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enkephalin, pen(2,5)-4-chloro-phe(4)- and morphine

enkephalin, pen(2,5)-4-chloro-phe(4)- has been researched along with morphine in 3 studies

Compound Research Comparison

Studies
(enkephalin, pen(2,5)-4-chloro-phe(4)-)
Trials
(enkephalin, pen(2,5)-4-chloro-phe(4)-)
Recent Studies (post-2010)
(enkephalin, pen(2,5)-4-chloro-phe(4)-)
Studies
(morphine)
Trials
(morphine)
Recent Studies (post-2010) (morphine)
120144,2705,2008,695

Protein Interaction Comparison

ProteinTaxonomyenkephalin, pen(2,5)-4-chloro-phe(4)- (IC50)morphine (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.2939
Delta-type opioid receptorRattus norvegicus (Norway rat)0.2278
Kappa-type opioid receptorMus musculus (house mouse)0.0828
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0385
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0545
Mu-type opioid receptorHomo sapiens (human)0.122
Delta-type opioid receptorHomo sapiens (human)0.1199
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.9308
Kappa-type opioid receptorHomo sapiens (human)0.655
Mu-type opioid receptorMus musculus (house mouse)0.3305
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.202
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.25

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (33.33)18.2507
2000's2 (66.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Al-Ghananeem, AM; Butterfield, DA; Byrn, SR; Crooks, PA; Kottayil, SG1
Appleyard, SM; Davis, TP; Hruby, VJ; Knapp, RJ; Lipkowski, AW; Misicka, A; Slaninova, J; Weber, SJ; Yamamura, HI1
Amico, JA; Brown, DC; Perkowski, SZ; Shofer, F1

Other Studies

3 other study(ies) available for enkephalin, pen(2,5)-4-chloro-phe(4)- and morphine

ArticleYear
Opiate receptor binding properties of morphine-, dihydromorphine-, and codeine 6-O-sulfate ester congeners.
    Bioorganic & medicinal chemistry letters, 2006, Aug-15, Volume: 16, Issue:16

    Topics: Animals; Codeine; Dihydromorphine; Esters; Guinea Pigs; Inhibitory Concentration 50; Kinetics; Ligands; Models, Chemical; Morphine; Protein Binding; Sulfates

2006
[125I-Tyr1]biphalin binding to opioid receptors of rat brain and NG108-15 cell membranes.
    Life sciences, 1998, Volume: 62, Issue:14

    Topics: Animals; Brain; Cell Line; Cell Membrane; Enkephalins; Iodine Radioisotopes; Morphine; Naltrexone; Narcotic Antagonists; Oligopeptides; Radioligand Assay; Rats; Receptors, Opioid

1998
Effect of centrally administered opioid receptor agonists on CSF and plasma oxytocin concentrations in dogs.
    American journal of veterinary research, 2001, Volume: 62, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Cross-Over Studies; Dogs; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Injections, Spinal; Male; Morphine; Oxytocin; Random Allocation; Receptors, Opioid

2001