Page last updated: 2024-08-21

erythromycin and em 201

erythromycin has been researched along with em 201 in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19901 (9.09)18.7374
1990's3 (27.27)18.2507
2000's6 (54.55)29.6817
2010's1 (9.09)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Inatomi, N; Itoh, Z; Marui, S; Omura, S; Sunazuka, T; Toyoda, H; Tsuzuki, K1
Edwards, CM; Faghih, R; Freiberg, L; Klein, LL; Lartey, PA; Marsh, K; Nellans, HN; Petersen, A; Plattner, JJ; Quigley, S1
Burgeon, E; Carreras, C; Depoortere, I; Liu, Y; Peeters, TL; Perret, J; Robberecht, P; Thielemans, L; Thijs, T1
Depoortere, I; Peeters, TL1
Matsushima, K; Nagatake, T; Oishi, K; Omura, T; Yoshimine, H1
Roberts, JJ; Shapiro, BL; Steinmetz, WE1
Akagawa, K; Iwata, S; Omura, T; Sunazuka, T1
Akagawa, K; Omura, T; Osawa, M; Sawai, T; Sunazuka, T1
Hanaki, H; Hirose, T; Nagai, K; Omura, S; Sharpless, KB; Sugawara, A; Sunazuka, T; Yamaguchi, Y1
Akagawa, KS; Iwamoto, A; Komuro, I; Omura, S; Sunazuka, T; Yokota, Y1
Hamasaki, Y; Hatamochi, A; Kitamura, Y; Namikawa, H; Omura, S; Sunazuka, T; Suzuki, T; Yamazaki, S1

Other Studies

11 other study(ies) available for erythromycin and em 201

ArticleYear
Macrolides with gastrointestinal motor stimulating activity.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:11

    Topics: Animals; Erythromycin; Gastrointestinal Motility; In Vitro Techniques; Muscle Contraction; Rabbits

1987
Synthesis of 4"-deoxy motilides: identification of a potent and orally active prokinetic drug candidate.
    Journal of medicinal chemistry, 1995, May-12, Volume: 38, Issue:10

    Topics: Administration, Oral; Animals; Biological Availability; Dogs; Erythromycin; Female; Gastrointestinal Motility; In Vitro Techniques; Male; Muscle, Smooth; Rabbits

1995
Desensitization of the human motilin receptor by motilides.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 313, Issue:3

    Topics: Animals; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Erythromycin; Humans; Muscle Contraction; Radioligand Assay; Receptors, Gastrointestinal Hormone; Receptors, Neuropeptide; Structure-Activity Relationship

2005
Transduction mechanism of motilin and motilides in rabbit duodenal smooth muscle.
    Regulatory peptides, 1995, Feb-14, Volume: 55, Issue:3

    Topics: Adenylyl Cyclases; Animals; Carbachol; Duodenum; Erythromycin; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Inositol; Inositol Phosphates; Motilin; Muscle, Smooth; Rabbits; Receptors, Gastrointestinal Hormone; Receptors, Neuropeptide; Signal Transduction; Tritium

1995
[Inhibition of neutrophil-derived IL-8 production caused by EM (erythromycin) 201 derivative: modification of the activities by the 5-position desosamine side chain].
    The Japanese journal of antibiotics, 1998, Volume: 51 Suppl A

    Topics: Anti-Bacterial Agents; Cells, Cultured; Clarithromycin; Erythromycin; Humans; Interleukin-8; Neutrophils; Structure-Activity Relationship

1998
The structure of erythromycin enol ether as a model for its activity as a motilide.
    Journal of medicinal chemistry, 2002, Oct-24, Volume: 45, Issue:22

    Topics: Erythromycin; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Mimicry; Motilin; Protein Structure, Secondary

2002
[Effects of EM201, an in vivo metabolite of erythromycin, on differentiation and functions of dendrite cells].
    The Japanese journal of antibiotics, 2004, Volume: 57 Suppl A

    Topics: Anti-Bacterial Agents; Cell Differentiation; Cells, Cultured; Dendritic Cells; Erythromycin; Humans; Interleukin-10; Interleukin-12; Monocytes

2004
[Effect of EM201, an in vivo metabolite of erythromycin (EM), on signal transduction of IL-2 receptor].
    The Japanese journal of antibiotics, 2004, Volume: 57 Suppl A

    Topics: Cells, Cultured; Chromones; Erythromycin; Flavonoids; Humans; Monocytes; Morpholines; Receptors, Interleukin-2; Signal Transduction; Sirolimus

2004
Design and synthesis via click chemistry of 8,9-anhydroerythromycin A 6,9-hemiketal analogues with anti-MRSA and -VRE activity.
    Bioorganic & medicinal chemistry letters, 2007, Nov-15, Volume: 17, Issue:22

    Topics: Anti-Bacterial Agents; Catalysis; Copper; Drug Design; Enterococcus; Erythromycin; Methicillin Resistance; Microbial Sensitivity Tests; Molecular Structure; Staphylococcus aureus; Vancomycin Resistance

2007
Erythromycin derivatives inhibit HIV-1 replication in macrophages through modulation of MAPK activity to induce small isoforms of C/EBPbeta.
    Proceedings of the National Academy of Sciences of the United States of America, 2008, Aug-26, Volume: 105, Issue:34

    Topics: CCAAT-Enhancer-Binding Protein-beta; CD4-Positive T-Lymphocytes; Cells, Cultured; Coculture Techniques; Disease Susceptibility; Erythromycin; HIV-1; Humans; Macrophages; Mitogen-Activated Protein Kinases; Protein Isoforms; Proto-Oncogene Proteins c-hck; Virus Replication

2008
Effect of erythromycin A and its new derivative EM201 on type I collagen production by cultured dermal fibroblasts.
    Archives of dermatological research, 2010, Volume: 302, Issue:5

    Topics: Adolescent; Adult; Cell Proliferation; Cells, Cultured; Collagen Type I; Dermis; Erythromycin; Female; Fibroblasts; Humans; Infant; Male; Skin Aging; Transgenes

2010