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emivirine and 6-(3,5-dimethylbenzyl)-1-(ethoxymethyl)-5-isopropyluracil

emivirine has been researched along with 6-(3,5-dimethylbenzyl)-1-(ethoxymethyl)-5-isopropyluracil in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (60.00)18.2507
2000's2 (40.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baba, M; De Clercq, E; Inouye, N; Miyasaka, T; Sekiya, K; Shigeta, S; Takashima, H; Tanaka, H; Ubasawa, M; Walker, RT1
Chrétien, JR; Grierson, DS; Kireev, DB; Monneret, C1
Baba, M; Hopkins, AL; Okamato, M; Ren, J; Stammers, DK; Stuart, DI; Tanaka, H1
Andries, K; Benjahad, A; Grierson, DS; Guillemont, J; Nguyen, CH1
El-Brollosy, NR; La Colla, P; Loddo, R; Pedersen, EB; Sanna, G; Sørensen, ER1

Other Studies

5 other study(ies) available for emivirine and 6-(3,5-dimethylbenzyl)-1-(ethoxymethyl)-5-isopropyluracil

ArticleYear
Synthesis and antiviral activity of 6-benzyl analogs of 1-[(2-hydroxyethoxy)methyl]-6-(phenylthio)thymine (HEPT) as potent and selective anti-HIV-1 agents.
    Journal of medicinal chemistry, 1995, Jul-21, Volume: 38, Issue:15

    Topics: Animals; Antiviral Agents; Benzyl Compounds; HIV Infections; HIV-1; Humans; Lymphocytes; Mice; Microbial Sensitivity Tests; Structure-Activity Relationship; Thymine

1995
A 3D QSAR study of a series of HEPT analogues: the influence of conformational mobility on HIV-1 reverse transcriptase inhibition.
    Journal of medicinal chemistry, 1997, Dec-19, Volume: 40, Issue:26

    Topics: Anti-HIV Agents; Drug Design; HIV Reverse Transcriptase; HIV-1; Models, Molecular; Molecular Conformation; Molecular Structure; Protein Binding; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Thymine

1997
Design of MKC-442 (emivirine) analogues with improved activity against drug-resistant HIV mutants.
    Journal of medicinal chemistry, 1999, Nov-04, Volume: 42, Issue:22

    Topics: Animals; Anti-HIV Agents; Cell Line; Crystallography, X-Ray; Drug Design; Drug Resistance, Microbial; HIV-1; Models, Molecular; Molecular Conformation; Mutation; Reverse Transcriptase Inhibitors; Uracil

1999
3-iodo-4-phenoxypyridinones (IOPY's), a new family of highly potent non-nucleoside inhibitors of HIV-1 reverse transcriptase.
    Bioorganic & medicinal chemistry letters, 2003, Dec-15, Volume: 13, Issue:24

    Topics: HIV-1; Models, Molecular; Molecular Conformation; Pyridones; Reverse Transcriptase Inhibitors; Structure-Activity Relationship

2003
Synthesis and antiviral evaluation of 6-(trifluoromethylbenzyl) and 6-(fluorobenzyl) analogues of HIV drugs emivirine and GCA-186.
    Archiv der Pharmazie, 2008, Volume: 341, Issue:1

    Topics: Anti-HIV Agents; Cell Line; Drug Resistance, Viral; HIV-1; Humans; Mutation; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Uracil

2008