Page last updated: 2024-09-05

eptapirone and buspirone

eptapirone has been researched along with buspirone in 1 studies

Compound Research Comparison

Studies
(eptapirone)
Trials
(eptapirone)
Recent Studies (post-2010)
(eptapirone)
Studies
(buspirone)
Trials
(buspirone)
Recent Studies (post-2010) (buspirone)
5212,096351382

Protein Interaction Comparison

ProteinTaxonomyeptapirone (IC50)buspirone (IC50)
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.025
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)1.75
Angiotensin-converting enzyme Homo sapiens (human)0.024
D(2) dopamine receptorHomo sapiens (human)0.323
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)2.125
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)4.16
DRattus norvegicus (Norway rat)0.12
D(3) dopamine receptorRattus norvegicus (Norway rat)0.12
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0266
D(2) dopamine receptorBos taurus (cattle)4
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)4.16
Alpha-1D adrenergic receptorHomo sapiens (human)1.077
D(1B) dopamine receptorRattus norvegicus (Norway rat)0.12
5-hydroxytryptamine receptor 2AHomo sapiens (human)2.286
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.016
D(4) dopamine receptorRattus norvegicus (Norway rat)0.12
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)2.125
D(3) dopamine receptorHomo sapiens (human)0.044
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.75
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)4.16
D(2) dopamine receptorRattus norvegicus (Norway rat)0.2055
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)3.9811
Alpha-2A adrenergic receptorBos taurus (cattle)0.025
Multidrug and toxin extrusion protein 1Homo sapiens (human)1.7
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.2666
Lysosomal alpha-glucosidaseBos taurus (cattle)0.03

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Adrover, M; Bailey, JE; Nash, J; Nutt, DJ; Rich, AS; Tournoux, A; Wilson, SJ1

Trials

1 trial(s) available for eptapirone and buspirone

ArticleYear
The use of sleep measures to compare a new 5HT1A agonist with buspirone in humans.
    Journal of psychopharmacology (Oxford, England), 2005, Volume: 19, Issue:6

    Topics: Adolescent; Adult; Arousal; Attention; Buspirone; Cross-Over Studies; Double-Blind Method; Drug Administration Schedule; Humans; Male; Polysomnography; Pyrimidines; Reaction Time; Serotonin 5-HT1 Receptor Agonists; Serotonin Receptor Agonists; Sleep Stages; Sleep, REM; Triazines; Wakefulness

2005
chemdatabank.com