ersentilide has been researched along with sotalol in 3 studies
Studies (ersentilide) | Trials (ersentilide) | Recent Studies (post-2010) (ersentilide) | Studies (sotalol) | Trials (sotalol) | Recent Studies (post-2010) (sotalol) |
---|---|---|---|---|---|
9 | 0 | 0 | 2,196 | 346 | 291 |
Protein | Taxonomy | ersentilide (IC50) | sotalol (IC50) |
---|---|---|---|
Beta-2 adrenergic receptor | Homo sapiens (human) | 3.8169 | |
Beta-1 adrenergic receptor | Homo sapiens (human) | 7.1087 | |
Beta-3 adrenergic receptor | Homo sapiens (human) | 7.2 | |
Beta-2 adrenergic receptor | Canis lupus familiaris (dog) | 5.0667 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 3 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Davey, DD; Gomez, RP; Lind, JM; Lis, R; Marisca, AJ; Morgan, TK; Phillips, GB; Sullivan, ME | 1 |
Benz, I; Kohlhardt, M | 2 |
3 other study(ies) available for ersentilide and sotalol
Article | Year |
---|---|
Synthesis of novel (aryloxy)propanolamines and related compounds possessing both class II and class III antiarrhythmic activity.
Topics: Action Potentials; Adrenergic beta-Antagonists; Animals; Anti-Arrhythmia Agents; Blood Pressure; Chemical Phenomena; Chemistry, Physical; Dogs; Drug Design; Epinephrine; Heart Rate; In Vitro Techniques; Propanolamines; Purkinje Fibers; Receptors, Adrenergic, beta | 1990 |
Distinct modes of blockade in cardiac ATP-sensitive K+ channels suggest multiple targets for inhibitory drug molecules.
Topics: Adenosine Triphosphate; Animals; Animals, Newborn; Binding Sites; Cells, Cultured; Glyburide; Imidazoles; Kinetics; Membrane Potentials; Myocardium; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Propanolamines; Rats; Sotalol; Verapamil | 1994 |
Characterization of the sensitivity of cardiac outwardly-rectifying K+ channels to class III antiarrhythmics: the influence of inhibitory sulfonamide derivatives.
Topics: Animals; Animals, Newborn; Anti-Arrhythmia Agents; Cells, Cultured; Glyburide; Heart; Imidazoles; Kinetics; Lethal Dose 50; Myocardium; Patch-Clamp Techniques; Potassium Channels; Propanolamines; Rats; Sotalol; Sulfonamides; Up-Regulation | 1995 |