enkephalin, leucine has been researched along with diazepam in 26 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 14 (53.85) | 18.7374 |
1990's | 7 (26.92) | 18.2507 |
2000's | 3 (11.54) | 29.6817 |
2010's | 1 (3.85) | 24.3611 |
2020's | 1 (3.85) | 2.80 |
Authors | Studies |
---|---|
Jia, Q; Sun, S; Zhang, Z | 1 |
Carmona, AV; Kumari, S; Tiwari, AK; Trippier, PC | 1 |
Goodwin, FK; Greenlaw, P; Marangos, PJ; Paul, SM; Skolnick, P | 1 |
Chance, WT; Krynock, GM; Rosecrans, JA; White, AC | 1 |
Duka, T; Herz, A; Wüster, M | 4 |
Andrews, N; File, SE; Rattray, M; Singhvi, S; Wu, PY | 1 |
Giros, B; Llorens-Cortes, C; Quach, TT; Schwartz, JC | 1 |
Giros, B; Llorens-Cortes, C; Quach, TT; Schwartz, JC; Van Amsterdam, JG | 1 |
Costa, E; Mocchetti, I | 1 |
Noble, EP; Noble, L; Ritchie, T; Syapin, PJ | 1 |
Bortolotto, ZA; Cavalheiro, EA; Ikonomidou-Turski, C; Turski, L; Turski, WA | 1 |
Jackson, HC; Sewell, RD | 1 |
Coletti-Previero, MA; Mattras, H; Previero, A | 1 |
Ito, J; Matsuoka, I; Sasa, M; Takahashi, H; Takaori, S | 1 |
Glebov, RN; Kaplun, AP; Kryzhanovskiĭ, GN; Maloletneva, OIu; Nikushkin, EV | 1 |
Fratta, W; Gessa, GL; Rossetti, Z | 1 |
Ansell, RJ; Mosbach, K; Ramström, O | 1 |
Lucas, LR; McEwen, BS; Pompei, P | 1 |
Satyapriya, A; Sheu, MJ; Sribanditmongkol, P; Tejwani, GA | 1 |
Kang, W; Wilson, MA; Wilson, SP | 2 |
Davies, A; Dominguez, M; Morrison, D; Mortishire-Smith, R; O'Connor, D | 1 |
Mascagni, F; McDonald, AJ; Primeaux, SD; Wilson, MA; Wilson, SP | 1 |
4 review(s) available for enkephalin, leucine and diazepam
Article | Year |
---|---|
Applications of amide isosteres in medicinal chemistry.
Topics: Amides; Chemistry, Pharmaceutical; Drug Design; Molecular Structure | 2019 |
Amide Bond Bioisosteres: Strategies, Synthesis, and Successes.
Topics: Amides; Carbamates; Click Chemistry; Drug Design; Pyridines; Structure-Activity Relationship; Triazoles; Urea | 2020 |
In vivo studies of the regulation of neuropeptide stores in structures of the rat brain.
Topics: Animals; Brain; Brain Chemistry; Chlorides; Diazepam; DNA; Drug Tolerance; Enkephalins; Haloperidol; Morphine; Neuropeptides; Nucleic Acid Hybridization; Pro-Opiomelanocortin; Protein Precursors; Receptors, Dopamine; Receptors, GABA-A; RNA, Messenger | 1987 |
Experimental vestibular pharmacology: a minireview with special reference to neuroactive substances and antivertigo drugs.
Topics: Acetylcholine; Action Potentials; Animals; Atropine; Cats; Diazepam; Dopamine; Enkephalins; Ethanol; gamma-Aminobutyric Acid; Histamine; Norepinephrine; Serotonin; Vasodilator Agents; Vertigo; Vestibular Nerve; Vestibular Nuclei | 1984 |
22 other study(ies) available for enkephalin, leucine and diazepam
Article | Year |
---|---|
Demonstration of an endogenous, competitive inhibitor(s) of [3H] diazepam binding in bovine brain.
Topics: Alprenolol; Animals; Binding, Competitive; Brain; Cattle; Chromatography, Thin Layer; Diazepam; Enkephalins; In Vitro Techniques; Kinetics; Molecular Weight; Receptors, Adrenergic, beta; Receptors, Opioid | 1978 |
Autoanalgesia: acquisition, blockade and relationship to opiate binding.
Topics: Analgesia; Animals; Brain; Conditioning, Classical; Diazepam; Enkephalins; Etorphine; In Vitro Techniques; Male; Naltrexone; Narcotics; Rats; Reaction Time; Spinal Cord | 1979 |
Rapid changes in enkephalin levels in rat striatum and hypothalamus induced by diazepam.
Topics: Animals; Brain Chemistry; Corpus Striatum; Diazepam; Endorphins; Enkephalins; Hypothalamus; Male; Rats; Time Factors | 1979 |
Regulation of glutamate decarboxylase and enkephalin mRNA levels in rat striatum by chronic benzodiazepine treatment.
Topics: Animals; Base Sequence; Brain; Corpus Striatum; Diazepam; Drug Administration Schedule; Enkephalins; Glutamate Decarboxylase; Kinetics; Molecular Sequence Data; Oligodeoxyribonucleotides; Protein Precursors; Rats; Reference Values; Substance Withdrawal Syndrome | 1992 |
Adaptative changes in two indices of enkephalin neuron activity in mouse striatum following GABAergic stimulation.
Topics: Animals; Corpus Striatum; Diazepam; Enkephalins; gamma-Aminobutyric Acid; Male; Mice; Muscimol; Oligopeptides; Protein Precursors; Receptors, GABA-A; RNA, Messenger | 1990 |
Enkephalin biosynthesis and release in mouse striatum are inhibited by GABA receptor stimulation: compared changes in preproenkephalin mRNA and Tyr-Gly-Gly levels.
Topics: Aminooxyacetic Acid; Animals; Corpus Striatum; Diazepam; Enkephalins; Flumazenil; Kinetics; Leucine; Male; Mice; Muscimol; Oligopeptides; Protein Precursors; Receptors, GABA-A; RNA, Messenger | 1990 |
Postmortem changes in rat brain: studies on membrane-bound enzymes and receptors.
Topics: Animals; Brain; Ca(2+) Mg(2+)-ATPase; Calcium-Transporting ATPases; Cell Membrane; Diazepam; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Female; Male; Naloxone; Postmortem Changes; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Neurotransmitter; Receptors, Opioid; Sodium-Potassium-Exchanging ATPase; Succinates | 1987 |
Convulsant action of morphine, [D-Ala2, D-Leu5]-enkephalin and naloxone in the rat amygdala: electroencephalographic, morphological and behavioural sequelae.
Topics: Amygdala; Animals; Brain; Convulsants; Diazepam; Drug Interactions; Electroencephalography; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Male; Microinjections; Morphine; Naloxone; Rats; Rats, Inbred Strains | 1987 |
Involvement of endogenous enkephalins in the feeding response to diazepam.
Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Eating; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Male; Rats; Rats, Inbred Strains | 1985 |
beta-Carboline and diazepam effect on the degradation of enkephalin by the human blood aminopeptidase.
Topics: Aminopeptidases; Carbolines; Diazepam; Enkephalin, Leucine; Humans; In Vitro Techniques; Indoles; Receptors, Cell Surface; Receptors, GABA-A; Structure-Activity Relationship | 1983 |
[Effect of neurotropic compounds on the transmembrane potential of synaptosomes].
Topics: Animals; Cerebral Cortex; Chlorpromazine; Colchicine; Cytochalasin B; Diazepam; Enkephalin, Leucine; Enkephalin, Methionine; Haloperidol; Imipramine; Membrane Potentials; Peptides; Psychotropic Drugs; Rats; Synaptosomes; Trifluoperazine; Tuftsin | 1983 |
Diazepam-induced release of opioid activity in the rat brain.
Topics: Analgesics; Animals; Bacitracin; Brain; Diazepam; Enkephalins; Male; Pain; Rats; Rats, Inbred Strains; Sensory Thresholds | 1980 |
Rapid depletion and restoration of striatal met-enkephalin after ketamine.
Topics: Animals; Corpus Striatum; Diazepam; Drug Interactions; Endorphins; Enkephalin, Methionine; Enkephalins; Ketamine; Male; Rats | 1981 |
Benzodiazepines modulate striatal enkephalin levels via a GABAergic mechanism.
Topics: Aminooxyacetic Acid; Animals; Bicuculline; Corpus Striatum; Diazepam; Endorphins; Enkephalin, Methionine; Enkephalins; Fentanyl; gamma-Aminobutyric Acid; Hypothalamus; Male; Muscimol; Radioimmunoassay; Rats | 1980 |
Diazepam effects on striatal met-enkephalin levels following long-term pharmacological manipulations.
Topics: Animals; Corpus Striatum; Diazepam; Endorphins; Enkephalin, Methionine; Enkephalins; Flunitrazepam; Male; Rats | 1980 |
Towards artificial antibodies prepared by molecular imprinting.
Topics: Antibodies; Atrazine; Binding, Competitive; Corticosterone; Cross Reactions; Diazepam; Enkephalin, Leucine; Enzyme-Linked Immunosorbent Assay; Humans; Hydrocortisone; Kinetics; Methylglucosides; Molecular Mimicry; Morphine; Polymers; Propranolol; Radioimmunoassay; Stereoisomerism; Theophylline; Yohimbine | 1996 |
Effects of deoxycorticosterone acetate and diazepam on neuropeptidergic neurons in rat striatum.
Topics: Analysis of Variance; Animals; Appetite; Corpus Striatum; Desoxycorticosterone; Diazepam; Dynorphins; Enkephalins; Male; Neurons; Protein Precursors; Rats; Rats, Sprague-Dawley; RNA, Messenger; Sodium, Dietary; Tachykinins; Transcription, Genetic | 1997 |
Inhibition of morphine tolerance and dependence by diazepam and its relation to mu-opioid receptors in the rat brain and spinal cord.
Topics: Analgesics, Opioid; Animals; Binding, Competitive; Brain Chemistry; Central Nervous System; Diazepam; Drug Interactions; Drug Tolerance; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Hypnotics and Sedatives; Male; Morphine; Naloxone; Narcotic Antagonists; Nociceptors; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Substance Withdrawal Syndrome; Tritium | 1998 |
Changes in nociceptive and anxiolytic responses following herpes virus-mediated preproenkephalin overexpression in rat amygdala are naloxone-reversible and transient.
Topics: Amygdala; Animals; Anti-Anxiety Agents; beta-Galactosidase; Diazepam; Enkephalins; Gene Expression Regulation; Genetic Vectors; Herpesviridae; Humans; Male; Maze Learning; Naloxone; Pain; Pain Measurement; Protein Precursors; Rats; Recombinant Proteins; RNA, Messenger; Transcription, Genetic | 1999 |
Overexpression of proenkephalin in the amygdala potentiates the anxiolytic effects of benzodiazepines.
Topics: Amygdala; Analysis of Variance; Animals; Anti-Anxiety Agents; beta-Galactosidase; Defective Viruses; Diazepam; DNA, Complementary; Enkephalins; Gene Transfer Techniques; Herpesvirus 4, Human; Humans; In Situ Hybridization; Maze Learning; Naloxone; Protein Precursors; Rats; Rats, Long-Evans; RNA, Messenger | 2000 |
Ultra-performance liquid chromatography coupled to time-of-flight mass spectrometry for robust, high-throughput quantitative analysis of an automated metabolic stability assay, with simultaneous determination of metabolic data.
Topics: Animals; Chromatography, High Pressure Liquid; Diazepam; Drug Evaluation, Preclinical; Drug Stability; Enkephalin, Leucine; Imipramine; Neurotransmitter Agents; Psychotropic Drugs; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Sensitivity and Specificity; Spectrometry, Mass, Electrospray Ionization | 2006 |
The role of delta opioid receptors in the anxiolytic actions of benzodiazepines.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Enkephalins; Male; Maze Learning; Naltrexone; Rats; Rats, Long-Evans; Receptors, GABA-A; Receptors, Opioid, delta | 2006 |