enzastaurin has been researched along with nvp-ast487 in 1 studies
Studies (enzastaurin) | Trials (enzastaurin) | Recent Studies (post-2010) (enzastaurin) | Studies (nvp-ast487) | Trials (nvp-ast487) | Recent Studies (post-2010) (nvp-ast487) |
---|---|---|---|---|---|
188 | 52 | 99 | 17 | 0 | 14 |
Protein | Taxonomy | enzastaurin (IC50) | nvp-ast487 (IC50) |
---|---|---|---|
Tyrosine-protein kinase ABL1 | Homo sapiens (human) | 0.58 | |
Breakpoint cluster region protein | Homo sapiens (human) | 0.58 | |
Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens (human) | 0.005 | |
Cyclin-dependent kinase-like 3 | Homo sapiens (human) | 0.0071 | |
MAP kinase-interacting serine/threonine-protein kinase 1 | Homo sapiens (human) | 1.76 | |
MAP kinase-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | 0.02 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 1 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Ciceri, P; Davis, MI; Herrgard, S; Hocker, M; Hunt, JP; Pallares, G; Treiber, DK; Wodicka, LM; Zarrinkar, PP | 1 |
1 other study(ies) available for enzastaurin and nvp-ast487
Article | Year |
---|---|
Comprehensive analysis of kinase inhibitor selectivity.
Topics: Catalysis; Drug Design; Enzyme Stability; High-Throughput Screening Assays; Humans; Protein Binding; Protein Kinase Inhibitors; Protein Kinases; Proteomics; Signal Transduction; Substrate Specificity | 2011 |