enkephalin, leucine has been researched along with piperidines in 29 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 6 (20.69) | 18.7374 |
1990's | 6 (20.69) | 18.2507 |
2000's | 13 (44.83) | 29.6817 |
2010's | 4 (13.79) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Colpaert, FC; Janssen, PA; Niemegeers, CJ; Van Ree, JM | 1 |
Galt, RH | 1 |
Berkowitz, DS; Burt, SK; Loew, GH | 1 |
Connors, M; Rothberg, RM; Wainer, BH; Wung, WE | 1 |
Bilotta, JM; Brackeen, MF; Feldman, PL; James, MK; Leighton, HJ; Schuster, SV | 1 |
Bird, ED; Crino, PB; Plager, MD; Vogt, BA | 1 |
Candeletti, S; Ferri, S; Romualdi, P; Spadaro, C; Spampinato, S | 1 |
Casy, AF; Jin, WQ; Kosterlitz, HW; Paterson, SJ | 1 |
Dubrovina, NI | 2 |
Campana, G; Di Toro, R; Murari, G; Sciarretta, V; Spampinato, S | 1 |
Brain, SD; Towler, PK | 1 |
Maldonado, R; Valjent, E; Valverde, O; Zimmer, A; Zimmer, AM | 1 |
Andrén, PE; Gunne, L; Hurd, YL; Pirker, W; Pontén, H; Tedroff, J | 1 |
Bakalkin, G; Esashi, A; Kisara, K; Nakagawasai, O; Niijima, F; Sakurada, C; Sakurada, T; Tadano, T; Tan-No, K; Terenius, L | 1 |
Cox, ML; Welch, SP | 1 |
Gogus, N; Kabalak, AA; Senel, OO | 1 |
Bakalkin, G; Marinova, Z; Nakagawasai, O; Niijima, F; Sakurada, S; Sato, T; Satoh, S; Tadano, T; Takahashi, H; Tan-No, K; Terenius, L; Yakovleva, T | 1 |
Bédard, PJ; Calon, F; Di Paolo, T; Dridi, M; Hadj Tahar, A; Meltzer, LT; Morissette, M | 1 |
Franklin, SO; Gerald, TM; Howlett, AC; Ward, GR | 1 |
Ellgren, M; Hurd, YL; Spano, SM | 1 |
Deniau, JM; Kemel, ML; Pérez, S; Tierney, A | 1 |
Bilbao, A; Fernandez-Espejo, E; Ferrer, B; Gorriti, MA; Martín, AB; Moratalla, R; Navarro, M; Rodriguez de Fonseca, F | 1 |
de Miguel, R; Fernández-Ruiz, J; Maestro, B; Michael Walker, J; Ramos, JA; Rubio, M | 1 |
Cabañero, D; Célérier, E; García-Nogales, P; Maldonado, R; Mata, M; Puig, MM; Roques, BP | 1 |
Di Paolo, T; Grégoire, L; Lévesque, D; Morissette, M; Ouattara, B; Rouillard, C; Samadi, P; Tamim, MK | 1 |
Campillo, A; González-Cuello, A; Laorden, ML; Puig, MM; Romero, A; Romero-Alejo, E; Vasconcelos, N | 1 |
Bassirirad, NM; Davis, P; Deekonda, S; Hruby, VJ; Kulkarni, V; Lai, J; Largent-Milnes, TM; Porreca, F; Rankin, D; Vanderah, TW; Wang, Y; Wugalter, L | 1 |
BassiriRad, NM; Cole, J; Davis, P; Deekonda, S; Hruby, VJ; Lai, J; Largent-Milnes, TM; Porecca, F; Rankin, D; Sunna, S; Vanderah, TW | 1 |
1 review(s) available for enkephalin, leucine and piperidines
Article | Year |
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Structure-activity studies of narcotic agonists and antagonists from quantum chemical calculations.
Topics: Animals; Chemical Phenomena; Chemistry, Physical; Enkephalins; In Vitro Techniques; Methadone; Models, Molecular; Molecular Conformation; Nalorphine; Narcotic Antagonists; Narcotics; Oxymorphone; Piperidines; Quantum Theory; Receptors, Opioid; Structure-Activity Relationship; Thermodynamics | 1978 |
28 other study(ies) available for enkephalin, leucine and piperidines
Article | Year |
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Narcotic cueing properties of intraventricularly administered sufentanil, fentanyl, morphine and met-enkephalin.
Topics: Analgesics, Opioid; Anilides; Animals; Cues; Dose-Response Relationship, Drug; Endorphins; Enkephalins; Fentanyl; Injections, Intraventricular; Morphine; Piperidines; Rats; Time Factors | 1978 |
The opiate anomalies--another possible explanation?
Topics: Benzomorphans; Chemical Phenomena; Chemistry; Enkephalins; Fentanyl; Narcotics; Piperidines; Receptors, Opioid; Structure-Activity Relationship | 1977 |
The specificity of antimorphine and antimeperidine antibodies and their reactivity with opioid peptides.
Topics: Antibody Specificity; Binding, Competitive; Cross Reactions; Drug Stability; Endorphins; Enkephalins; Immunoglobulin G; Meperidine; Molecular Conformation; Morphine; Piperidines | 1979 |
Opioid receptor activity of GI 87084B, a novel ultra-short acting analgesic, in isolated tissues.
Topics: Alkylation; Animals; Enkephalin, Leucine; Guinea Pigs; Ileum; Kinetics; Male; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle, Smooth; Naloxone; Naltrexone; Narcotic Antagonists; Piperidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Remifentanil; Vas Deferens | 1991 |
Laminar distributions of muscarinic acetylcholine, serotonin, GABA and opioid receptors in human posterior cingulate cortex.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aged; Autoradiography; Cerebral Cortex; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Female; Humans; Iodocyanopindolol; Ketanserin; Male; Middle Aged; Oxotremorine; Paroxetine; Pindolol; Piperidines; Pirenzepine; Receptors, Cell Surface; Receptors, Cholinergic; Receptors, GABA-A; Receptors, Muscarinic; Receptors, Opioid; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes | 1990 |
Studies on the antinociceptive effect of intrathecal salmon calcitonin.
Topics: Analgesics; Animals; Benzomorphans; Calcitonin; Enkephalin, Leucine; Haloperidol; Ketanserin; Male; Methysergide; Nociceptors; Phentolamine; Piperidines; Rats; Receptors, Opioid | 1985 |
Interactions of some 4-anilinopiperidines and 4-phenylpiperidines with the mu, delta- and kappa-binding sites.
Topics: Animals; Brain; Enkephalins; Guinea Pigs; Male; Piperidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1983 |
[Contribution of dopamine autoreceptors in the reactive effect of opioid antagonists].
Topics: Animals; Avoidance Learning; Dopamine Agonists; Enkephalin, Leucine; Male; Mice; Mice, Inbred BALB C; Naloxone; Narcotic Antagonists; Piperidines; Receptors, Dopamine; Receptors, Opioid, delta; Receptors, Opioid, mu | 1995 |
Dopamine and opioid regulation of the memory retrieval recovery in mice.
Topics: Animals; Avoidance Learning; Dopamine Agonists; Enkephalin, Leucine; Male; Memory; Mice; Mice, Inbred BALB C; Narcotic Antagonists; Piperidines; Quinpirole; Receptors, Dopamine D2; Receptors, Opioid, delta | 1996 |
Regulation of delta opioid receptors by delta9-tetrahydrocannabinol in NG108-15 hybrid cells.
Topics: Animals; Colforsin; Dose-Response Relationship, Drug; Dronabinol; Enkephalin, Leucine; Glioma; Mice; Neuroblastoma; Piperidines; Pyrazoles; Rats; Receptors, Opioid, delta; Rimonabant; RNA, Messenger; Tumor Cells, Cultured | 1998 |
Activity of tachykinin NK1 and bradykinin B2 receptor antagonists, and an opioid ligand at different stimulation parameters in neurogenic inflammation in the rat.
Topics: Animals; Bradykinin; Bradykinin Receptor Antagonists; Edema; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Extravasation of Diagnostic and Therapeutic Materials; Male; Neurogenic Inflammation; Neurokinin-1 Receptor Antagonists; Neurons, Afferent; Peptide Fragments; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptor, Bradykinin B2; Receptors, Neurokinin-1; Receptors, Opioid, mu; Substance P; Time Factors | 1998 |
Cannabinoid withdrawal syndrome is reduced in pre-proenkephalin knock-out mice.
Topics: Acute Disease; Analysis of Variance; Animals; Autoradiography; Behavior, Animal; Body Temperature; Body Weight; Brain; Chronic Disease; Dronabinol; Drug Tolerance; Enkephalins; Hyperalgesia; Mice; Mice, Inbred C57BL; Mice, Knockout; Piperidines; Protein Precursors; Psychotropic Drugs; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Substance Withdrawal Syndrome | 2000 |
Coadministration of (-)-OSU6162 with l-DOPA normalizes preproenkephalin mRNA expression in the sensorimotor striatum of primates with unilateral 6-OHDA lesions.
Topics: Animals; Autoradiography; Callithrix; Caudate Nucleus; Corpus Striatum; Disease Models, Animal; Dopamine Agents; Drug Administration Schedule; Drug Therapy, Combination; Enkephalins; Female; In Situ Hybridization; Injections, Subcutaneous; Levodopa; Ligands; Male; Oxidopamine; Parkinson Disease, Secondary; Piperidines; Protein Precursors; Putamen; RNA, Messenger; Tritium | 2001 |
Intrathecally administered big dynorphin, a prodynorphin-derived peptide, produces nociceptive behavior through an N-methyl-D-aspartate receptor mechanism.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Analgesics, Opioid; Animals; Behavior, Animal; Dizocilpine Maleate; Dynorphins; Endorphins; Enkephalins; Excitatory Amino Acid Antagonists; Injections, Spinal; Kynurenic Acid; Male; Mice; Morphine; Neurokinin A; Nociceptors; Peptide Fragments; Piperidines; Protein Precursors; Receptors, N-Methyl-D-Aspartate; Receptors, Tachykinin; Substance P | 2002 |
The antinociceptive effect of Delta9-tetrahydrocannabinol in the arthritic rat.
Topics: Animals; Arthritis, Experimental; Cannabinoid Receptor Antagonists; Dose-Response Relationship, Drug; Dronabinol; Dynorphins; Enkephalin, Leucine; Enkephalin, Methionine; Freund's Adjuvant; Injections, Intradermal; Injections, Intraperitoneal; Male; Morphine; Mycobacterium; Naloxone; Naltrexone; Narcotic Antagonists; Pain; Pain Measurement; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Opioid; Rimonabant | 2004 |
The effects of transcranial electrical stimulation on opiate-induced analgesia in rats.
Topics: Analgesia; Analgesics, Opioid; Animals; Brain; Electric Stimulation; Enkephalins; Magnetics; Male; Pain Threshold; Piperidines; Rats; Rats, Wistar; Remifentanil | 2004 |
Pronociceptive role of dynorphins in uninjured animals: N-ethylmaleimide-induced nociceptive behavior mediated through inhibition of dynorphin degradation.
Topics: Agmatine; Analysis of Variance; Animals; Behavior, Animal; Biguanides; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Interactions; Dynorphins; Enkephalins; Enzyme Inhibitors; Ethylmaleimide; Excitatory Amino Acid Antagonists; Immune Sera; Injections, Spinal; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Morphine; Narcotics; Nociceptin Receptor; Piperidines; Protein Precursors; Receptors, Opioid; Spinal Cord; Time Factors | 2005 |
Prevention of levodopa-induced dyskinesias by a selective NR1A/2B N-methyl-D-aspartate receptor antagonist in parkinsonian monkeys: implication of preproenkephalin.
Topics: Animals; Antiparkinson Agents; Benserazide; Benzoxazoles; Corpus Striatum; Dopamine; Drug Therapy, Combination; Dyskinesia, Drug-Induced; Enkephalins; Female; Gene Expression; Levodopa; Macaca fascicularis; Parkinsonian Disorders; Piperidines; Protein Precursors; Receptors, N-Methyl-D-Aspartate; RNA, Messenger | 2006 |
CB1 knockout mice display significant changes in striatal opioid peptide and D4 dopamine receptor gene expression.
Topics: Animals; Corpus Striatum; Dynorphins; Enkephalins; Gene Expression; Mice; Mice, Knockout; Opioid Peptides; Piperidines; Protein Precursors; Pyrazoles; Receptor, Cannabinoid, CB1; Receptors, Dopamine D2; Receptors, Dopamine D4; Reverse Transcriptase Polymerase Chain Reaction; Rimonabant; RNA, Messenger | 2006 |
Adolescent cannabis exposure alters opiate intake and opioid limbic neuronal populations in adult rats.
Topics: Analgesics, Non-Narcotic; Analgesics, Opioid; Analysis of Variance; Animals; Animals, Newborn; Benzoxazines; Dose-Response Relationship, Drug; Dronabinol; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Gene Expression Regulation; Guanosine 5'-O-(3-Thiotriphosphate); Heroin; In Situ Hybridization; Limbic System; Male; Morpholines; Naphthalenes; Neurons; Piperidines; Protein Precursors; Pyrazoles; Radioligand Assay; Rats; Rats, Long-Evans; Reinforcement, Psychology; Rimonabant; Self Administration; Sulfur Isotopes; Tritium | 2007 |
Tachykinin regulation of cholinergic transmission in the limbic/prefrontal territory of the rat dorsal striatum: implication of new neurokinine 1-sensitive receptor binding site and interaction with enkephalin/mu opioid receptor transmission.
Topics: Acetylcholine; Animals; Binding Sites; Binding, Competitive; Cholinergic Fibers; Circadian Rhythm; Enkephalins; Limbic System; Male; Morpholines; Narcotic Antagonists; Neostriatum; Neural Pathways; Neurokinin-1 Receptor Antagonists; Organ Culture Techniques; Piperidines; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Receptors, Opioid, mu; Synaptic Transmission; Tachykinins | 2007 |
Expression and function of CB1 receptor in the rat striatum: localization and effects on D1 and D2 dopamine receptor-mediated motor behaviors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Arachidonic Acids; Behavior, Animal; Corpus Striatum; Dopamine Agonists; Enkephalins; Gene Expression Regulation; Grooming; Male; Models, Biological; Motor Activity; Movement; Nerve Tissue Proteins; Neurons; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Dopamine D1; Receptors, Dopamine D2; Rimonabant; Substance P | 2008 |
CB1 receptor blockade reduces the anxiogenic-like response and ameliorates the neurochemical imbalances associated with alcohol withdrawal in rats.
Topics: Animals; Anxiety; Appetite; Arachidonic Acids; Autoradiography; Benzoxazines; Brain Chemistry; Cannabinoid Receptor Modulators; Central Nervous System Depressants; Chromatography, High Pressure Liquid; Emotions; Endocannabinoids; Enkephalins; Ethanol; Ethanolamines; Glycerides; In Situ Hybridization; Male; Morpholines; Motor Activity; Naphthalenes; Neuropeptide Y; Neurotransmitter Agents; Piperidines; Polyunsaturated Alkamides; Protein Precursors; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Rimonabant; RNA, Messenger; Stress, Psychological; Substance Withdrawal Syndrome | 2008 |
The pro-nociceptive effects of remifentanil or surgical injury in mice are associated with a decrease in delta-opioid receptor mRNA levels: Prevention of the nociceptive response by on-site delivery of enkephalins.
Topics: Analgesics; Animals; Disease Models, Animal; Disulfides; Down-Regulation; Enkephalins; Ganglia, Spinal; Male; Methyl Ethers; Mice; Pain Measurement; Pain Threshold; Pain, Postoperative; Phenylalanine; Piperidines; Protein Precursors; Receptors, Opioid, delta; Receptors, Opioid, mu; Remifentanil; RNA, Messenger; Sevoflurane; Spinal Cord; Time Factors | 2009 |
Effect of non-dopaminergic drug treatment on Levodopa induced dyskinesias in MPTP monkeys: common implication of striatal neuropeptides.
Topics: Animals; Antiparkinson Agents; Benzoxazoles; Cocaine; Corpus Striatum; Disease Models, Animal; Docosahexaenoic Acids; Dopamine; Dopamine Uptake Inhibitors; Dynorphins; Dyskinesia, Drug-Induced; Enkephalins; Female; Iodine Isotopes; Levodopa; Macaca fascicularis; Naltrexone; Neuropeptides; Ovariectomy; Parkinsonian Disorders; Piperidines; Protein Precursors; RNA, Messenger; Sulfonamides; Tachykinins; Thiazoles; Time Factors | 2010 |
Effects of surgery and/or remifentanil administration on the expression of pERK1/2, c-Fos and dynorphin in the dorsal root ganglia in mice.
Topics: Analgesics, Opioid; Animals; Behavior, Animal; Dynorphins; Enkephalins; Ganglia, Spinal; Hyperalgesia; Male; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Pain, Postoperative; Piperidines; Protein Precursors; Proto-Oncogene Proteins c-fos; Remifentanil; RNA, Messenger | 2012 |
Design and synthesis of novel bivalent ligands (MOR and DOR) by conjugation of enkephalin analogues with 4-anilidopiperidine derivatives.
Topics: Analgesics; Animals; Dose-Response Relationship, Drug; Drug Design; Enkephalins; Guinea Pigs; Ligands; Mice; Molecular Conformation; Muscle Contraction; Pain Measurement; Pain Threshold; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid; Structure-Activity Relationship | 2015 |
Enkephalin analogues with N-phenyl-N-(piperidin-2-ylmethyl)propionamide derivatives: Synthesis and biological evaluations.
Topics: Amides; Analgesics; Animals; Dose-Response Relationship, Drug; Enkephalins; Guinea Pigs; Humans; Ileum; Ligands; Mice; Molecular Structure; Pain; Piperidines; Rats; Receptors, Opioid, delta; Receptors, Opioid, mu; Structure-Activity Relationship | 2016 |