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enkephalin, ser(2), leu(5), thr(6)- and deltorphin i, ala(2)-

enkephalin, ser(2), leu(5), thr(6)- has been researched along with deltorphin i, ala(2)- in 3 studies

Compound Research Comparison

Studies
(enkephalin, ser(2), leu(5), thr(6)-)
Trials
(enkephalin, ser(2), leu(5), thr(6)-)
Recent Studies (post-2010)
(enkephalin, ser(2), leu(5), thr(6)-)
Studies
(deltorphin i, ala(2)-)
Trials
(deltorphin i, ala(2)-)
Recent Studies (post-2010) (deltorphin i, ala(2)-)
2240512204

Protein Interaction Comparison

ProteinTaxonomyenkephalin, ser(2), leu(5), thr(6)- (IC50)deltorphin i, ala(2)- (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.0003
Delta-type opioid receptorRattus norvegicus (Norway rat)0.0005
Mu-type opioid receptorHomo sapiens (human)0.225
Delta-type opioid receptorHomo sapiens (human)0.0009
Kappa-type opioid receptorHomo sapiens (human)7.33

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bernard, D; Coop, A; MacKerell, AD1
Crook, TJ; Hill, RG; Kitchen, I1
Crook, TJ; Hill, RG; Kitchen, I; Muhammad, BY1

Other Studies

3 other study(ies) available for enkephalin, ser(2), leu(5), thr(6)- and deltorphin i, ala(2)-

ArticleYear
Quantitative conformationally sampled pharmacophore for delta opioid ligands: reevaluation of hydrophobic moieties essential for biological activity.
    Journal of medicinal chemistry, 2007, Apr-19, Volume: 50, Issue:8

    Topics: Animals; Cell Line, Tumor; Enkephalin, Leucine; Hydrophobic and Hydrophilic Interactions; Ligands; Models, Molecular; Molecular Conformation; Phenylalanine; Quantitative Structure-Activity Relationship; Rats; Receptors, Opioid, delta

2007
Effects of the delta-opioid receptor antagonist naltrindole on antinociceptive responses to selective delta-agonists in post-weanling rats.
    British journal of pharmacology, 1992, Volume: 107, Issue:2

    Topics: Analgesics; Animals; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalins; Indoles; Male; Morphinans; Naloxone; Naltrexone; Narcotic Antagonists; Oligopeptides; Pain Measurement; Rats; Rats, Wistar; Receptors, Opioid, delta

1992
Evidence that weaning stimulates the developmental expression of a delta-opioid receptor subtype in the rat.
    Brain research. Developmental brain research, 1994, Mar-18, Volume: 78, Issue:1

    Topics: Analgesics; Animals; Dose-Response Relationship, Drug; Enkephalin, Leucine; Female; Male; Naltrexone; Narcotic Antagonists; Oligopeptides; Rats; Rats, Wistar; Receptors, Opioid, delta; Weaning

1994