Page last updated: 2024-09-05

enzastaurin and sk&f 86002

enzastaurin has been researched along with sk&f 86002 in 1 studies

Compound Research Comparison

Studies
(enzastaurin)
Trials
(enzastaurin)
Recent Studies (post-2010)
(enzastaurin)
Studies
(sk&f 86002)
Trials
(sk&f 86002)
Recent Studies (post-2010) (sk&f 86002)
188529983413

Protein Interaction Comparison

ProteinTaxonomyenzastaurin (IC50)sk&f 86002 (IC50)
Mitogen-activated protein kinase 13Homo sapiens (human)3.8
Prostaglandin G/H synthase 1Ovis aries (sheep)5.4
Polyunsaturated fatty acid 5-lipoxygenaseRattus norvegicus (Norway rat)10
Mitogen-activated protein kinase 12Homo sapiens (human)3.8
Mitogen-activated protein kinase 11Homo sapiens (human)3.8
Mitogen-activated protein kinase 14Homo sapiens (human)2.1217

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1

Other Studies

1 other study(ies) available for enzastaurin and sk&f 86002

ArticleYear
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013