enpiperate has been researched along with piperidines in 63 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 39 (61.90) | 18.7374 |
1990's | 16 (25.40) | 18.2507 |
2000's | 8 (12.70) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Bartfai, T; Hedlund, B; Järv, J | 2 |
Gabrio, T; Göber, B; Höhn, H | 1 |
Bartfai, T; Grabczewska, E; Maslinski, W; Ryzewski, J | 1 |
Cohen-Armon, M; Sokolovsky, M | 1 |
Cohen-Armon, M; Henis, YI; Kloog, Y; Sokolovsky, M | 1 |
Du, YL; Lou, YQ | 1 |
Bartfai, T; Danielsson, E; Grundin, R; Ogren, SO; Peterson, LL | 1 |
Bian, CF; Xing, SH; Xu, PC | 1 |
Mei, ZT | 1 |
Sokolovsky, M; van Koppen, CJ | 1 |
Blatt, I; Egozi, Y; Matzkel, A; Schejter, E; Sokolovsky, M; Soreq, H; Zakut, H | 1 |
Barenholz, Y; Henis, YI; Moscona-Amir, E; Sokolovsky, M; Yechiel, E | 1 |
Kloog, Y; Sokolovsky, M | 1 |
Balderman, D; Galron, R; Kloog, Y; Sokolovsky, M | 1 |
Henis, YI; Schreiber, G; Sokolovsky, M | 2 |
Egozi, Y; Kloog, Y | 1 |
Egozi, Y; Henis, YI; Moscona-Amir, E; Sokolovsky, M | 1 |
Baron, B; Kloog, Y | 1 |
Friedman, M; Schreiber, G; Sokolovsky, M | 1 |
Henis, YI; Sokolovsky, M | 1 |
Bartfai, T; Grynfarb, M; Hedlund, B | 1 |
Amitai, G; Avissar, S; Balderman, D; Sokolovsky, M | 1 |
Bartfai, T; Hedlund, B; Lundberg, JM | 1 |
Korczyn, AD; Michaelson, DM; Sokolovsky, M | 1 |
Avissar, S; Galron, R; Henis, YI; Sokolovsky, M | 1 |
Eliyahu, D; Gurwitz, D; Sokolovsky, M; Soreq, H | 1 |
Avissar, S; Egozi, Y; Sokolovsky, M | 4 |
Gavish, M; Sokolovsky, M | 1 |
Avissar, S; Moscona-Amir, E; Sokolovsky, M | 1 |
Avissar, S; Sokolovsky, M | 1 |
Egozi, Y; Kloog, Y; Sokolovsky, M | 1 |
Ben-Baruch, G; Egozi, Y; Kloog, Y; Mashiach, S; Sokolovsky, M | 1 |
Bartfai, T; Fuxe, K; Grynfarb, M; Hedlund, B; Westlind, A | 1 |
Avissar, S; Galron, R; Sokolovsky, M | 1 |
Galron, R; Gurwitz, D; Sokolovsky, M | 1 |
Gurwitz, D; Sokolovsky, M | 1 |
Carey, JE; Frey, KA; Kilbourn, MR; Koeppe, RA; Kuhl, DE; Mulholland, GK; Sherman, P | 1 |
Inoue, O; Kobayashi, K; Satoh, T; Suhara, T; Tateno, Y | 1 |
Inoue, O; Kobayashi, K; Miwa, S; Onoe, H; Suziki, K; Tanaka, M; Tani, Y; Watanabe, Y | 1 |
Inoue, O; Kobayashi, K; Suhara, T; Suzuki, K; Tateno, Y | 1 |
Fröhlich, L; Göber, B; Pietzyk, B | 1 |
el-Fakahany, EE; Hejnová, L; Tucek, S | 1 |
Asahina, M; Shinotoh, H | 1 |
Futatsubashi, M; Kakiuchi, T; Nishiyama, S; Ouchi, Y; Tsukada, H | 1 |
Fukumura, T; Ichimiya, A; Ichiya, Y; Kuwabara, Y; Masuda, K; Ogomori, K; Sasaki, M; Takita, M; Yoshida, T | 2 |
Frey, KA; Koeppe, RA; Kuhl, DE; Mulholland, GK; Zubieta, JK | 1 |
Asahina, M; Hattori, T; Inoue, O; Shinotoh, H; Suhara, T; Suzuki, K | 1 |
Matsushita, M; Okauchi, T; Okubo, Y; Sasaki, Y; Sassa, T; Sudo, Y; Suhara, T; Suzuki, K; Uchida, S; Yoshikawa, K | 1 |
Bergström, M; Höglund, AU; Lângström, B; Sihver, S; Sihver, W; Sjöberg, P; Watanabe, Y | 1 |
Hosoi, R; Inoue, O; Kobayashi, K; Watanabe, Y | 1 |
Pennell, PB | 1 |
Harada, N; Kakiuchi, T; Nishiyama, S; Sato, K; Tsukada, H | 1 |
Foster, NL; Frey, KA; Kilbourn, MR; Koeppe, RA; Kuhl, DE; Mangner, TJ; Zubieta, JK | 1 |
Hatazawa, J; Kakiuchi, T; Miura, S; Nishiyama, S; Ohba, H; Okudera, T; Sato, K; Takahashi, K; Tsukada, H | 1 |
Harada, N; Kakiuchi, T; Nakanishi, S; Nishiyama, S; Ohba, H; Sato, K; Tsukada, H | 1 |
Abe, K; Hatazawa, J; Hosoi, R; Inoue, O; Kashiwagi, Y; Tokumura, M | 1 |
Inoue, O; Itoh, T; Kobayashi, K; Suzuki, K; Tanaka, M | 1 |
2 review(s) available for enpiperate and piperidines
Article | Year |
---|---|
[Muscarinic cholinergic receptor imaging of parkinsonian brain using 11C-NMPB and PET].
Topics: Animals; Benzilates; Brain; Carbon Radioisotopes; Humans; Parkinson Disease; Piperidines; Receptors, Muscarinic; Tomography, Emission-Computed | 1997 |
PET: cholinergic neuroreceptor mapping.
Topics: Benzilates; Brain; Calcium Channel Blockers; Epilepsy, Temporal Lobe; Flumazenil; GABA Modulators; Humans; Piperidines; Receptors, Cholinergic; Tomography, Emission-Computed | 2000 |
1 trial(s) available for enpiperate and piperidines
Article | Year |
---|---|
An acute effect of triazolam on muscarinic cholinergic receptor binding in the human brain measured by positron emission tomography.
Topics: Adolescent; Adult; Benzilates; Brain; Humans; Male; Mental Recall; Parasympatholytics; Piperidines; Receptors, Muscarinic; Tomography, Emission-Computed; Triazolam | 1994 |
60 other study(ies) available for enpiperate and piperidines
Article | Year |
---|---|
Isomerization of the muscarinic receptor . antagonist complex.
Topics: Animals; Benzilates; Cerebral Cortex; Intestine, Small; Kinetics; Male; Mathematics; Muscle, Smooth; Piperidines; Protein Binding; Quinuclidines; Rats; Receptors, Cholinergic; Receptors, Muscarinic | 1979 |
[Pharmacokinetics (rats and rabbits) of N-methyl-4- piperidinylbenzilate (Po)3].
Topics: Administration, Oral; Animals; Benzilates; Female; Injections, Intravenous; Male; Piperidines; Rabbits; Rats; Rats, Inbred Strains; Species Specificity | 1990 |
Muscarinic antagonist binding to intact rat thymocytes.
Topics: Animals; Atropine; Benzilates; Kinetics; Male; Muscarine; N-Methylscopolamine; Piperidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives; Thymus Gland | 1990 |
Interactions between the muscarinic receptors, sodium channels, and guanine nucleotide-binding protein(s) in rat atria.
Topics: Acetylcholine; Animals; Batrachotoxins; Benzilates; Carbachol; Dibucaine; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Heart Atria; Ion Channels; Kinetics; Male; Mathematics; Myocardium; Oxotremorine; Piperidines; Rats; Receptors, Muscarinic; Sodium; Veratridine | 1986 |
Batrachotoxin changes the properties of the muscarinic receptor in rat brain and heart: possible interaction(s) between muscarinic receptors and sodium channels.
Topics: Aconitine; Animals; Batrachotoxins; Benzilates; Binding, Competitive; Brain; Carbachol; Guanylyl Imidodiphosphate; Ion Channels; Kinetics; Macromolecular Substances; Male; Myocardium; Piperidines; Rats; Receptors, Muscarinic; Sodium; Veratridine | 1985 |
[Calcium antagonism of enpiperate on isolated rabbit aorta strips and guinea pig ileum].
Topics: Animals; Aorta; Benzilates; Calcium Channel Blockers; Guinea Pigs; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Piperidines; Rabbits | 1989 |
Anticholinergic potency of psychoactive drugs in human and rat cerebral cortex and striatum.
Topics: Aged; Animals; Antidepressive Agents; Antipsychotic Agents; Benzilates; Cerebral Cortex; Corpus Striatum; Humans; In Vitro Techniques; Male; Parasympatholytics; Piperidines; Psychotropic Drugs; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Species Specificity | 1985 |
[The interactions between dihydroetorphine, L-tetrahydropalmatine, B-7601 and diazepam].
Topics: Alkaloids; Anesthesia, General; Anesthesia, Intravenous; Animals; Antipsychotic Agents; Benzilates; Berberine Alkaloids; Diazepam; Dogs; Drug Interactions; Etorphine; Female; Male; Mice; Morphinans; Piperidines; Rabbits | 1986 |
[Effects of glycolate esters on conditioned behavior].
Topics: Animals; Avoidance Learning; Benzilates; Conditioning, Psychological; Discrimination Learning; Female; Glycolates; Male; Parasympatholytics; Piperidines; Quinuclidines; Quinuclidinyl Benzilate; Rats | 1985 |
Chemical modification of rat cerebral cortex M1 muscarinic receptors: role of histidyl residues in antagonist and agonist binding.
Topics: Animals; Atropine; Benzilates; Binding Sites; Carbachol; Cerebral Cortex; Diethyl Pyrocarbonate; Histidine; Hydrogen-Ion Concentration; Oxotremorine; Piperidines; Rats; Receptors, Muscarinic; Synaptosomes | 1988 |
Divergent regulation of muscarinic binding sites and acetylcholinesterase in discrete regions of the developing human fetal brain.
Topics: Acetylcholine; Acetylcholinesterase; Benzilates; Brain; Embryonic and Fetal Development; Gestational Age; Humans; Kinetics; Neurons; Oxotremorine; Piperidines; Receptors, Muscarinic | 1986 |
Role of lipids in age-related changes in the properties of muscarinic receptors in cultured rat heart myocytes.
Topics: Acetylcholine; Animals; Animals, Newborn; Benzilates; Carbachol; Cells, Cultured; Guanylyl Imidodiphosphate; Kinetics; Liposomes; Myocardium; Oxotremorine; Piperidines; Rats; Receptors, Muscarinic | 1986 |
Bisquaternary pyridinium oximes as allosteric inhibitors of rat brain muscarinic receptors.
Topics: Animals; Benzilates; Brain; Dose-Response Relationship, Drug; Kinetics; Mathematics; Obidoxime Chloride; Oximes; Piperidines; Pyridinium Compounds; Rats; Receptors, Muscarinic | 1985 |
Reversible and irreversible inhibition of rat brain muscarinic receptors is related to different substitutions on bisquaternary pyridinium oximes.
Topics: Animals; Benzilates; Binding, Competitive; Brain Stem; Cell-Free System; Obidoxime Chloride; Oximes; Parasympatholytics; Piperidines; Pyridinium Compounds; Rats; Receptors, Muscarinic; Structure-Activity Relationship; Trimedoxime | 1985 |
Analysis of ligand binding to receptors by competition kinetics. Application to muscarinic antagonists in rat brain cortex.
Topics: Animals; Benzilates; Binding, Competitive; Cerebral Cortex; In Vitro Techniques; Kinetics; Male; N-Methylscopolamine; Parasympatholytics; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives | 1985 |
Rate constants of agonist binding to muscarinic receptors in rat brain medulla. Evaluation by competition kinetics.
Topics: Animals; Benzilates; Binding Sites; Binding, Competitive; In Vitro Techniques; Kinetics; Male; Medulla Oblongata; Parasympathomimetics; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Tritium | 1985 |
Muscarinic receptors in the preoptic area are sensitive to 17 beta-estradiol during the critical period.
Topics: Animals; Benzilates; Binding, Competitive; Clomiphene; Estradiol; Estrus; Female; Hypothalamus; Oxotremorine; Piperidines; Pregnancy; Preoptic Area; Proestrus; Rats; Receptors, Muscarinic; Time Factors | 1985 |
Effect of Ca2+ on the binding characteristics of muscarinic receptors in rat adenohypophysis--variation during the estrous cycle.
Topics: Animals; Benzilates; Binding Sites; Binding, Competitive; Calcium; Calcium Channel Blockers; Diestrus; Estrus; Female; Gallopamil; Male; Oxotremorine; Piperidines; Pituitary Gland, Anterior; Pregnancy; Proestrus; Rats; Receptors, Muscarinic | 1985 |
Fatty acid incorporation increases the affinity of muscarinic cholinergic receptors for agonists.
Topics: Animals; Benzilates; Carbachol; Cell Membrane; Cerebral Cortex; Cobalt; Fatty Acids; Guanosine Triphosphate; Medulla Oblongata; Piperidines; Rats; Receptors, Muscarinic; Structure-Activity Relationship | 1984 |
Interaction of bretylium tosylate with rat cardiac muscarinic receptors. Possible pharmacological relevance to antiarrhythmic action.
Topics: Animals; Anti-Arrhythmia Agents; Benzilates; Binding, Competitive; Brain; Bretylium Compounds; Bretylium Tosylate; Cerebral Cortex; Drug Interactions; In Vitro Techniques; Male; Medulla Oblongata; Myocardium; Piperidines; Rats; Receptors, Muscarinic | 1984 |
Muscarinic antagonists induce different receptor conformations in rat adenohypophysis.
Topics: Allosteric Regulation; Animals; Benzilates; Binding, Competitive; In Vitro Techniques; Male; Models, Chemical; N-Methylscopolamine; Parasympatholytics; Piperidines; Pituitary Gland, Anterior; Protein Conformation; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Scopolamine Derivatives | 1983 |
Two ligands may bind simultaneously to the muscarine receptor.
Topics: Animals; Atropine; Benzilates; Benzodiazepinones; Binding Sites; Binding, Competitive; In Vitro Techniques; Kinetics; Ligands; Male; Models, Biological; Piperidines; Pirenzepine; Quinuclidinyl Benzilate; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Scopolamine | 1982 |
Affinity labeling of muscarinic receptors in rat cerebral cortex with a photolabile antagonist.
Topics: Affinity Labels; Animals; Azides; Benzilates; Binding, Competitive; Brain Chemistry; Parasympatholytics; Photochemistry; Piperidines; Quinuclidines; Quinuclidinyl Benzilate; Rats; Receptors, Cholinergic; Receptors, Muscarinic | 1982 |
Vasoactive intestinal polypeptide enhances muscarinic ligand binding in cat submandibular salivary gland.
Topics: Animals; Benzilates; Binding, Competitive; Carbachol; Cats; Gastrointestinal Hormones; Kinetics; Parasympatholytics; Piperidines; Receptors, Cholinergic; Receptors, Muscarinic; Submandibular Gland; Vasoactive Intestinal Peptide | 1982 |
Antibodies to muscarinic acetylcholine receptors in myasthenia gravis.
Topics: Autoantibodies; Benzilates; Humans; Immunoglobulin G; Kinetics; Myasthenia Gravis; Parasympatholytics; Piperidines; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic | 1982 |
Interactions between antagonist-occupied muscarinic binding sites in rat adenohypophysis.
Topics: Animals; Benzilates; Male; Mathematics; Parasympatholytics; Piperidines; Pituitary Gland, Anterior; Quinuclidinyl Benzilate; Rats; Receptors, Cholinergic; Receptors, Muscarinic | 1982 |
Altered ontogenesis of muscarinic receptors in agranular cerebellar cortex.
Topics: Aging; Animals; Benzilates; Cerebellar Cortex; Heterozygote; Homozygote; Hyperbilirubinemia, Hereditary; Kinetics; Mice; Mice, Inbred Strains; Parasympatholytics; Piperidines; Rats; Rats, Gunn; Rats, Inbred Strains; Receptors, Cholinergic; Receptors, Muscarinic; Species Specificity | 1982 |
Muscarinic mechanisms and sex hormone secretion in rat adenohypophysis and preoptic area.
Topics: Animals; Benzilates; Biomechanical Phenomena; Female; Gonadal Steroid Hormones; Hypothalamus; Male; Muscarine; Oxotremorine; Piperidines; Pituitary Gland, Anterior; Preoptic Area; Rats; Rats, Inbred Strains | 1982 |
Solubilization of muscarinic acetylcholine receptor by zwitterionic detergent from rat brain cortex.
Topics: Animals; Benzilates; Cerebral Cortex; Cholic Acids; Detergents; Kinetics; Piperidines; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Solubility | 1982 |
Photoaffinity labeling reveals two muscarinic receptor macromolecules associated with the presence of calcium in rat adenohypophysis.
Topics: Affinity Labels; Animals; Benzilates; Calcium; Female; Kinetics; Piperidines; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains; Receptors, Cholinergic; Receptors, Muscarinic | 1982 |
Biochemical characterization and sex dimorphism of muscarinic receptors in rat adenohypophysis.
Topics: Animals; Benzilates; Binding, Competitive; Estrus; Female; Kinetics; Male; Piperidines; Pituitary Gland, Anterior; Pregnancy; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Sex Differentiation; Sex Factors | 1981 |
Guanine nucleotides preferentially inhibit binding of antagonists (male) and agonists (female) to muscarinic receptors of rat adenohypophysis.
Topics: Animals; Benzilates; Estrus; Female; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Male; Oxotremorine; Parasympatholytics; Piperidines; Pituitary Gland, Anterior; Pregnancy; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Sex Factors | 1981 |
Biochemical characterization of muscarinic receptors.
Topics: Animals; Atropine; Benzilates; Binding, Competitive; Brain; Kinetics; Mice; Parasympatholytics; Piperidines; Receptors, Cholinergic; Receptors, Muscarinic; Scopolamine; Tissue Distribution | 1980 |
Altered ontogenesis of muscarinic cholinergic receptor in mouse brain: effect of L-thyroxine and betamethasone.
Topics: Aging; Animals; Animals, Newborn; Benzilates; Betamethasone; Brain; Cerebellum; Cerebral Cortex; Kinetics; Mice; Parasympatholytics; Piperidines; Receptors, Cholinergic; Receptors, Muscarinic; Thyroxine | 1981 |
Studies on muscarinic receptors in mouse and rat hypothalamus: a comparison of sex and cyclical differences.
Topics: Animals; Benzilates; Female; Hydroxydopamines; Hypothalamus; Kinetics; Male; Oxotremorine; Piperidines; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Sex Factors; Species Specificity | 1981 |
Muscarinic supersensitivity induced by septal lesion or chronic atropine treatment.
Topics: Animals; Atropine; Benzilates; Cerebral Cortex; Corpus Striatum; Hippocampus; Hypothalamus; Male; Piperidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Cholinergic; Receptors, Muscarinic; Septum Pellucidum | 1981 |
Temperature dependence of agonist binding to muscarinic receptors in rat hypothalamic regions.
Topics: Animals; Benzilates; Brain; Female; Hypothalamus; Kinetics; Male; Mice; Oxotremorine; Parasympatholytics; Piperidines; Preoptic Area; Receptors, Cholinergic; Receptors, Muscarinic; Sex Factors; Thermodynamics; Tissue Distribution | 1981 |
Aging process decreases the density of muscarinic receptors in rat adenohypophysis.
Topics: Adrenal Cortex; Adrenal Medulla; Aging; Animals; Benzilates; Female; Hypothalamus; Organ Specificity; Piperidines; Pituitary Gland, Anterior; Preoptic Area; Rats; Rats, Inbred Strains; Receptors, Cholinergic; Receptors, Muscarinic | 1981 |
Kinetic studies on muscarinic antagonist-agonist competition.
Topics: Animals; Atropine; Benzilates; Binding, Competitive; Carbachol; Intestine, Small; Kinetics; Male; Muscle, Smooth; Oxotremorine; Parasympatholytics; Piperidines; Rats; Receptors, Cholinergic; Receptors, Muscarinic | 1980 |
Muscarinic receptor binding in mouse brain: regulation by guanine nucleotides.
Topics: Animals; Benzilates; Brain; Guanine Nucleotides; Guanosine Triphosphate; Magnesium; Male; Medulla Oblongata; Mice; Oxotremorine; Piperidines; Pons; Receptors, Cholinergic; Receptors, Muscarinic; Structure-Activity Relationship | 1980 |
Induced interconversion of agonist affinity states in muscarinic receptor from mice brain: effects of temperature and sugars.
Topics: Animals; Benzilates; Brain; Cerebral Cortex; Hydrogen-Ion Concentration; Medulla Oblongata; Mice; Oxotremorine; Parasympathomimetics; Piperidines; Pons; Protein Conformation; Receptors, Cholinergic; Receptors, Muscarinic; Structure-Activity Relationship; Temperature | 1980 |
Synthesis, in vivo biodistribution and dosimetry of [11C]N-methylpiperidyl benzilate ([11C]NMPB), a muscarinic acetylcholine receptor antagonist.
Topics: Animals; Benzilates; Carbon Radioisotopes; Female; Male; Mice; Muscarinic Antagonists; Piperidines; Radiation Dosage; Rats; Rats, Sprague-Dawley; Tissue Distribution | 1995 |
Effect of 6R-tetrahydrobiopterin on the central muscarinic cholinergic receptor as evaluated by positron emission tomography studies using rhesus monkey.
Topics: Animals; Benzilates; Biopterins; Brain; Carbon Radioisotopes; Macaca mulatta; Male; Molecular Structure; Organ Specificity; Piperidines; Receptors, Muscarinic; Tomography, Emission-Computed | 1993 |
Age-related changes in human muscarinic acetylcholine receptors measured by positron emission tomography.
Topics: Adolescent; Adult; Aged; Aging; Benzilates; Brain Chemistry; Humans; Ligands; Magnetic Resonance Imaging; Male; Middle Aged; Parasympatholytics; Piperidines; Receptors, Cholinergic; Tomography, Emission-Computed | 1993 |
[The biomimetic oxidation of propiverine hydrochloride and 1-methyl-4-piperidylbenzilate].
Topics: Animals; Benzilates; Chromatography, Thin Layer; Mass Spectrometry; Oxidation-Reduction; Piperidines; Rats; Spectrophotometry, Ultraviolet | 1995 |
Positive and negative allosteric interactions on muscarinic receptors.
Topics: Alcuronium; Allosteric Regulation; Animals; Atropine; Benzilates; In Vitro Techniques; Male; Muscarinic Antagonists; Myocardium; Piperidines; Quinuclidinyl Benzilate; Rats; Rats, Wistar; Receptors, Muscarinic | 1995 |
Changes in cerebral blood flow and postsynaptic muscarinic cholinergic activity in rats with bilateral carotid artery ligation.
Topics: Animals; Benzilates; Brain; Brain Ischemia; Carbon Radioisotopes; Carotid Artery, Common; Cerebrovascular Circulation; Ligation; Male; Muscarinic Antagonists; Oxygen Radioisotopes; Piperidines; Radiopharmaceuticals; Rats; Rats, Wistar; Receptors, Muscarinic; Time Factors; Tomography, Emission-Computed; Water | 1998 |
Cerebral muscarinic acetylcholinergic receptor measurement in Alzheimer's disease patients on 11C-N-methyl-4-piperidyl benzilate--comparison with cerebral blood flow and cerebral glucose metabolism.
Topics: Aged; Aged, 80 and over; Alzheimer Disease; Benzilates; Brain; Carbon Radioisotopes; Case-Control Studies; Cerebrovascular Circulation; Female; Glucose; Humans; Male; Middle Aged; Piperidines; Receptors, Muscarinic; Tissue Distribution; Tomography, Emission-Computed | 1998 |
Quantification of muscarinic cholinergic receptors with [11C]NMPB and positron emission tomography: method development and differentiation of tracer delivery from receptor binding.
Topics: Adult; Benzilates; Biological Transport; Brain; Carbon Radioisotopes; Female; Humans; Male; Occipital Lobe; Parasympathomimetics; Piperidines; Receptors, Muscarinic; Sensitivity and Specificity; Tissue Distribution; Tomography, Emission-Computed | 1998 |
Brain muscarinic receptors in progressive supranuclear palsy and Parkinson's disease: a positron emission tomographic study.
Topics: Aged; Benzilates; Brain; Brain Mapping; Carbon Radioisotopes; Cholinergic Fibers; Female; Humans; Male; Middle Aged; Neuropsychological Tests; Parasympatholytics; Parkinson Disease; Piperidines; Receptors, Cholinergic; Receptors, Muscarinic; Supranuclear Palsy, Progressive; Tomography, Emission-Computed | 1998 |
Muscarinic receptor occupancy by biperiden in living human brain.
Topics: Adult; Animals; Benzilates; Binding Sites; Biperiden; Brain; Humans; Macaca mulatta; Male; Muscarinic Antagonists; Piperidines; Receptors, Muscarinic; Time Factors; Tomography, Emission-Computed | 1999 |
Quantitative autoradiography with short-lived positron emission tomography tracers: a study on muscarinic acetylcholine receptors with N-[(11)C]methyl-4-piperidylbenzilate.
Topics: Animals; Autoradiography; Benzilates; Cerebral Cortex; Half-Life; Image Processing, Computer-Assisted; Male; Neostriatum; Piperidines; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Spinal Cord; Tomography, Emission-Computed | 1999 |
Sex-related differences in the muscarinic acetylcholinergic receptor in the healthy human brain--a positron emission tomography study.
Topics: Adult; Aged; Aging; Benzilates; Brain; Carbon Radioisotopes; Female; Humans; Ligands; Male; Middle Aged; Piperidines; Receptors, Muscarinic; Sex Characteristics; Tomography, Emission-Computed | 2000 |
Evaluation of in vivo binding properties of 3H-NMPB and 3H-QNB in mouse brain.
Topics: Animals; Benzilates; Biperiden; Brain; Male; Mice; Muscarinic Antagonists; Parasympatholytics; Piperidines; Quinuclidinyl Benzilate; Receptors, Muscarinic | 1999 |
Development and evaluation of muscarinic cholinergic receptor ligands N-[11C]ethyl-4-piperidyl benzilate and N-[11C]propyl-4-piperidyl benzilate: a PET study in comparison with N-[11C]methyl-4-piperidyl benzilate in the conscious monkey brain.
Topics: Animals; Benzilates; Brain; Isotope Labeling; Ligands; Macaca mulatta; Magnetic Resonance Imaging; Male; Piperidines; Radiopharmaceuticals; Receptors, Muscarinic; Tomography, Emission-Computed | 2000 |
Assessment of muscarinic receptor concentrations in aging and Alzheimer disease with [11C]NMPB and PET.
Topics: Adult; Age Factors; Aged; Aging; Alzheimer Disease; Benzilates; Biological Transport; Brain; Brain Chemistry; Carbon Radioisotopes; Computer Simulation; Female; Humans; Kinetics; Male; Middle Aged; Piperidines; Receptors, Muscarinic; Tomography, Emission-Computed | 2001 |
Evaluation of novel PET ligands (+)N-[11C]methyl-3-piperidyl benzilate ([11C](+)3-MPB) and its stereoisomer [11C](-)3-MPB for muscarinic cholinergic receptors in the conscious monkey brain: a PET study in comparison with.
Topics: Animals; Benzilates; Brain; Carbon Radioisotopes; Consciousness; Hallucinogens; Macaca mulatta; Male; Piperidines; Receptors, Muscarinic; Stereoisomerism; Tomography, Emission-Computed | 2001 |
Age-related changes in muscarinic cholinergic receptors in the living brain: a PET study using N-[11C]methyl-4-piperidyl benzilate combined with cerebral blood flow measurement in conscious monkeys.
Topics: Acetylcholine; Aging; Animals; Benzilates; Binding, Competitive; Brain; Brain Mapping; Cerebrovascular Circulation; Consciousness; Macaca mulatta; Magnetic Resonance Imaging; Male; Oxygen Radioisotopes; Parasympatholytics; Pharmacokinetics; Piperidines; Radioligand Assay; Receptors, Muscarinic; Tomography, Emission-Computed | 2001 |
Discrepancy between cell injury and benzodiazepine receptor binding after transient middle cerebral artery occlusion in rats.
Topics: Animals; Autoradiography; Benzazepines; Benzilates; Binding Sites; Binding, Competitive; Cerebral Cortex; Cerebral Infarction; Corpus Striatum; Disease Models, Animal; Down-Regulation; Flumazenil; Infarction, Middle Cerebral Artery; Male; Nerve Degeneration; Piperidines; Radioligand Assay; Rats; Rats, Wistar; Reaction Time; Receptors, Dopamine D1; Receptors, GABA-A; Receptors, Muscarinic; Reperfusion Injury; Sensitivity and Specificity; Tritium | 2004 |
Binding kinetics of 11C-N-methyl piperidyl benzilate (11C-NMPB) in a rhesus monkey brain using the cerebellum as a reference region.
Topics: Animals; Benzilates; Binding Sites; Brain; Brain Mapping; Cerebellum; Macaca mulatta; Male; Metabolic Clearance Rate; Piperidines; Positron-Emission Tomography; Protein Binding; Radiopharmaceuticals; Receptors, Muscarinic; Reference Values; Tissue Distribution | 2005 |