Page last updated: 2024-09-05

erlotinib and nvp-aew541

erlotinib has been researched along with nvp-aew541 in 1 studies

Compound Research Comparison

Studies
(erlotinib)
Trials
(erlotinib)
Recent Studies (post-2010)
(erlotinib)
Studies
(nvp-aew541)
Trials
(nvp-aew541)
Recent Studies (post-2010) (nvp-aew541)
221018095061

Protein Interaction Comparison

ProteinTaxonomyerlotinib (IC50)nvp-aew541 (IC50)
3-phosphoinositide-dependent protein kinase 1Homo sapiens (human)8.9
Epidermal growth factor receptorHomo sapiens (human)5.2
Insulin receptorHomo sapiens (human)0.7885
Tyrosine-protein kinase LckHomo sapiens (human)5.6
Tyrosine-protein kinase LynHomo sapiens (human)1.4
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)3.3
Insulin-like growth factor 1 receptorHomo sapiens (human)0.0534
Mast/stem cell growth factor receptor KitHomo sapiens (human)6.3
Fibroblast growth factor receptor 1Homo sapiens (human)4.3
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)4
Platelet-derived growth factor receptor alphaHomo sapiens (human)0.8
Fibroblast growth factor receptor 2Homo sapiens (human)2.7
Fibroblast growth factor receptor 4Homo sapiens (human)5
Vascular endothelial growth factor receptor 2Homo sapiens (human)7.1
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)1.4
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform Homo sapiens (human)3.2
Activin receptor type-1Homo sapiens (human)2.9
Tyrosine-protein kinase BTKHomo sapiens (human)7.6
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)0.13
Receptor tyrosine-protein kinase erbB-4Homo sapiens (human)1.7

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bantscheff, M; Bergamini, G; Gohlke, B; Gupta, V; Handa, H; Heinzlmeir, S; Helm, D; Klaeger, S; Kuster, B; Médard, G; Perrin, J; Preissner, R; Qiao, H; Savitski, MM1

Other Studies

1 other study(ies) available for erlotinib and nvp-aew541

ArticleYear
Chemical Proteomics Reveals Ferrochelatase as a Common Off-target of Kinase Inhibitors.
    ACS chemical biology, 2016, 05-20, Volume: 11, Issue:5

    Topics: Benzocycloheptenes; Cell Line, Tumor; Ferrochelatase; Heme; Humans; Imidazoles; Indoles; Molecular Docking Simulation; Protein Binding; Protein Kinase Inhibitors; Proteomics; Pyrazines; Pyridines; Quinolines; Sulfonamides; Vemurafenib

2016