Page last updated: 2024-09-05

erlotinib and cb-839

erlotinib has been researched along with cb-839 in 2 studies

Compound Research Comparison

Studies
(erlotinib)
Trials
(erlotinib)
Recent Studies (post-2010)
(erlotinib)
Studies
(cb-839)
Trials
(cb-839)
Recent Studies (post-2010) (cb-839)
221018071271

Protein Interaction Comparison

ProteinTaxonomyerlotinib (IC50)cb-839 (IC50)
Glutaminase kidney isoform, mitochondrialMus musculus (house mouse)0.02
Glutaminase kidney isoform, mitochondrialHomo sapiens (human)0.2025

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (50.00)24.3611
2020's1 (50.00)2.80

Authors

AuthorsStudies
Bian, J; Li, L; Li, Z; Meng, Y; Wang, J; Xu, P; Xu, X1
Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M1

Other Studies

2 other study(ies) available for erlotinib and cb-839

ArticleYear
Overview of the Development of Glutaminase Inhibitors: Achievements and Future Directions.
    Journal of medicinal chemistry, 2019, 02-14, Volume: 62, Issue:3

    Topics: Animals; Benzophenanthridines; Benzoquinones; Catalytic Domain; Cell Line, Tumor; Drug Discovery; Enzyme Inhibitors; Glutaminase; Humans; Mice; Molecular Docking Simulation; Protein Binding; Sulfides; Thiadiazoles; Thiazolidinediones

2019
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
    Disease models & mechanisms, 2023, 03-01, Volume: 16, Issue:3

    Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries

2023