Page last updated: 2024-09-05

enzastaurin and 4-benzyl-2-methyl-1,2,4-thiadiazolidine-3,5-dione

enzastaurin has been researched along with 4-benzyl-2-methyl-1,2,4-thiadiazolidine-3,5-dione in 1 studies

Compound Research Comparison

Studies
(enzastaurin)
Trials
(enzastaurin)
Recent Studies (post-2010)
(enzastaurin)
Studies
(4-benzyl-2-methyl-1,2,4-thiadiazolidine-3,5-dione)
Trials
(4-benzyl-2-methyl-1,2,4-thiadiazolidine-3,5-dione)
Recent Studies (post-2010) (4-benzyl-2-methyl-1,2,4-thiadiazolidine-3,5-dione)
1885299126184

Protein Interaction Comparison

ProteinTaxonomyenzastaurin (IC50)4-benzyl-2-methyl-1,2,4-thiadiazolidine-3,5-dione (IC50)
[tau protein] kinase Oryctolagus cuniculus (rabbit)2
G2/mitotic-specific cyclin-B2Homo sapiens (human)10
Cyclin-dependent kinase 1Homo sapiens (human)10
Replicase polyprotein 1abSevere acute respiratory syndrome-related coronavirus2.15
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 21.145
G2/mitotic-specific cyclin-B1Homo sapiens (human)10
Glycogen synthase kinase-3 alphaHomo sapiens (human)4.5
Glycogen synthase kinase-3 betaHomo sapiens (human)2.0608
G2/mitotic-specific cyclin-B3Homo sapiens (human)10

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Biru, T; Cinatl, J; Doerr, HW; Loeschmann, N; Michaelis, M; Ogbomo, H1

Other Studies

1 other study(ies) available for enzastaurin and 4-benzyl-2-methyl-1,2,4-thiadiazolidine-3,5-dione

ArticleYear
The anti-tumoral drug enzastaurin inhibits natural killer cell cytotoxicity via activation of glycogen synthase kinase-3β.
    Biochemical pharmacology, 2011, Jan-15, Volume: 81, Issue:2

    Topics: Antineoplastic Agents; Cell Line; Dose-Response Relationship, Drug; Enzyme Activation; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Indoles; Killer Cells, Natural; Perforin; Phosphorylation; Thiadiazoles

2011