Page last updated: 2024-09-05

enzastaurin and rottlerin

enzastaurin has been researched along with rottlerin in 1 studies

Compound Research Comparison

Studies
(enzastaurin)
Trials
(enzastaurin)
Recent Studies (post-2010)
(enzastaurin)
Studies
(rottlerin)
Trials
(rottlerin)
Recent Studies (post-2010) (rottlerin)
18852995561202

Protein Interaction Comparison

ProteinTaxonomyenzastaurin (IC50)rottlerin (IC50)
Eukaryotic elongation factor 2 kinaseHomo sapiens (human)5.3
B2 bradykinin receptorCavia porcellus (domestic guinea pig)1.2
Ubiquitin carboxyl-terminal hydrolase 1Homo sapiens (human)8
Beta-lactamaseEscherichia coli K-121.5
Malate dehydrogenaseThermus thermophilus0.7
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)1.2
MAP kinase-activated protein kinase 2Homo sapiens (human)5.4
Protein kinase C delta typeHomo sapiens (human)3
MAP kinase-activated protein kinase 5Homo sapiens (human)1.9
WD repeat-containing protein 48Homo sapiens (human)8
RuvB-like 1Homo sapiens (human)10

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's1 (100.00)2.80

Authors

AuthorsStudies
Alaoui-Jamali, MA; Amzil, H; Bijian, K; Lim, FPL; Miron, CE; Moitessier, N; Nivedha, AK; Su, J; Wernic, D1

Other Studies

1 other study(ies) available for enzastaurin and rottlerin

ArticleYear
Novel Aurora A and Protein Kinase C (α, β1, β2, and θ) Multitarget Inhibitors: Impact of Selenium Atoms on the Potency and Selectivity.
    Journal of medicinal chemistry, 2022, 02-24, Volume: 65, Issue:4

    Topics: Antineoplastic Agents; Aurora Kinase A; Breast Neoplasms; Cell Line, Tumor; Drug Screening Assays, Antitumor; Female; Humans; Hydrogen Bonding; Isoenzymes; Molecular Docking Simulation; Protein Kinase C; Protein Kinase Inhibitors; Selenium Compounds; Small Molecule Libraries; Structure-Activity Relationship; Substrate Specificity; Tumor Stem Cell Assay

2022