enkephalin, leucine and tan 67

enkephalin, leucine has been researched along with tan 67 in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (80.00)18.2507
2000's1 (10.00)29.6817
2010's1 (10.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Alt, A; Banks, M; Bassoni, DL; Budenholzer, LM; Burford, NT; Canals, M; Christopoulos, A; Filizola, M; Gerritz, SW; Han, Y; Herbst, JJ; Livingston, KE; O'Connell, J; Ryan, MR; Shang, Y; Traynor, JR; Wehrman, TS; Zhang, L1
Calderon, SN; De Leon, IA; Knapp, RJ; Landsman, R; Malatynska, E; Nagase, H; Rice, K; Santoro, G; Varga, E; Waite, S1
Endoh, T; Misawa, M; Mori, T; Nagase, H; Suzuki, T; Tsuji, M2
Calderon, SN; Hruby, VJ; Kawai, K; Knapp, RJ; Landsman, RS; Li, X; Malatynska, E; Mizusura, A; Nagase, H; Rice, K; Roeske, WR; Stropova, D; Varga, EV; Yamamura, HI; Zalewska, T1
Kamei, J; Kawai, K; Mizoguchi, H; Mizusuna, A; Nagase, H; Narita, M; Suzuki, T; Tseng, LF1
Kishimoto, Y; Maeda, J; Misawa, M; Mori, T; Nagase, H; Suzuki, T; Tsuji, M1
Burkey, TH; Hosohata, K; Hosohata, Y; Hruby, VJ; Knapp, RJ; Nagase, H; Porreca, F; Quock, RM; Rice, KC; Roeske, WR; Yamamura, HI; Zhang, X1
Kamei, J; Nagase, H; Ohsawa, M1
Bespalova, ZhD; Lasukova, TV; Maslov, LN; Nagase, H; Oldgen, P; Rice, KK1

Other Studies

10 other study(ies) available for enkephalin, leucine and tan 67

ArticleYear
Discovery, synthesis, and molecular pharmacology of selective positive allosteric modulators of the δ-opioid receptor.
    Journal of medicinal chemistry, 2015, May-28, Volume: 58, Issue:10

    Topics: Animals; Arrestins; Benzamides; beta-Arrestins; Binding, Competitive; Cell Membrane; Chemistry Techniques, Synthetic; CHO Cells; Cricetulus; Drug Discovery; Drug Evaluation, Preclinical; Enkephalin, Leucine; Enzyme Activation; Extracellular Signal-Regulated MAP Kinases; Molecular Structure; Molecular Targeted Therapy; Piperazines; Protein Binding; Quinolines; Receptors, Opioid, delta; Structure-Activity Relationship

2015
Efficacy of peptide and nonpeptidic agonists at the cloned human delta opioid receptor.
    Proceedings of the Western Pharmacology Society, 1995, Volume: 38

    Topics: Analgesics; Animals; Benzamides; Binding, Competitive; CHO Cells; Cloning, Molecular; Cricetinae; Cyclic AMP; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Humans; Kinetics; Opioid Peptides; Piperazines; Quinolines; Receptors, Opioid, delta; Recombinant Proteins

1995
Effects of a highly selective nonpeptide delta opioid receptor agonist, TAN-67, on morphine-induced antinociception in mice.
    Life sciences, 1995, Volume: 57, Issue:2

    Topics: Analgesics; Animals; Drug Interactions; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Injections, Subcutaneous; Male; Mice; Mice, Inbred Strains; Morphine; Naltrexone; Nociceptors; Oligopeptides; Quinolines; Receptors, Opioid, delta

1995
Effect of the highly selective and nonpeptide delta opioid receptor agonist TAN-67 on the morphine-induced place preference in mice.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 279, Issue:1

    Topics: Analgesics; Animals; Benzylidene Compounds; Dopamine; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Limbic System; Male; Mice; Morphine; Naltrexone; Quinolines; Receptors, Opioid, delta; Reward

1996
The third extracellular loop of the human delta-opioid receptor determines the selectivity of delta-opioid agonists.
    Molecular pharmacology, 1996, Volume: 50, Issue:6

    Topics: Amino Acid Sequence; Animals; COS Cells; Enkephalins; Humans; Molecular Sequence Data; Mutagenesis, Site-Directed; Oligopeptides; Quinolines; Receptors, Opioid, delta; Recombinant Fusion Proteins

1996
Delta-1 opioid receptor-mediated antinociceptive properties of a nonpeptidic delta opioid receptor agonist, (-)TAN-67, in the mouse spinal cord.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 280, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Hyperalgesia; Injections, Spinal; Male; Mice; Mice, Inbred ICR; Pain; Pain Measurement; Pyrrolidines; Quinolines; Reaction Time; Receptors, Opioid, delta; Spinal Cord

1997
Differential effects of mu-, delta- and kappa-opioid receptor agonists on the discriminative stimulus properties of cocaine in rats.
    European journal of pharmacology, 1997, Apr-11, Volume: 324, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Analysis of Variance; Animals; Cocaine; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Injections, Intraventricular; Male; Morphine; Narcotics; Pyrrolidines; Quinolines; Rats; Rats, Inbred F344; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Substance-Related Disorders

1997
Relative efficacies of delta-opioid receptor agonists at the cloned human delta-opioid receptor.
    European journal of pharmacology, 1997, May-12, Volume: 326, Issue:1

    Topics: Animals; Benzamides; CHO Cells; Cloning, Molecular; Cricetinae; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Naltrexone; Narcotic Antagonists; Piperazines; Quinolines; Receptors, Opioid, delta; Sulfur Radioisotopes

1997
Role of intracellular calcium in modification of mu and delta opioid receptor-mediated antinociception by diabetes in mice.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 286, Issue:2

    Topics: Analgesics; Analgesics, Opioid; Animals; Calcium; Calcium Chloride; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Egtazic Acid; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Injections, Intraventricular; Male; Mice; Mice, Inbred ICR; Pain Measurement; Quinolines; Receptors, Opioid, delta; Receptors, Opioid, mu; Ryanodine

1998
Delta-opioid receptor antagonists exhibit properties of partial delta-receptor agonists in isolated perfused heart.
    Bulletin of experimental biology and medicine, 2004, Volume: 138, Issue:4

    Topics: Animals; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Heart; In Vitro Techniques; Male; Myocardial Contraction; Myocardial Ischemia; Naltrexone; Oligopeptides; Perfusion; Quinolines; Rats; Rats, Wistar; Receptors, Opioid, delta

2004