enkephalin, pen(2,5)-4-chloro-phe(4)- has been researched along with bw 373u86 in 1 studies
Studies (enkephalin, pen(2,5)-4-chloro-phe(4)-) | Trials (enkephalin, pen(2,5)-4-chloro-phe(4)-) | Recent Studies (post-2010) (enkephalin, pen(2,5)-4-chloro-phe(4)-) | Studies (bw 373u86) | Trials (bw 373u86) | Recent Studies (post-2010) (bw 373u86) |
---|---|---|---|---|---|
12 | 0 | 1 | 80 | 0 | 4 |
Protein | Taxonomy | enkephalin, pen(2,5)-4-chloro-phe(4)- (IC50) | bw 373u86 (IC50) |
---|---|---|---|
Delta-type opioid receptor | Rattus norvegicus (Norway rat) | 0.02 | |
Mu-type opioid receptor | Rattus norvegicus (Norway rat) | 0.9346 | |
Mu-type opioid receptor | Homo sapiens (human) | 0.0021 | |
Delta-type opioid receptor | Homo sapiens (human) | 0.0002 | |
Kappa-type opioid receptor | Cavia porcellus (domestic guinea pig) | 0.0003 | |
Kappa-type opioid receptor | Homo sapiens (human) | 0.02 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Alfaro-Lopez, J; Davis, P; Hosohata, K; Hruby, VJ; Jernigan, KA; Li, X; Liao, S; Lin, J; Porreca, F; Shenderovich, MD; Stropova, D; Yamamura, HI | 1 |
1 other study(ies) available for enkephalin, pen(2,5)-4-chloro-phe(4)- and bw 373u86
Article | Year |
---|---|
De novo design, synthesis, and biological activities of high-affinity and selective non-peptide agonists of the delta-opioid receptor.
Topics: Animals; Benzhydryl Compounds; Brain; Drug Design; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Ligands; Male; Mice; Mice, Inbred ICR; Molecular Mimicry; Muscle Contraction; Muscle, Smooth; Mutation; Peptides; Piperazines; Radioligand Assay; Rats; Receptors, Opioid, delta; Stereoisomerism; Structure-Activity Relationship; Vas Deferens | 1998 |