Page last updated: 2024-09-03

ersentilide and glyburide

ersentilide has been researched along with glyburide in 2 studies

Compound Research Comparison

Studies
(ersentilide)
Trials
(ersentilide)
Recent Studies (post-2010)
(ersentilide)
Studies
(glyburide)
Trials
(glyburide)
Recent Studies (post-2010) (glyburide)
9006,5546201,344

Protein Interaction Comparison

ProteinTaxonomyersentilide (IC50)glyburide (IC50)
ATP-binding cassette sub-family C member 9Homo sapiens (human)0.22
Bile salt export pumpRattus norvegicus (Norway rat)5.7
Bile salt export pumpHomo sapiens (human)5.5333
Cytochrome P450 2C9 Homo sapiens (human)1.602
ATP-binding cassette sub-family C member 8Homo sapiens (human)0.0043
ATP-sensitive inward rectifier potassium channel 11Homo sapiens (human)0.1121
NACHT, LRR and PYD domains-containing protein 3 Mus musculus (house mouse)10
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)1.8

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Benz, I; Kohlhardt, M2

Other Studies

2 other study(ies) available for ersentilide and glyburide

ArticleYear
Distinct modes of blockade in cardiac ATP-sensitive K+ channels suggest multiple targets for inhibitory drug molecules.
    The Journal of membrane biology, 1994, Volume: 142, Issue:3

    Topics: Adenosine Triphosphate; Animals; Animals, Newborn; Binding Sites; Cells, Cultured; Glyburide; Imidazoles; Kinetics; Membrane Potentials; Myocardium; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Propanolamines; Rats; Sotalol; Verapamil

1994
Characterization of the sensitivity of cardiac outwardly-rectifying K+ channels to class III antiarrhythmics: the influence of inhibitory sulfonamide derivatives.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:3

    Topics: Animals; Animals, Newborn; Anti-Arrhythmia Agents; Cells, Cultured; Glyburide; Heart; Imidazoles; Kinetics; Lethal Dose 50; Myocardium; Patch-Clamp Techniques; Potassium Channels; Propanolamines; Rats; Sotalol; Sulfonamides; Up-Regulation

1995