enkephalin, leucine has been researched along with tan 67 in 10 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 8 (80.00) | 18.2507 |
2000's | 1 (10.00) | 29.6817 |
2010's | 1 (10.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Alt, A; Banks, M; Bassoni, DL; Budenholzer, LM; Burford, NT; Canals, M; Christopoulos, A; Filizola, M; Gerritz, SW; Han, Y; Herbst, JJ; Livingston, KE; O'Connell, J; Ryan, MR; Shang, Y; Traynor, JR; Wehrman, TS; Zhang, L | 1 |
Calderon, SN; De Leon, IA; Knapp, RJ; Landsman, R; Malatynska, E; Nagase, H; Rice, K; Santoro, G; Varga, E; Waite, S | 1 |
Endoh, T; Misawa, M; Mori, T; Nagase, H; Suzuki, T; Tsuji, M | 2 |
Calderon, SN; Hruby, VJ; Kawai, K; Knapp, RJ; Landsman, RS; Li, X; Malatynska, E; Mizusura, A; Nagase, H; Rice, K; Roeske, WR; Stropova, D; Varga, EV; Yamamura, HI; Zalewska, T | 1 |
Kamei, J; Kawai, K; Mizoguchi, H; Mizusuna, A; Nagase, H; Narita, M; Suzuki, T; Tseng, LF | 1 |
Kishimoto, Y; Maeda, J; Misawa, M; Mori, T; Nagase, H; Suzuki, T; Tsuji, M | 1 |
Burkey, TH; Hosohata, K; Hosohata, Y; Hruby, VJ; Knapp, RJ; Nagase, H; Porreca, F; Quock, RM; Rice, KC; Roeske, WR; Yamamura, HI; Zhang, X | 1 |
Kamei, J; Nagase, H; Ohsawa, M | 1 |
Bespalova, ZhD; Lasukova, TV; Maslov, LN; Nagase, H; Oldgen, P; Rice, KK | 1 |
10 other study(ies) available for enkephalin, leucine and tan 67
Article | Year |
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Discovery, synthesis, and molecular pharmacology of selective positive allosteric modulators of the δ-opioid receptor.
Topics: Animals; Arrestins; Benzamides; beta-Arrestins; Binding, Competitive; Cell Membrane; Chemistry Techniques, Synthetic; CHO Cells; Cricetulus; Drug Discovery; Drug Evaluation, Preclinical; Enkephalin, Leucine; Enzyme Activation; Extracellular Signal-Regulated MAP Kinases; Molecular Structure; Molecular Targeted Therapy; Piperazines; Protein Binding; Quinolines; Receptors, Opioid, delta; Structure-Activity Relationship | 2015 |
Efficacy of peptide and nonpeptidic agonists at the cloned human delta opioid receptor.
Topics: Analgesics; Animals; Benzamides; Binding, Competitive; CHO Cells; Cloning, Molecular; Cricetinae; Cyclic AMP; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Humans; Kinetics; Opioid Peptides; Piperazines; Quinolines; Receptors, Opioid, delta; Recombinant Proteins | 1995 |
Effects of a highly selective nonpeptide delta opioid receptor agonist, TAN-67, on morphine-induced antinociception in mice.
Topics: Analgesics; Animals; Drug Interactions; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Injections, Subcutaneous; Male; Mice; Mice, Inbred Strains; Morphine; Naltrexone; Nociceptors; Oligopeptides; Quinolines; Receptors, Opioid, delta | 1995 |
Effect of the highly selective and nonpeptide delta opioid receptor agonist TAN-67 on the morphine-induced place preference in mice.
Topics: Analgesics; Animals; Benzylidene Compounds; Dopamine; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Limbic System; Male; Mice; Morphine; Naltrexone; Quinolines; Receptors, Opioid, delta; Reward | 1996 |
The third extracellular loop of the human delta-opioid receptor determines the selectivity of delta-opioid agonists.
Topics: Amino Acid Sequence; Animals; COS Cells; Enkephalins; Humans; Molecular Sequence Data; Mutagenesis, Site-Directed; Oligopeptides; Quinolines; Receptors, Opioid, delta; Recombinant Fusion Proteins | 1996 |
Delta-1 opioid receptor-mediated antinociceptive properties of a nonpeptidic delta opioid receptor agonist, (-)TAN-67, in the mouse spinal cord.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Hyperalgesia; Injections, Spinal; Male; Mice; Mice, Inbred ICR; Pain; Pain Measurement; Pyrrolidines; Quinolines; Reaction Time; Receptors, Opioid, delta; Spinal Cord | 1997 |
Differential effects of mu-, delta- and kappa-opioid receptor agonists on the discriminative stimulus properties of cocaine in rats.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Analysis of Variance; Animals; Cocaine; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Injections, Intraventricular; Male; Morphine; Narcotics; Pyrrolidines; Quinolines; Rats; Rats, Inbred F344; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Substance-Related Disorders | 1997 |
Relative efficacies of delta-opioid receptor agonists at the cloned human delta-opioid receptor.
Topics: Animals; Benzamides; CHO Cells; Cloning, Molecular; Cricetinae; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Naltrexone; Narcotic Antagonists; Piperazines; Quinolines; Receptors, Opioid, delta; Sulfur Radioisotopes | 1997 |
Role of intracellular calcium in modification of mu and delta opioid receptor-mediated antinociception by diabetes in mice.
Topics: Analgesics; Analgesics, Opioid; Animals; Calcium; Calcium Chloride; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Egtazic Acid; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Injections, Intraventricular; Male; Mice; Mice, Inbred ICR; Pain Measurement; Quinolines; Receptors, Opioid, delta; Receptors, Opioid, mu; Ryanodine | 1998 |
Delta-opioid receptor antagonists exhibit properties of partial delta-receptor agonists in isolated perfused heart.
Topics: Animals; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Heart; In Vitro Techniques; Male; Myocardial Contraction; Myocardial Ischemia; Naltrexone; Oligopeptides; Perfusion; Quinolines; Rats; Rats, Wistar; Receptors, Opioid, delta | 2004 |