Page last updated: 2024-09-05

erlotinib and sb-590885

erlotinib has been researched along with sb-590885 in 2 studies

Compound Research Comparison

Studies
(erlotinib)
Trials
(erlotinib)
Recent Studies (post-2010)
(erlotinib)
Studies
(sb-590885)
Trials
(sb-590885)
Recent Studies (post-2010) (sb-590885)
2210180906
22101801008

Protein Interaction Comparison

ProteinTaxonomyerlotinib (IC50)sb-590885 (IC50)
Serine/threonine-protein kinase B-rafHomo sapiens (human)0.1934

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Li, QS; Sun, S; Tang, JF; Wang, XL; Yang, YS; Zhang, F; Zhang, YB; Zhu, HL1
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1

Other Studies

2 other study(ies) available for erlotinib and sb-590885

ArticleYear
Design, modification and 3D QSAR studies of novel 2,3-dihydrobenzo[b][1,4]dioxin-containing 4,5-dihydro-1H-pyrazole derivatives as inhibitors of B-Raf kinase.
    Bioorganic & medicinal chemistry, 2012, Oct-15, Volume: 20, Issue:20

    Topics: Binding Sites; Cell Line, Tumor; Cell Proliferation; Dioxanes; Dioxins; Drug Design; Erlotinib Hydrochloride; Humans; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins B-raf; Pyrazoles; Quantitative Structure-Activity Relationship; Quinazolines; Thermodynamics

2012
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013