Page last updated: 2024-09-05

emd 53998 and thapsigargin

emd 53998 has been researched along with thapsigargin in 3 studies

Compound Research Comparison

Studies
(emd 53998)
Trials
(emd 53998)
Recent Studies (post-2010)
(emd 53998)
Studies
(thapsigargin)
Trials
(thapsigargin)
Recent Studies (post-2010) (thapsigargin)
112095,2343918

Protein Interaction Comparison

ProteinTaxonomyemd 53998 (IC50)thapsigargin (IC50)
Sarcoplasmic/endoplasmic reticulum calcium ATPase 1Oryctolagus cuniculus (rabbit)0.002

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bletz, C; Rüegg, JC; Strauss, JD1
Hongo, K; Konishi, M; Kurihara, S; Kusakari, Y; Mochizuki, S1
Hongo, K; Kawai, M; Konishi, M; Kurihara, S; Kusakari, Y; Mochizuki, S1

Other Studies

3 other study(ies) available for emd 53998 and thapsigargin

ArticleYear
The calcium sensitizer EMD 53998 antagonizes phosphate-induced increases in energy cost of isometric tension in cardiac skinned fibres.
    European journal of pharmacology, 1994, Feb-03, Volume: 252, Issue:2

    Topics: Adenosine Diphosphate; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Calcium; Calcium-Transporting ATPases; Energy Metabolism; Heart; In Vitro Techniques; Isometric Contraction; Myocardium; NAD; Phosphates; Phosphodiesterase Inhibitors; Quinolines; Swine; Terpenes; Thapsigargin; Thiadiazines

1994
Estimation of myofibrillar responsiveness to Ca2+ in isolated rat ventricular myocytes.
    Pflugers Archiv : European journal of physiology, 1998, Volume: 436, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Calcium; Cell Size; Cells, Cultured; Electric Stimulation; Fluorescence; Fura-2; Heart Ventricles; Male; Myocardial Contraction; Myocardium; Myofibrils; Quinolines; Rats; Rats, Wistar; Tetany; Thapsigargin; Thiadiazines; Ventricular Function

1998
Use of tetanus to investigate myofibrillar responsiveness to Ca(2+) in isolated mouse ventricular myocytes.
    The Japanese journal of physiology, 2002, Volume: 52, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-Agonists; Animals; Calcium; Calcium-Transporting ATPases; Cardiotonic Agents; Cell Separation; Enzyme Inhibitors; Fluorescence; Isoproterenol; Mice; Muscle Contraction; Myocardium; Myofibrils; Phosphodiesterase Inhibitors; Quinolines; Thapsigargin; Thiadiazines; Ventricular Function

2002