterlein, M1
Broxterman, HJ; Heijn, M; Lankelma, J; Wielinga, PR1
Garnier-Suillerot, A; Marbeuf-Gueye, C; Quidu, P; Salerno, M1
Borst, P; de Haas, M; Evers, R; Kool, M; Smith, AJ; van Deemter, L1
Anagnostopoulos, N; Androutsos, G; Galanopoulos, A; Kalmantis, T; Meletis, J; Paterakis, G; Rombos, Y; Sagriotis, A; Symeonidis, A; Tiniakou, M; Tsimberidou, AM; Yataganas, X; Zoumbos, N1
Albertioni, F; Eriksson, S; Lotfi, K; Månsson, E; Peterson, C1
Chorvath, B; Duraj, J; Hunakova, L; Jakubikova, J; Sedlak, J1
Litman, T; Skovsgaard, T; Stein, WD1
Driessen, AJ; Konings, WN; Lubelski, J; Mazurkiewicz, P; van Merkerk, R1
Castanys, S; Cortés-Selva, F; Gamarro, F; Jiménez, IA; Lu, P; Muñoz-Martínez, F; Pérez-Victoria, JM; Ravelo, AG; Sharom, FJ1
Garweg, JG; Goldblum, D; Wegmann-Burns, M1
Hu, X; Lu, Q; Pan, Q; Sun, M; Xu, X1
Bacsó, Z; Fenyvesi, F; Goda, K; Juhász, I; Krasznai, Z; Márián, T; Megyeri, A; Nagy, H; Szabó, G; Vecsernyés, M1
Kitagawa, S; Nabekura, T; Ueno, K; Yamaki, T1
Kitagawa, S; Nabekura, T; Yamaki, T1
Ampasavate, C; Phattanawasin, P; Piyapolrungroj, N; Sotanaphun, U1
Borska, S; Chmielewska, M; Dziegiel, P; Sopel, M; Zabel, M1
Schmitt, SM; Stefan, K; Wiese, M2
Elshawadfy, R; Namasivayam, V; Silbermann, K; Stefan, SM; Wiese, M1

Other Studies

35 other study(ies) available for erythrosine and daunorubicin

ArticleYear
Polycyanoacrylate nanocapsules as potential lysosomotropic carriers: preparation, morphological and sorptive properties.
    The Journal of pharmacy and pharmacology, 1979, Volume: 31, Issue:5

    Topics: Adsorption; Capsules; Chemistry, Pharmaceutical; Cyanoacrylates; Daunorubicin; Fluoresceins; Hydrogen-Ion Concentration; Lysosomes; Microscopy, Electron, Scanning; Microspheres; Particle Size

1979
Release of macromolecules and daunomycin from hydrophilic gels containing enzymatically degradable bonds.
    Journal of biomaterials science. Polymer edition, 1990, Volume: 1, Issue:4

    Topics: Amino Acid Sequence; Animals; Biodegradation, Environmental; Chymotrypsin; Daunorubicin; Dextrans; Fluorescein-5-isothiocyanate; Fluoresceins; Gels; Kinetics; Liver; Molecular Sequence Data; Molecular Structure; Oligopeptides; Polymethacrylic Acids; Rats

1990
Fluorescent double labeling of normal and malignant hematopoietic cells by monoclonal antibodies (FITC) and anthracycline cytostatic drug (Daunomycin): a cytometric technique for analysis of drug uptake in hematopoietic cell subpopulations.
    Neoplasma, 1991, Volume: 38, Issue:1

    Topics: Antibodies, Monoclonal; Antigens, CD; Cell Line; Daunorubicin; Drug Resistance; Flow Cytometry; Fluorescein-5-isothiocyanate; Fluoresceins; Fluorescent Antibody Technique; Granulocytes; Hematopoietic Stem Cells; Humans; Lymphocytes; Thiocyanates; Tumor Cells, Cultured

1991
Chemotherapeutic drug sensitivity testing of human leukemia cells in vitro using a semiautomated fluorometric assay.
    Leukemia, 1990, Volume: 4, Issue:8

    Topics: Cell Count; Cell Survival; Daunorubicin; Drug Resistance; Drug Screening Assays, Antitumor; Fluoresceins; Fluorometry; Humans; Leukemia; Leukemia, Myeloid; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Tumor Cells, Cultured; Vincristine

1990
Estimation of cell survival by flow cytometric quantification of fluorescein diacetate/propidium iodide viable cell number.
    Cancer research, 1989, Jul-15, Volume: 49, Issue:14

    Topics: Animals; Antineoplastic Agents; Cell Count; Cell Cycle; Cell Line; Cell Survival; Dactinomycin; Daunorubicin; Flow Cytometry; Fluoresceins; Humans; Indicators and Reagents; Propidium; Tumor Stem Cell Assay; Vincristine

1989
Specific immunosuppression by immunotoxins containing daunomycin.
    Science (New York, N.Y.), 1986, Jan-10, Volume: 231, Issue:4734

    Topics: Animals; Autoimmune Diseases; Concanavalin A; Daunorubicin; Fluorescein; Fluoresceins; Immunosuppression Therapy; Immunosuppressive Agents; Lymphocyte Activation; Mice; Mice, Inbred CBA; Nitrohydroxyiodophenylacetate; Ovalbumin; Picrates; Spleen; T-Lymphocytes

1986
Anthracycline-induced inhibition of membrane permeability functions dependent on metabolic energy.
    British journal of cancer, 1986, Volume: 54, Issue:6

    Topics: Adenosine Triphosphate; Cell Membrane Permeability; Cell Survival; Daunorubicin; Doxorubicin; Energy Metabolism; Fluoresceins; Glucose; HeLa Cells; Humans; Time Factors

1986
Drug loading studies on ultrafine solid carriers by sorption procedures.
    Pharmaceutica acta Helvetiae, 1982, Volume: 57, Issue:8

    Topics: Absorption; Chemistry, Pharmaceutical; Dactinomycin; Daunorubicin; Fluorescein; Fluoresceins

1982
ATP-dependent efflux of calcein by the multidrug resistance protein (MRP): no inhibition by intracellular glutathione depletion.
    FEBS letters, 1995, Jul-17, Volume: 368, Issue:2

    Topics: Adenosine Triphosphate; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Biological Transport, Active; Buthionine Sulfoximine; Cytoplasm; Daunorubicin; Fluoresceins; Glutathione; Humans; Indicators and Reagents; Methionine Sulfoximine; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Probenecid; Tumor Cells, Cultured

1995
Functional detection of MDR1/P170 and MRP/P190-mediated multidrug resistance in tumour cells by flow cytometry.
    British journal of cancer, 1995, Volume: 72, Issue:3

    Topics: Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Daunorubicin; Drug Resistance, Multiple; Flow Cytometry; Fluoresceins; Fluorescent Dyes; Humans; KB Cells; Multidrug Resistance-Associated Proteins; Rhodamine 123; Rhodamines; Sensitivity and Specificity

1995
Inhibition of the multidrug efflux pump in isolated hepatocyte couplets by immunosuppressants FK506 and cyclosporine.
    Transplantation, 1993, Volume: 55, Issue:3

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bile Canaliculi; Cyclosporine; Daunorubicin; Drug Resistance; Fluoresceins; Fluorescent Dyes; Fura-2; Liver; Membrane Glycoproteins; Microscopy, Fluorescence; Progesterone; Rats; Signal Processing, Computer-Assisted; Tacrolimus; Verapamil; Vinblastine

1993
Interactions between cladribine (2-chlorodeoxyadenosine) and standard antileukemic drugs in primary cultures of human tumor cells from patients with acute myelocytic leukemia.
    Leukemia, 1994, Volume: 8, Issue:10

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Amsacrine; Antineoplastic Agents; Cladribine; Cytarabine; Daunorubicin; Drug Interactions; Drug Screening Assays, Antitumor; Drug Synergism; Etoposide; Female; Fluoresceins; Humans; Leukemia, Myeloid, Acute; Male; Middle Aged; Mitoxantrone; Tumor Cells, Cultured

1994
On the relationship between the probenecid-sensitive transport of daunorubicin or calcein and the glutathione status of cells overexpressing the multidrug resistance-associated protein (MRP).
    International journal of cancer, 1995, Dec-11, Volume: 63, Issue:6

    Topics: Antimetabolites, Antineoplastic; ATP-Binding Cassette Transporters; Biological Transport; Buthionine Sulfoximine; Daunorubicin; Fluoresceins; Glutathione; Humans; Methionine Sulfoximine; Multidrug Resistance-Associated Proteins; Probenecid; Tumor Cells, Cultured

1995
Calcein is excreted from the intestinal mucosal cell membrane by the active transport system.
    Life sciences, 1997, Volume: 60, Issue:4-5

    Topics: Animals; Azides; Biological Transport, Active; Caco-2 Cells; Calcium Channel Blockers; Cell Membrane; Cell Membrane Permeability; Daunorubicin; Enzyme Inhibitors; Fluoresceins; Fluorescent Dyes; Humans; In Vitro Techniques; Intestinal Mucosa; Jejunum; Probenecid; Rats; Renal Agents; Sodium Azide; Sodium Fluoride; Verapamil

1997
Chemosensitization and drug accumulation effects of VX-710, verapamil, cyclosporin A, MS-209 and GF120918 in multidrug resistant HL60/ADR cells expressing the multidrug resistance-associated protein MRP.
    Anti-cancer drugs, 1997, Volume: 8, Issue:2

    Topics: Acridines; Affinity Labels; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Cyclosporine; Daunorubicin; Doxorubicin; Drug Resistance, Multiple; Etoposide; Fluoresceins; HL-60 Cells; Humans; Isoquinolines; Multidrug Resistance-Associated Proteins; Piperidines; Pyridines; Quinolines; Tetrahydroisoquinolines; Tritium; Verapamil; Vincristine

1997
Possible role of the multidrug resistance-associated protein (MRP) in chemoresistance of human melanoma cells.
    International journal of cancer, 1997, Mar-28, Volume: 71, Issue:1

    Topics: Adult; Aged; Aged, 80 and over; Antibiotics, Antineoplastic; Antineoplastic Agents; ATP-Binding Cassette Transporters; Benzbromarone; Blotting, Northern; Cisplatin; Daunorubicin; Doxorubicin; Drug Resistance, Neoplasm; Enzyme Inhibitors; Ethylmaleimide; Etoposide; Female; Fluoresceins; Humans; Male; Melanoma; Middle Aged; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Probenecid; RNA, Messenger; Tumor Cells, Cultured; Uricosuric Agents; Vinblastine

1997
P-glycoprotein-independent decrease in drug accumulation by phorbol ester treatment of tumor cells.
    Biochemical pharmacology, 1997, Oct-01, Volume: 54, Issue:7

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Daunorubicin; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Etoposide; Fluoresceins; Humans; Hydrogen-Ion Concentration; KB Cells; Protein Kinase C; Tetradecanoylphorbol Acetate

1997
Inhibition of the P-glycoprotein- and multidrug resistance protein-mediated efflux of anthracyclines and calceinacetoxymethyl ester by PAK-104P.
    European journal of pharmacology, 2000, Mar-17, Volume: 391, Issue:3

    Topics: Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Cyclic P-Oxides; Daunorubicin; Depression, Chemical; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Epirubicin; Fluoresceins; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Nicotinic Acids; Tumor Cells, Cultured

2000
Inhibitory effect of the reversal agents V-104, GF120918 and Pluronic L61 on MDR1 Pgp-, MRP1- and MRP2-mediated transport.
    British journal of cancer, 2000, Volume: 83, Issue:3

    Topics: Acridines; Anion Transport Proteins; Antibiotics, Antineoplastic; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport, Active; Carrier Proteins; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Etoposide; Fluoresceins; Humans; Isoquinolines; Methamphetamine; Poloxamer; Tetrahydroisoquinolines; Time Factors; Vinblastine

2000
Evaluation of the clinical relevance of the expression and function of P-glycoprotein, multidrug resistance protein and lung resistance protein in patients with primary acute myelogenous leukemia.
    Leukemia research, 2002, Volume: 26, Issue:2

    Topics: Acute Disease; Adolescent; Adult; Age Factors; Aged; Antineoplastic Combined Chemotherapy Protocols; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bone Marrow Transplantation; Calcium Channel Blockers; Carbocyanines; Combined Modality Therapy; Cytarabine; Daunorubicin; Disease-Free Survival; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Enzyme Inhibitors; Female; Fluoresceins; Fluorescent Dyes; Genistein; Humans; Idarubicin; Immunophenotyping; Leukemia, Myeloid; Male; Middle Aged; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Probenecid; Prognosis; Prospective Studies; Rhodamine 123; Survival Analysis; Tumor Cells, Cultured; Vault Ribonucleoprotein Particles; Verapamil

2002
Low level of mitochondrial deoxyguanosine kinase is the dominant factor in acquired resistance to 9-beta-D-arabinofuranosylguanine cytotoxicity.
    Biochemical and biophysical research communications, 2002, May-24, Volume: 293, Issue:5

    Topics: Anthracyclines; Antineoplastic Agents; Arabinonucleosides; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Cells, Cultured; Cyclosporine; Daunorubicin; Deoxycytidine Kinase; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Electrophoresis, Polyacrylamide Gel; Flow Cytometry; Fluoresceins; Humans; Mitochondria; Nucleosides; Phosphorylation; Phosphotransferases (Alcohol Group Acceptor); Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tumor Cells, Cultured

2002
PK11195, an isoquinoline carboxamide ligand of the mitochondrial benzodiazepine receptor, increased drug uptake and facilitated drug-induced apoptosis in human multidrug-resistant leukemia cells in vitro.
    Neoplasma, 2002, Volume: 49, Issue:4

    Topics: Antineoplastic Agents; Apoptosis; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Carcinoma; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Synergism; Female; Fluoresceins; Fluorescent Dyes; HL-60 Cells; Humans; Isoquinolines; Leukemia, Myeloid; Ligands; Mitochondrial Proteins; Ovarian Neoplasms; Receptors, GABA-A; Tumor Cells, Cultured

2002
Pumping of drugs by P-glycoprotein: a two-step process?
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 307, Issue:3

    Topics: Algorithms; Animals; Anti-Bacterial Agents; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Calcium Channel Blockers; Carcinoma, Ehrlich Tumor; Cell Line, Tumor; Cyclosporine; Daunorubicin; Fluoresceins; Humans; Immunosuppressive Agents; Kinetics; Models, Biological; Pharmaceutical Preparations; Quinolines; Verapamil; Vinblastine

2003
ydaG and ydbA of Lactococcus lactis encode a heterodimeric ATP-binding cassette-type multidrug transporter.
    The Journal of biological chemistry, 2004, Aug-13, Volume: 279, Issue:33

    Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Antibiotics, Antineoplastic; ATP-Binding Cassette Transporters; Biological Transport; Cell Membrane; Daunorubicin; Dimerization; DNA; Drug Resistance, Multiple; Electrophoresis, Polyacrylamide Gel; Ethidium; Fluoresceins; Fluorescent Dyes; Lactococcus lactis; Protein Binding; RNA; Time Factors; Up-Regulation

2004
Celastraceae sesquiterpenes as a new class of modulators that bind specifically to human P-glycoprotein and reverse cellular multidrug resistance.
    Cancer research, 2004, Oct-01, Volume: 64, Issue:19

    Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Azides; Benzimidazoles; Binding, Competitive; Celastraceae; Cell Membrane; Daunorubicin; Dihydropyridines; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Fluoresceins; Humans; Kinetics; Liposomes; Membrane Transport Modulators; Membrane Transport Proteins; Mice; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; NIH 3T3 Cells; Photoaffinity Labels; Protein Binding; Sesquiterpenes; Substrate Specificity; Vinblastine

2004
Effects of daunorubicin, mitomycin C, azathioprine and cyclosporin A on human retinal pigmented epithelial, corneal endothelial and conjunctival cell lines.
    Graefe's archive for clinical and experimental ophthalmology = Albrecht von Graefes Archiv fur klinische und experimentelle Ophthalmologie, 2006, Volume: 244, Issue:3

    Topics: Antimetabolites; Azathioprine; Cell Count; Cell Line; Cell Proliferation; Conjunctiva; Cyclosporine; Daunorubicin; Endothelium, Corneal; Epithelial Cells; Fluoresceins; Humans; Immunosuppressive Agents; Mitomycin; Pigment Epithelium of Eye; Propidium

2006
Schisandrin B: a dual inhibitor of P-glycoprotein and multidrug resistance-associated protein 1.
    Cancer letters, 2007, Feb-08, Volume: 246, Issue:1-2

    Topics: Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclooctanes; Daunorubicin; Dose-Response Relationship, Drug; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Fluoresceins; Gene Expression Regulation, Neoplastic; HL-60 Cells; Humans; Lignans; Molecular Structure; Multidrug Resistance-Associated Proteins; Polycyclic Compounds; Probenecid; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

2007
Complete inhibition of P-glycoprotein by simultaneous treatment with a distinct class of modulators and the UIC2 monoclonal antibody.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 320, Issue:1

    Topics: Animals; Antibodies, Monoclonal; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporine; Cyclosporins; Daunorubicin; Fluoresceins; Humans; Mice; NIH 3T3 Cells; Vinblastine

2007
Inhibition of P-glycoprotein and multidrug resistance protein 1 by dietary phytochemicals.
    Cancer chemotherapy and pharmacology, 2008, Volume: 62, Issue:5

    Topics: Adenosine Triphosphatases; Antibiotics, Antineoplastic; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Daunorubicin; Diet; Doxorubicin; Drug Resistance, Neoplasm; Flavonoids; Fluoresceins; Glycyrrhetinic Acid; Humans; KB Cells; Plants; Vinblastine

2008
Effects of chemopreventive citrus phytochemicals on human P-glycoprotein and multidrug resistance protein 1.
    European journal of pharmacology, 2008, Dec-14, Volume: 600, Issue:1-3

    Topics: Adenosine Triphosphatases; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Citrus; Daunorubicin; Fluoresceins; Food-Drug Interactions; Humans; KB Cells

2008
Effects of Curcuma spp. on P-glycoprotein function.
    Phytomedicine : international journal of phytotherapy and phytopharmacology, 2010, Volume: 17, Issue:7

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Caco-2 Cells; Cell Line; Curcuma; Curcumin; Daunorubicin; Dose-Response Relationship, Drug; Drug Resistance; Fluoresceins; Herb-Drug Interactions; Humans; Plant Extracts; Rhodamines; Swine

2010
Quercetin as a potential modulator of P-glycoprotein expression and function in cells of human pancreatic carcinoma line resistant to daunorubicin.
    Molecules (Basel, Switzerland), 2010, Feb-09, Volume: 15, Issue:2

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Cell Death; Cell Line, Tumor; Cell Membrane; Daunorubicin; Drug Resistance, Neoplasm; Fluoresceins; Gene Expression Regulation, Neoplastic; Humans; Pancreatic Neoplasms; Quercetin

2010
Pyrrolopyrimidine Derivatives as Novel Inhibitors of Multidrug Resistance-Associated Protein 1 (MRP1, ABCC1).
    Journal of medicinal chemistry, 2016, Apr-14, Volume: 59, Issue:7

    Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Cell Line, Tumor; Chlorophyll; Daunorubicin; Dogs; Doxorubicin; Drug Evaluation, Preclinical; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Fluoresceins; Humans; Inhibitory Concentration 50; Madin Darby Canine Kidney Cells; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pyridines; Pyrroles; Structure-Activity Relationship

2016
Pyrrolopyrimidine derivatives and purine analogs as novel activators of Multidrug Resistance-associated Protein 1 (MRP1, ABCC1).
    Biochimica et biophysica acta. Biomembranes, 2017, Volume: 1859, Issue:1

    Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily G, Member 2; Cell Line, Tumor; Daunorubicin; Dogs; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Fluoresceins; Fluorescent Dyes; Gene Expression; Humans; Kinetics; Madin Darby Canine Kidney Cells; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Purines; Pyrimidines; Pyrroles; Structure-Activity Relationship

2017
Identification of Thienopyrimidine Scaffold as an Inhibitor of the ABC Transport Protein ABCC1 (MRP1) and Related Transporters Using a Combined Virtual Screening Approach.
    Journal of medicinal chemistry, 2019, 05-09, Volume: 62, Issue:9

    Topics: ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily G, Member 2; Cell Line, Tumor; Chlorophyll; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Fluoresceins; Humans; Irinotecan; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pyrimidines; Small Molecule Libraries; Thiophenes

2019