Page last updated: 2024-09-05

erlotinib and jq1 compound

erlotinib has been researched along with jq1 compound in 3 studies

Compound Research Comparison

Studies
(erlotinib)
Trials
(erlotinib)
Recent Studies (post-2010)
(erlotinib)
Studies
(jq1 compound)
Trials
(jq1 compound)
Recent Studies (post-2010) (jq1 compound)
22101801090105

Protein Interaction Comparison

ProteinTaxonomyerlotinib (IC50)jq1 compound (IC50)
Histone deacetylase 3Homo sapiens (human)0.291
Bromodomain-containing protein 4Homo sapiens (human)0.142
Cytochrome P450 1A2Homo sapiens (human)0.82
Cytochrome P450 3A4Homo sapiens (human)0.0527
Bromodomain-containing protein 2Homo sapiens (human)0.0959
Histone deacetylase 4Homo sapiens (human)0.291
Histone deacetylase 1Homo sapiens (human)0.291
Bromodomain-containing protein 3Homo sapiens (human)0.0573
Bromodomain testis-specific proteinHomo sapiens (human)0.1902
Histone deacetylase 7Homo sapiens (human)0.291
Histone deacetylase 2Homo sapiens (human)0.291
CREB-binding proteinHomo sapiens (human)9.573
Polyamine deacetylase HDAC10Homo sapiens (human)0.291
Histone deacetylase 11 Homo sapiens (human)0.291
Histone deacetylase 8Homo sapiens (human)0.291
Histone deacetylase 6Homo sapiens (human)0.291
Histone deacetylase 9Homo sapiens (human)0.291
Histone deacetylase 5Homo sapiens (human)0.291

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (33.33)24.3611
2020's2 (66.67)2.80

Authors

AuthorsStudies
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1
Duan, G; Liu, T; Wan, Y; Xia, C; Xiao, Y1
Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M1

Reviews

1 review(s) available for erlotinib and jq1 compound

ArticleYear
Dual-Target Inhibitors Based on HDACs: Novel Antitumor Agents for Cancer Therapy.
    Journal of medicinal chemistry, 2020, 09-10, Volume: 63, Issue:17

    Topics: Antineoplastic Agents; DNA Damage; Histone Deacetylase Inhibitors; Histone Deacetylases; Humans; Neoplasms; Protein Kinases; Proteins; Structure-Activity Relationship; Topoisomerase Inhibitors

2020

Other Studies

2 other study(ies) available for erlotinib and jq1 compound

ArticleYear
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
    Disease models & mechanisms, 2023, 03-01, Volume: 16, Issue:3

    Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries

2023