Page last updated: 2024-09-05

enzastaurin and nvp-ast487

enzastaurin has been researched along with nvp-ast487 in 1 studies

Compound Research Comparison

Studies
(enzastaurin)
Trials
(enzastaurin)
Recent Studies (post-2010)
(enzastaurin)
Studies
(nvp-ast487)
Trials
(nvp-ast487)
Recent Studies (post-2010) (nvp-ast487)
188529917014

Protein Interaction Comparison

ProteinTaxonomyenzastaurin (IC50)nvp-ast487 (IC50)
Tyrosine-protein kinase ABL1Homo sapiens (human)0.58
Breakpoint cluster region proteinHomo sapiens (human)0.58
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)0.005
Cyclin-dependent kinase-like 3Homo sapiens (human)0.0071
MAP kinase-interacting serine/threonine-protein kinase 1Homo sapiens (human)1.76
MAP kinase-interacting serine/threonine-protein kinase 2Homo sapiens (human)0.02

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ciceri, P; Davis, MI; Herrgard, S; Hocker, M; Hunt, JP; Pallares, G; Treiber, DK; Wodicka, LM; Zarrinkar, PP1

Other Studies

1 other study(ies) available for enzastaurin and nvp-ast487

ArticleYear
Comprehensive analysis of kinase inhibitor selectivity.
    Nature biotechnology, 2011, Oct-30, Volume: 29, Issue:11

    Topics: Catalysis; Drug Design; Enzyme Stability; High-Throughput Screening Assays; Humans; Protein Binding; Protein Kinase Inhibitors; Protein Kinases; Proteomics; Signal Transduction; Substrate Specificity

2011