epibatidine and piperidines

epibatidine has been researched along with piperidines in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (33.33)18.2507
2000's2 (22.22)29.6817
2010's4 (44.44)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hezký, P; Krejcí, I; Proska, J; Rádl, S1
Ellis, JL; Gonzalez, J; Harman, D; Liu, R; Shen, TY; Spera, ML; Wypij, DM; Zuo, F1
Gillberg, PG; Nordberg, A; Sihver, W; Svensson, AL1
Reid, RT; Sabbagh, MN1
Arias, HR; Bouzat, C; Feuerbach, D; Gumilar, F; Jozwiak, K; Moaddel, R; Rosenberg, A; Targowska-Duda, KM; Wainer, IW1
Allen, JD; Bergmeier, SC; Bonnell, AB; Boyd, RT; González-Cestari, TF; Henderson, BJ; Li, C; McKay, DB; Orac, CM; Pavlovicz, RE; Zhu, MX1
Nakamura, K; Shimizu, T; Tanaka, K; Taniuchi, K; Yokotani, K1
Higashi, Y; Nakamura, K; Saito, M; Shimizu, S; Shimizu, T; Tanaka, K; Taniuchi, K; Ueba, T; Yawata, T; Yuri, K1
Dick, ALW; Duncan, JR; Gibbs, S; Giles, E; Lawrence, AJ; Pooters, T; Qama, A1

Other Studies

9 other study(ies) available for epibatidine and piperidines

ArticleYear
Analgetically active substances derived from structures of anpirtoline and epibatidine.
    General physiology and biophysics, 1998, Volume: 17 Suppl 1

    Topics: Analgesics, Non-Narcotic; Animals; Bridged Bicyclo Compounds, Heterocyclic; Drug Design; Mice; Molecular Conformation; Piperidines; Pyridines; Structure-Activity Relationship; Thermodynamics

1998
Development of muscarinic analgesics derived from epibatidine: role of the M4 receptor subtype.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 288, Issue:3

    Topics: Alkaloids; Analgesics, Non-Narcotic; Animals; Body Temperature; Bridged Bicyclo Compounds, Heterocyclic; Female; Furans; Mice; Muscarinic Agonists; Naphthalenes; Oxadiazoles; Piperidines; Pyridines; Receptor, Muscarinic M4; Receptors, Muscarinic; Salivation

1999
Autoradiographic comparison of [3H](-)nicotine, [3H]cytisine and [3H]epibatidine binding in relation to vesicular acetylcholine transport sites in the temporal cortex in Alzheimer's disease.
    Neuroscience, 1999, Volume: 94, Issue:3

    Topics: Acetylcholine; Age Factors; Aged; Aged, 80 and over; Alkaloids; Alzheimer Disease; Autoradiography; Azocines; Bridged Bicyclo Compounds, Heterocyclic; Carrier Proteins; Female; Humans; Male; Membrane Transport Proteins; Middle Aged; Nicotine; Piperidines; Pyridines; Quinolizines; Reference Values; Temporal Lobe; Tritium; Vesicular Acetylcholine Transport Proteins; Vesicular Transport Proteins

1999
Effects of donepezil treatment on rat nicotinic acetylcholine receptor levels in vivo and in vitro.
    Journal of Alzheimer's disease : JAD, 2003, Volume: 5, Issue:6

    Topics: Aconitine; Animals; Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Cholinesterase Inhibitors; Donepezil; Drug Administration Schedule; Hippocampus; In Vitro Techniques; Indans; Male; Nicotinic Agonists; Nicotinic Antagonists; Pheochromocytoma; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic

2003
Interaction of bupropion with muscle-type nicotinic acetylcholine receptors in different conformational states.
    Biochemistry, 2009, Jun-02, Volume: 48, Issue:21

    Topics: Animals; Binding, Competitive; Biological Transport; Bridged Bicyclo Compounds, Heterocyclic; Bupropion; Calcium; Cell Line; Drug Discovery; Electric Conductivity; Humans; Imipramine; Immobilized Proteins; Ion Channel Gating; Kinetics; Mice; Models, Molecular; Muscles; Nicotinic Antagonists; Piperidines; Protein Binding; Protein Conformation; Pyridines; Receptors, Nicotinic; Thermodynamics; Torpedo

2009
Negative allosteric modulators that target human alpha4beta2 neuronal nicotinic receptors.
    The Journal of pharmacology and experimental therapeutics, 2010, Sep-01, Volume: 334, Issue:3

    Topics: Algorithms; Biphenyl Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Humans; Hydrogen Bonding; Models, Molecular; Mutagenesis, Site-Directed; Neurons; Nicotinic Agonists; Piperidines; Pyridines; Quantitative Structure-Activity Relationship; Receptors, Nicotinic; Structure-Activity Relationship

2010
Brain phospholipase C, diacylglycerol lipase and monoacylglycerol lipase are involved in (±)-epibatidine-induced activation of central adrenomedullary outflow in rats.
    European journal of pharmacology, 2012, Sep-15, Volume: 691, Issue:1-3

    Topics: Adrenal Medulla; Animals; Arachidonic Acids; Benzodioxoles; Brain; Bridged Bicyclo Compounds, Heterocyclic; Catecholamines; Cyclohexanones; Esterases; Estrenes; Lipoprotein Lipase; Male; Monoacylglycerol Lipases; Neurons; Nicotinic Agonists; Organophosphonates; Paraventricular Hypothalamic Nucleus; Piperidines; Pyridines; Pyrrolidinones; Rats; Rats, Wistar; Type C Phospholipases

2012
Possible inhibitory role of endogenous 2-arachidonoylglycerol as an endocannabinoid in (±)-epibatidine-induced activation of central adrenomedullary outflow in the rat.
    Neuropharmacology, 2015, Volume: 95

    Topics: Adrenal Medulla; Animals; Arachidonic Acids; Bridged Bicyclo Compounds, Heterocyclic; Catecholamines; Dose-Response Relationship, Drug; Endocannabinoids; Glycerides; Immunohistochemistry; Male; Neurons; Neurotransmitter Agents; Nicotinic Agonists; Paraventricular Hypothalamic Nucleus; Piperidines; Pyrazoles; Pyridines; Rats, Wistar; Receptor, Cannabinoid, CB1

2015
NMDA receptor binding is reduced within mesocorticolimbic regions following chronic inhalation of toluene in adolescent rats.
    Brain research, 2015, Oct-22, Volume: 1624

    Topics: Animals; Animals, Newborn; Autoradiography; Bridged Bicyclo Compounds, Heterocyclic; Excitatory Amino Acid Agents; Gene Expression; Limbic System; Male; Nicotinic Agonists; Piperidines; Protein Binding; Pyridines; Rats; Receptors, N-Methyl-D-Aspartate; RNA, Messenger; Solvents; Somatosensory Cortex; Toluene; Tritium

2015