Page last updated: 2024-09-05

enzastaurin and docetaxel anhydrous

enzastaurin has been researched along with docetaxel anhydrous in 2 studies

Compound Research Comparison

Studies
(enzastaurin)
Trials
(enzastaurin)
Recent Studies (post-2010)
(enzastaurin)
Studies
(docetaxel anhydrous)
Trials
(docetaxel anhydrous)
Recent Studies (post-2010) (docetaxel anhydrous)
188529912,1103,2166,920

Protein Interaction Comparison

ProteinTaxonomyenzastaurin (IC50)docetaxel anhydrous (IC50)
Kinesin-like protein KIF11Homo sapiens (human)0.0014
Nucleotide-binding oligomerization domain-containing protein 2Homo sapiens (human)5.0119

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1
Dreicer, R; Garcia, J; Kania, M; Raghavan, D; Rini, B; Shi, P; Somer, B; Srinivas, S; Vogelzang, N1

Trials

1 trial(s) available for enzastaurin and docetaxel anhydrous

ArticleYear
A randomized, double-blind, placebo-controlled, Phase II study with and without enzastaurin in combination with docetaxel-based chemotherapy in patients with castration-resistant metastatic prostate cancer.
    Investigational new drugs, 2013, Volume: 31, Issue:4

    Topics: Aged; Aged, 80 and over; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Docetaxel; Double-Blind Method; Humans; Indoles; Kaplan-Meier Estimate; Male; Middle Aged; Placebos; Prostatic Neoplasms, Castration-Resistant; Taxoids; Treatment Outcome

2013

Other Studies

1 other study(ies) available for enzastaurin and docetaxel anhydrous

ArticleYear
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013