epibatidine and varenicline

epibatidine has been researched along with varenicline in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (10.00)29.6817
2010's8 (80.00)24.3611
2020's1 (10.00)2.80

Authors

AuthorsStudies
Brooks, EA; Jutkiewicz, EM; Kynaston, AD; Rice, KC; Woods, JH1
Blythe, EE; Dougherty, DA; Lester, HA; Van Arnam, EB1
Arias, HR; Feuerbach, D; Jozwiak, K; Kaczor, AA; Poso, A; Targowska-Duda, K1
Carroll, FI; Cunningham, CS; Javors, MA; McMahon, LR; Moerke, MJ1
de Moura, FB; McMahon, LR2
Bergman, J; de Moura, FB1
Brieaddy, LE; Burgess, JP; Damaj, MI; Ivy Carroll, F; Lee, JR; Ma, W; Martin, BR; Navarro, HA; Yokota, Y1
Bertrand, D; Bertrand, S; Bréthous, L; Garcia-Delgado, N; Reymond, JL; Schwartz, J1
Bartkowiak, JM; Carroll, FI; Castro, AH; Damaj, MI; Luetje, CW; Mascarella, SW; Navarro, HA; Ondachi, PW1

Other Studies

10 other study(ies) available for epibatidine and varenicline

ArticleYear
Patterns of nicotinic receptor antagonism: nicotine discrimination studies.
    The Journal of pharmacology and experimental therapeutics, 2011, Volume: 339, Issue:1

    Topics: Animals; Benzazepines; Bridged Bicyclo Compounds, Heterocyclic; Cytosine; Data Interpretation, Statistical; Dihydro-beta-Erythroidine; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Male; Mecamylamine; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Pyridines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Varenicline

2011
An unusual pattern of ligand-receptor interactions for the α7 nicotinic acetylcholine receptor, with implications for the binding of varenicline.
    Molecular pharmacology, 2013, Volume: 84, Issue:2

    Topics: Acetylcholine; alpha7 Nicotinic Acetylcholine Receptor; Animals; Benzazepines; Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Humans; Hydrogen Bonding; Ligands; Models, Molecular; Nicotinic Agonists; Oocytes; Pyridines; Quinoxalines; Rats; Varenicline; Xenopus laevis

2013
Pharmacological and molecular studies on the interaction of varenicline with different nicotinic acetylcholine receptor subtypes. Potential mechanism underlying partial agonism at human α4β2 and α3β4 subtypes.
    Biochimica et biophysica acta, 2015, Volume: 1848, Issue:2

    Topics: Allosteric Regulation; Allosteric Site; Animals; Benzazepines; Bridged Bicyclo Compounds, Heterocyclic; Calcium; CHO Cells; Cricetulus; Gene Expression; HEK293 Cells; Humans; Hydrogen Bonding; Molecular Docking Simulation; Nicotinic Agonists; Protein Binding; Protein Isoforms; Protein Structure, Secondary; Pyridines; Quinoxalines; Receptors, Nicotinic; Structural Homology, Protein; Torpedo; Transgenes; Varenicline

2015
Attenuated nicotine-like effects of varenicline but not other nicotinic ACh receptor agonists in monkeys receiving nicotine daily.
    British journal of pharmacology, 2016, Volume: 173, Issue:24

    Topics: Animals; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Female; Macaca mulatta; Male; Nicotine; Nicotinic Agonists; Pyridines; Receptors, Nicotinic; Structure-Activity Relationship; Varenicline

2016
The contribution of α4β2 and non-α4β2 nicotinic acetylcholine receptors to the discriminative stimulus effects of nicotine and varenicline in mice.
    Psychopharmacology, 2017, Volume: 234, Issue:5

    Topics: Aconitine; Alkaloids; alpha7 Nicotinic Acetylcholine Receptor; Animals; Azocines; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cocaine; Dihydro-beta-Erythroidine; Discrimination, Psychological; Dopamine Uptake Inhibitors; Hypnotics and Sedatives; Ibogaine; Male; Mecamylamine; Mice; Mice, Inbred C57BL; Midazolam; Nerve Tissue Proteins; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Pyridines; Quinolizines; Receptors, Nicotinic; Varenicline

2017
Differential cross-tolerance to the effects of nicotinic acetylcholine receptor drugs in C57BL/6J mice following chronic varenicline.
    Behavioural pharmacology, 2019, Volume: 30, Issue:5

    Topics: Alkaloids; Animals; Azocines; Bridged Bicyclo Compounds, Heterocyclic; Cocaine; Conditioning, Operant; Drug Tolerance; Female; Male; Mice; Mice, Inbred C57BL; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Pyridines; Quinolizines; Receptors, Nicotinic; Reinforcement, Psychology; Smoking Cessation; Varenicline

2019
Enhancement of Opioid Antinociception by Nicotinic Ligands.
    The Journal of pharmacology and experimental therapeutics, 2021, Volume: 377, Issue:1

    Topics: Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Bridged Bicyclo Compounds, Heterocyclic; Conditioning, Operant; Drug Synergism; Fentanyl; Male; Nalbuphine; Nicotinic Agonists; Nociception; Pyridines; Saimiri; Varenicline

2021
Synthesis, nicotinic acetylcholine receptor binding, and pharmacological properties of 3'-(substituted phenyl)deschloroepibatidine analogs.
    Bioorganic & medicinal chemistry, 2008, Jan-15, Volume: 16, Issue:2

    Topics: Analgesics; Animals; Body Temperature; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Disease Models, Animal; Dose-Response Relationship, Drug; Mice; Molecular Structure; Nicotinic Antagonists; Pain; Protein Binding; Pyridines; Radioligand Assay; Receptors, Nicotinic; Structure-Activity Relationship

2008
Synthesis and nicotinic receptor activity of chemical space analogues of N-(3R)-1-azabicyclo[2.2.2]oct-3-yl-4-chlorobenzamide (PNU-282,987) and 1,4-diazabicyclo[3.2.2]nonane-4-carboxylic acid 4-bromophenyl ester (SSR180711).
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Allosteric Regulation; Animals; Benzamides; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Databases, Factual; Female; Humans; Models, Molecular; Nicotinic Agonists; Nicotinic Antagonists; Oocytes; Patch-Clamp Techniques; Receptors, Nicotinic; Stereoisomerism; Structure-Activity Relationship; Xenopus

2012
Synthesis, nicotinic acetylcholine receptor binding, and antinociceptive properties of 2'-fluoro-3'-(substituted pyridinyl)-7-deschloroepibatidine analogues.
    Journal of medicinal chemistry, 2014, Feb-13, Volume: 57, Issue:3

    Topics: Analgesics; Animals; Body Temperature; Bridged Bicyclo Compounds, Heterocyclic; Contraindications; Female; Male; Mice; Nicotinic Agonists; Nicotinic Antagonists; Oocytes; Pain; Patch-Clamp Techniques; Pyridines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Structure-Activity Relationship; Xenopus

2014