Page last updated: 2024-09-05

eptapirone and sibutramine

eptapirone has been researched along with sibutramine in 1 studies

Compound Research Comparison

Studies
(eptapirone)
Trials
(eptapirone)
Recent Studies (post-2010)
(eptapirone)
Studies
(sibutramine)
Trials
(sibutramine)
Recent Studies (post-2010) (sibutramine)
521967218204

Protein Interaction Comparison

ProteinTaxonomyeptapirone (IC50)sibutramine (IC50)
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)5.665
Alpha-2B adrenergic receptorHomo sapiens (human)2.39
Sodium-dependent noradrenaline transporter Homo sapiens (human)5.665
Sodium-dependent serotonin transporterHomo sapiens (human)2.085
Sodium-dependent dopamine transporter Homo sapiens (human)0.632

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Babbs, AJ; Chatfield, RE; Krülle, TM; McCormack, JG; Provost, D; Thomas, GH; Widdowson, PS1

Other Studies

1 other study(ies) available for eptapirone and sibutramine

ArticleYear
5-HT(1A) activation counteracts cardiovascular but not hypophagic effects of sibutramine in rats.
    Obesity (Silver Spring, Md.), 2009, Volume: 17, Issue:3

    Topics: Adrenergic Uptake Inhibitors; Animals; Appetite Depressants; Blood Pressure; Cyclobutanes; Dose-Response Relationship, Drug; Eating; Fluoxetine; Heart Rate; Male; Models, Animal; Morpholines; Norepinephrine; Pyrimidines; Rats; Rats, Sprague-Dawley; Reboxetine; Receptor, Serotonin, 5-HT1A; Serotonin 5-HT1 Receptor Agonists; Triazines

2009