Page last updated: 2024-09-05

enzastaurin and tanespimycin

enzastaurin has been researched along with tanespimycin in 1 studies

Compound Research Comparison

Studies
(enzastaurin)
Trials
(enzastaurin)
Recent Studies (post-2010)
(enzastaurin)
Studies
(tanespimycin)
Trials
(tanespimycin)
Recent Studies (post-2010) (tanespimycin)
188529992139496

Protein Interaction Comparison

ProteinTaxonomyenzastaurin (IC50)tanespimycin (IC50)
Corticotropin releasing hormone receptor 2Sus scrofa (pig)0.004
Lysine-specific demethylase 6BHomo sapiens (human)0.4
Lysine-specific demethylase 4BHomo sapiens (human)0.7
Tyrosine-protein kinase ABL1Homo sapiens (human)3
ATP-dependent molecular chaperone HSP82Saccharomyces cerevisiae S288C7.65
Receptor tyrosine-protein kinase erbB-2Homo sapiens (human)0.031
Heat shock protein HSP 90-alphaHomo sapiens (human)0.9391
Heat shock protein HSP 90-betaHomo sapiens (human)0.5124
Breakpoint cluster region proteinHomo sapiens (human)3
Lysine-specific demethylase 5AHomo sapiens (human)0.13
EndoplasminCanis lupus familiaris (dog)0.031
Heat shock protein 75 kDa, mitochondrialHomo sapiens (human)1.496
Putative heat shock protein HSP 90-alpha A4Homo sapiens (human)0.78
Lysine-specific demethylase 4CHomo sapiens (human)0.7

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Jane, EP; Pollack, IF1

Other Studies

1 other study(ies) available for enzastaurin and tanespimycin

ArticleYear
The heat shock protein antagonist 17-AAG potentiates the activity of enzastaurin against malignant human glioma cells.
    Cancer letters, 2008, Sep-08, Volume: 268, Issue:1

    Topics: Apoptosis; Benzoquinones; Caspase 3; Cell Line, Tumor; Cell Proliferation; Cell Survival; Cytochromes c; Down-Regulation; Drug Synergism; Glioma; HSP90 Heat-Shock Proteins; Humans; Indoles; Lactams, Macrocyclic; Oncogene Protein v-akt; Phosphorylation

2008