Page last updated: 2024-09-03

enkephalin-met, arg(6)-phe(7)- and norbinaltorphimine

enkephalin-met, arg(6)-phe(7)- has been researched along with norbinaltorphimine in 5 studies

Compound Research Comparison

Studies
(enkephalin-met, arg(6)-phe(7)-)
Trials
(enkephalin-met, arg(6)-phe(7)-)
Recent Studies (post-2010)
(enkephalin-met, arg(6)-phe(7)-)
Studies
(norbinaltorphimine)
Trials
(norbinaltorphimine)
Recent Studies (post-2010) (norbinaltorphimine)
1891109180205

Protein Interaction Comparison

ProteinTaxonomyenkephalin-met, arg(6)-phe(7)- (IC50)norbinaltorphimine (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.0104
Kappa-type opioid receptorMus musculus (house mouse)0.0029
Mu-type opioid receptorHomo sapiens (human)0.212
Delta-type opioid receptorHomo sapiens (human)0.024
Kappa-type opioid receptorHomo sapiens (human)0.0036

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (20.00)18.2507
2000's3 (60.00)29.6817
2010's1 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Benyhe, S; Borsodi, A; Medzihradszky, K; Orosz, G; Rónai, AZ; Sartania, N; Szatmári, I1
Cheong, YP; Cho, KP; Kim, CJ; Kim, JK; Kim, KW; Kwun, J; Woo, RS1
Bujdosó, E; Farkas, J; Jászberényi, M; Telegdy, G; Tóth, G; Wollemann, M1
Barlow, MA; Caffrey, JL; Deo, S; Johnson, S1
Bagosi, Z; Csabafi, K; Jászberényi, M; Telegdy, G; Tóth, G; Wollemann, M1

Other Studies

5 other study(ies) available for enkephalin-met, arg(6)-phe(7)- and norbinaltorphimine

ArticleYear
Irreversible labelling of the opioid receptors by a melphalan-substituted [Met5]enkephalin-Arg-Phe derivative.
    European journal of pharmacology, 1999, Jun-04, Volume: 373, Issue:2-3

    Topics: Affinity Labels; Amino Acid Sequence; Amino Acid Substitution; Animals; Binding Sites; Binding, Competitive; Brain; Enkephalin, Methionine; Female; Guinea Pigs; Male; Melphalan; Membranes; Naloxone; Naltrexone; Narcotic Antagonists; Radioligand Assay; Rats; Receptors, Opioid

1999
Receptor selectivity of Met-enkephalin-Arg6-Phe7, an endogenous opioid peptide, in cerebral cortex of human and rat.
    Life sciences, 2000, May-26, Volume: 67, Issue:1

    Topics: Adult; Animals; Benzeneacetamides; Benzomorphans; Binding Sites; Cerebral Cortex; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Methionine; Ethylketocyclazocine; Female; Humans; Male; Naloxone; Naltrexone; Norepinephrine; Oligopeptides; Peptide Fragments; Peptides; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Somatostatin

2000
Behavioral and neuroendocrine actions of the Met-enkephalin-related peptide MERF.
    Hormones and behavior, 2003, Volume: 43, Issue:2

    Topics: Analysis of Variance; Animals; Behavior, Animal; Corticotropin-Releasing Hormone; Dopamine; Enkephalin, Methionine; Exploratory Behavior; Haloperidol; Hormone Antagonists; Hypothalamo-Hypophyseal System; Male; Mice; Motor Activity; Naloxone; Naltrexone; Narcotic Antagonists; Neostriatum; Organ Culture Techniques; Peptide Fragments; Pituitary-Adrenal System

2003
Vagotonic effects of enkephalin are not mediated by sympatholytic mechanisms.
    Experimental biology and medicine (Maywood, N.J.), 2006, Volume: 231, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Dogs; Enkephalin, Methionine; Female; Heart Rate; Male; Naltrexone; Receptors, Opioid, kappa; Sympatholytics; Vagus Nerve

2006
The action of a synthetic derivative of Met5-enkephalin-Arg6-Phe7 on behavioral and endocrine responses.
    Peptides, 2011, Volume: 32, Issue:8

    Topics: Animals; Behavior, Animal; Enkephalin, Methionine; Enkephalins; Hypothalamo-Hypophyseal System; Male; Mice; Mice, Inbred Strains; Naloxone; Naltrexone; Oligopeptides; Pituitary-Adrenal System

2011