entinostat and laq824
entinostat has been researched along with laq824 in 8 studies
Research
Studies (8)
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 4 (50.00) | 29.6817 |
| 2010's | 3 (37.50) | 24.3611 |
| 2020's | 1 (12.50) | 2.80 |
Authors
| Authors | Studies |
|---|---|
| Belvedere, S; Miller, TA; Witter, DJ | 1 |
| Besterman, JM; Bonfils, C; Fournel, M; Frechette, S; Lefebvre, S; Leit, SM; Li, Z; Liu, J; Lu, AH; Mallais, TC; Moradei, OM; Paquin, I; Rahil, J; Tessier, PE; Trachy-Bourget, MC; Vaisburg, AF; Wang, J; Yan, TP | 1 |
| Bottomley, MJ; Carfí, A; De Francesco, R; Gallinari, P; Jones, P; Koch, U; Lahm, A; Lo Surdo, P; Nardi, MC; Neddermann, P; Pallaoro, M; Paolini, C; Sambucini, S; Steinkühler, C | 1 |
| Altamura, S; De Francesco, R; Gallinari, P; Jones, P; Lahm, A; Neddermann, P; Rowley, M; Serafini, S; Steinkühler, C | 1 |
| Bradner, JE; Grachan, ML; Greenberg, EF; Haggarty, SJ; Mazitschek, R; Warnow, T; West, N | 1 |
| Atadja, P; Cao, X; Chen, CH; Cho, YS; Davis, NR; Eckman, J; Fan, J; Fekete, A; Firestone, B; Flynn, J; Green, J; Growney, JD; Holmqvist, M; Hsu, M; Jansson, D; Jiang, L; Kwon, P; Liu, G; Lombardo, F; Lu, Q; Majumdar, D; Meta, C; Perez, L; Pu, M; Ramsey, T; Remiszewski, S; Shultz, MD; Skolnik, S; Traebert, M; Urban, L; Uttamsingh, V; Wang, P; Whitebread, S; Whitehead, L; Yan-Neale, Y; Yao, YM; Zhou, L | 1 |
| Atadja, P; Bickford, S; Buteau, K; Cao, X; Chen, C; Cho, YS; Davis, N; Fan, J; Holmqvist, M; Hsu, M; Jiang, L; Liu, G; Lu, Q; Patel, C; Selvaraj, M; Shultz, M; Suresh, JR; Urban, L; Wang, P; Whitehead, L; Yan-Neale, Y; Zhang, H; Zhou, L | 1 |
| Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M | 1 |
Reviews
1 review(s) available for entinostat and laq824
| Article | Year |
|---|---|
Histone deacetylase inhibitors.
Topics: Animals; Antineoplastic Agents; Binding Sites; Crystallography, X-Ray; Enzyme Inhibitors; Histone Deacetylase Inhibitors; Humans; Models, Molecular; Sequence Alignment; Structure-Activity Relationship | 2003 |
Other Studies
7 other study(ies) available for entinostat and laq824
| Article | Year |
|---|---|
Novel aminophenyl benzamide-type histone deacetylase inhibitors with enhanced potency and selectivity.
Topics: Antineoplastic Agents; Benzamides; Catalytic Domain; Cell Line; Histone Deacetylase 1; Histone Deacetylase Inhibitors; Histone Deacetylases; Humans; Models, Molecular; NADH, NADPH Oxidoreductases; Structure-Activity Relationship | 2007 |
Unraveling the hidden catalytic activity of vertebrate class IIa histone deacetylases.
Topics: Amino Acid Sequence; Animals; Binding Sites; Catalysis; Enzyme Activation; HeLa Cells; Histidine; Histone Deacetylases; Humans; Models, Molecular; Mutation; Protein Structure, Tertiary; Substrate Specificity; Urochordata; Vertebrates | 2007 |
Probing the elusive catalytic activity of vertebrate class IIa histone deacetylases.
Topics: Acetylation; Benzamides; Catalysis; Cells, Cultured; Escherichia coli; Histone Deacetylase Inhibitors; Histone Deacetylases; Humans; Hydroxamic Acids; Kidney; Molecular Structure; Mutation; Peptides, Cyclic; Pyridines; Pyrimidines; Sulfonamides | 2008 |
Chemical phylogenetics of histone deacetylases.
Topics: | 2010 |
Optimization of the in vitro cardiac safety of hydroxamate-based histone deacetylase inhibitors.
Topics: Acrylamides; Animals; Antineoplastic Agents; Drug Screening Assays, Antitumor; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Half-Life; HCT116 Cells; Histone Deacetylase Inhibitors; Humans; Hydroxamic Acids; In Vitro Techniques; Mice; Mice, Nude; Microsomes, Liver; Models, Molecular; Neoplasm Transplantation; Patch-Clamp Techniques; Radioligand Assay; Rats; Rats, Sprague-Dawley; Stereoisomerism; Structure-Activity Relationship; Tissue Distribution; Transplantation, Heterologous | 2011 |
The design, synthesis and structure-activity relationships of novel isoindoline-based histone deacetylase inhibitors.
Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Design; Drug Screening Assays, Antitumor; Histone Deacetylase 1; Histone Deacetylase Inhibitors; Humans; Hydroxamic Acids; Isoindoles; Molecular Structure; Stereoisomerism; Structure-Activity Relationship | 2011 |
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries | 2023 |