enkephalin, leucine and diazepam

enkephalin, leucine has been researched along with diazepam in 26 studies

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-199014 (53.85)18.7374
1990's7 (26.92)18.2507
2000's3 (11.54)29.6817
2010's1 (3.85)24.3611
2020's1 (3.85)2.80

Authors

AuthorsStudies
Jia, Q; Sun, S; Zhang, Z1
Carmona, AV; Kumari, S; Tiwari, AK; Trippier, PC1
Goodwin, FK; Greenlaw, P; Marangos, PJ; Paul, SM; Skolnick, P1
Chance, WT; Krynock, GM; Rosecrans, JA; White, AC1
Duka, T; Herz, A; Wüster, M4
Andrews, N; File, SE; Rattray, M; Singhvi, S; Wu, PY1
Giros, B; Llorens-Cortes, C; Quach, TT; Schwartz, JC1
Giros, B; Llorens-Cortes, C; Quach, TT; Schwartz, JC; Van Amsterdam, JG1
Costa, E; Mocchetti, I1
Noble, EP; Noble, L; Ritchie, T; Syapin, PJ1
Bortolotto, ZA; Cavalheiro, EA; Ikonomidou-Turski, C; Turski, L; Turski, WA1
Jackson, HC; Sewell, RD1
Coletti-Previero, MA; Mattras, H; Previero, A1
Ito, J; Matsuoka, I; Sasa, M; Takahashi, H; Takaori, S1
Glebov, RN; Kaplun, AP; Kryzhanovskiĭ, GN; Maloletneva, OIu; Nikushkin, EV1
Fratta, W; Gessa, GL; Rossetti, Z1
Ansell, RJ; Mosbach, K; Ramström, O1
Lucas, LR; McEwen, BS; Pompei, P1
Satyapriya, A; Sheu, MJ; Sribanditmongkol, P; Tejwani, GA1
Kang, W; Wilson, MA; Wilson, SP2
Davies, A; Dominguez, M; Morrison, D; Mortishire-Smith, R; O'Connor, D1
Mascagni, F; McDonald, AJ; Primeaux, SD; Wilson, MA; Wilson, SP1

Reviews

4 review(s) available for enkephalin, leucine and diazepam

ArticleYear
Applications of amide isosteres in medicinal chemistry.
    Bioorganic & medicinal chemistry letters, 2019, 09-15, Volume: 29, Issue:18

    Topics: Amides; Chemistry, Pharmaceutical; Drug Design; Molecular Structure

2019
Amide Bond Bioisosteres: Strategies, Synthesis, and Successes.
    Journal of medicinal chemistry, 2020, 11-12, Volume: 63, Issue:21

    Topics: Amides; Carbamates; Click Chemistry; Drug Design; Pyridines; Structure-Activity Relationship; Triazoles; Urea

2020
In vivo studies of the regulation of neuropeptide stores in structures of the rat brain.
    Neuropharmacology, 1987, Volume: 26, Issue:7B

    Topics: Animals; Brain; Brain Chemistry; Chlorides; Diazepam; DNA; Drug Tolerance; Enkephalins; Haloperidol; Morphine; Neuropeptides; Nucleic Acid Hybridization; Pro-Opiomelanocortin; Protein Precursors; Receptors, Dopamine; Receptors, GABA-A; RNA, Messenger

1987
Experimental vestibular pharmacology: a minireview with special reference to neuroactive substances and antivertigo drugs.
    Acta oto-laryngologica. Supplementum, 1984, Volume: 419

    Topics: Acetylcholine; Action Potentials; Animals; Atropine; Cats; Diazepam; Dopamine; Enkephalins; Ethanol; gamma-Aminobutyric Acid; Histamine; Norepinephrine; Serotonin; Vasodilator Agents; Vertigo; Vestibular Nerve; Vestibular Nuclei

1984

Other Studies

22 other study(ies) available for enkephalin, leucine and diazepam

ArticleYear
Demonstration of an endogenous, competitive inhibitor(s) of [3H] diazepam binding in bovine brain.
    Life sciences, 1978, Jun-05, Volume: 22, Issue:21

    Topics: Alprenolol; Animals; Binding, Competitive; Brain; Cattle; Chromatography, Thin Layer; Diazepam; Enkephalins; In Vitro Techniques; Kinetics; Molecular Weight; Receptors, Adrenergic, beta; Receptors, Opioid

1978
Autoanalgesia: acquisition, blockade and relationship to opiate binding.
    European journal of pharmacology, 1979, Oct-15, Volume: 58, Issue:4

    Topics: Analgesia; Animals; Brain; Conditioning, Classical; Diazepam; Enkephalins; Etorphine; In Vitro Techniques; Male; Naltrexone; Narcotics; Rats; Reaction Time; Spinal Cord

1979
Rapid changes in enkephalin levels in rat striatum and hypothalamus induced by diazepam.
    Naunyn-Schmiedeberg's archives of pharmacology, 1979, Volume: 309, Issue:1

    Topics: Animals; Brain Chemistry; Corpus Striatum; Diazepam; Endorphins; Enkephalins; Hypothalamus; Male; Rats; Time Factors

1979
Regulation of glutamate decarboxylase and enkephalin mRNA levels in rat striatum by chronic benzodiazepine treatment.
    Biochemical Society transactions, 1992, Volume: 20, Issue:3

    Topics: Animals; Base Sequence; Brain; Corpus Striatum; Diazepam; Drug Administration Schedule; Enkephalins; Glutamate Decarboxylase; Kinetics; Molecular Sequence Data; Oligodeoxyribonucleotides; Protein Precursors; Rats; Reference Values; Substance Withdrawal Syndrome

1992
Adaptative changes in two indices of enkephalin neuron activity in mouse striatum following GABAergic stimulation.
    Progress in clinical and biological research, 1990, Volume: 328

    Topics: Animals; Corpus Striatum; Diazepam; Enkephalins; gamma-Aminobutyric Acid; Male; Mice; Muscimol; Oligopeptides; Protein Precursors; Receptors, GABA-A; RNA, Messenger

1990
Enkephalin biosynthesis and release in mouse striatum are inhibited by GABA receptor stimulation: compared changes in preproenkephalin mRNA and Tyr-Gly-Gly levels.
    Brain research. Molecular brain research, 1990, Volume: 8, Issue:3

    Topics: Aminooxyacetic Acid; Animals; Corpus Striatum; Diazepam; Enkephalins; Flumazenil; Kinetics; Leucine; Male; Mice; Muscimol; Oligopeptides; Protein Precursors; Receptors, GABA-A; RNA, Messenger

1990
Postmortem changes in rat brain: studies on membrane-bound enzymes and receptors.
    Journal of neurochemistry, 1987, Volume: 48, Issue:4

    Topics: Animals; Brain; Ca(2+) Mg(2+)-ATPase; Calcium-Transporting ATPases; Cell Membrane; Diazepam; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Female; Male; Naloxone; Postmortem Changes; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Neurotransmitter; Receptors, Opioid; Sodium-Potassium-Exchanging ATPase; Succinates

1987
Convulsant action of morphine, [D-Ala2, D-Leu5]-enkephalin and naloxone in the rat amygdala: electroencephalographic, morphological and behavioural sequelae.
    Neuroscience, 1987, Volume: 20, Issue:2

    Topics: Amygdala; Animals; Brain; Convulsants; Diazepam; Drug Interactions; Electroencephalography; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Male; Microinjections; Morphine; Naloxone; Rats; Rats, Inbred Strains

1987
Involvement of endogenous enkephalins in the feeding response to diazepam.
    European journal of pharmacology, 1985, Jan-08, Volume: 107, Issue:3

    Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Eating; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Male; Rats; Rats, Inbred Strains

1985
beta-Carboline and diazepam effect on the degradation of enkephalin by the human blood aminopeptidase.
    Bioscience reports, 1983, Volume: 3, Issue:1

    Topics: Aminopeptidases; Carbolines; Diazepam; Enkephalin, Leucine; Humans; In Vitro Techniques; Indoles; Receptors, Cell Surface; Receptors, GABA-A; Structure-Activity Relationship

1983
[Effect of neurotropic compounds on the transmembrane potential of synaptosomes].
    Biulleten' eksperimental'noi biologii i meditsiny, 1983, Volume: 96, Issue:9

    Topics: Animals; Cerebral Cortex; Chlorpromazine; Colchicine; Cytochalasin B; Diazepam; Enkephalin, Leucine; Enkephalin, Methionine; Haloperidol; Imipramine; Membrane Potentials; Peptides; Psychotropic Drugs; Rats; Synaptosomes; Trifluoperazine; Tuftsin

1983
Diazepam-induced release of opioid activity in the rat brain.
    Neuroscience letters, 1980, Volume: 16, Issue:3

    Topics: Analgesics; Animals; Bacitracin; Brain; Diazepam; Enkephalins; Male; Pain; Rats; Rats, Inbred Strains; Sensory Thresholds

1980
Rapid depletion and restoration of striatal met-enkephalin after ketamine.
    Life sciences, 1981, Jul-06, Volume: 29, Issue:1

    Topics: Animals; Corpus Striatum; Diazepam; Drug Interactions; Endorphins; Enkephalin, Methionine; Enkephalins; Ketamine; Male; Rats

1981
Benzodiazepines modulate striatal enkephalin levels via a GABAergic mechanism.
    Life sciences, 1980, Mar-10, Volume: 26, Issue:10

    Topics: Aminooxyacetic Acid; Animals; Bicuculline; Corpus Striatum; Diazepam; Endorphins; Enkephalin, Methionine; Enkephalins; Fentanyl; gamma-Aminobutyric Acid; Hypothalamus; Male; Muscimol; Radioimmunoassay; Rats

1980
Diazepam effects on striatal met-enkephalin levels following long-term pharmacological manipulations.
    Neuropharmacology, 1980, Volume: 19, Issue:6

    Topics: Animals; Corpus Striatum; Diazepam; Endorphins; Enkephalin, Methionine; Enkephalins; Flunitrazepam; Male; Rats

1980
Towards artificial antibodies prepared by molecular imprinting.
    Clinical chemistry, 1996, Volume: 42, Issue:9

    Topics: Antibodies; Atrazine; Binding, Competitive; Corticosterone; Cross Reactions; Diazepam; Enkephalin, Leucine; Enzyme-Linked Immunosorbent Assay; Humans; Hydrocortisone; Kinetics; Methylglucosides; Molecular Mimicry; Morphine; Polymers; Propranolol; Radioimmunoassay; Stereoisomerism; Theophylline; Yohimbine

1996
Effects of deoxycorticosterone acetate and diazepam on neuropeptidergic neurons in rat striatum.
    Neuroreport, 1997, Mar-03, Volume: 8, Issue:4

    Topics: Analysis of Variance; Animals; Appetite; Corpus Striatum; Desoxycorticosterone; Diazepam; Dynorphins; Enkephalins; Male; Neurons; Protein Precursors; Rats; Rats, Sprague-Dawley; RNA, Messenger; Sodium, Dietary; Tachykinins; Transcription, Genetic

1997
Inhibition of morphine tolerance and dependence by diazepam and its relation to mu-opioid receptors in the rat brain and spinal cord.
    Brain research, 1998, Jun-29, Volume: 797, Issue:2

    Topics: Analgesics, Opioid; Animals; Binding, Competitive; Brain Chemistry; Central Nervous System; Diazepam; Drug Interactions; Drug Tolerance; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Hypnotics and Sedatives; Male; Morphine; Naloxone; Narcotic Antagonists; Nociceptors; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Substance Withdrawal Syndrome; Tritium

1998
Changes in nociceptive and anxiolytic responses following herpes virus-mediated preproenkephalin overexpression in rat amygdala are naloxone-reversible and transient.
    Annals of the New York Academy of Sciences, 1999, Jun-29, Volume: 877

    Topics: Amygdala; Animals; Anti-Anxiety Agents; beta-Galactosidase; Diazepam; Enkephalins; Gene Expression Regulation; Genetic Vectors; Herpesviridae; Humans; Male; Maze Learning; Naloxone; Pain; Pain Measurement; Protein Precursors; Rats; Recombinant Proteins; RNA, Messenger; Transcription, Genetic

1999
Overexpression of proenkephalin in the amygdala potentiates the anxiolytic effects of benzodiazepines.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2000, Volume: 22, Issue:1

    Topics: Amygdala; Analysis of Variance; Animals; Anti-Anxiety Agents; beta-Galactosidase; Defective Viruses; Diazepam; DNA, Complementary; Enkephalins; Gene Transfer Techniques; Herpesvirus 4, Human; Humans; In Situ Hybridization; Maze Learning; Naloxone; Protein Precursors; Rats; Rats, Long-Evans; RNA, Messenger

2000
Ultra-performance liquid chromatography coupled to time-of-flight mass spectrometry for robust, high-throughput quantitative analysis of an automated metabolic stability assay, with simultaneous determination of metabolic data.
    Rapid communications in mass spectrometry : RCM, 2006, Volume: 20, Issue:5

    Topics: Animals; Chromatography, High Pressure Liquid; Diazepam; Drug Evaluation, Preclinical; Drug Stability; Enkephalin, Leucine; Imipramine; Neurotransmitter Agents; Psychotropic Drugs; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Sensitivity and Specificity; Spectrometry, Mass, Electrospray Ionization

2006
The role of delta opioid receptors in the anxiolytic actions of benzodiazepines.
    Pharmacology, biochemistry, and behavior, 2006, Volume: 85, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Enkephalins; Male; Maze Learning; Naltrexone; Rats; Rats, Long-Evans; Receptors, GABA-A; Receptors, Opioid, delta

2006