em 523 has been researched along with tetrodotoxin in 2 studies
Studies (em 523) | Trials (em 523) | Recent Studies (post-2010) (em 523) | Studies (tetrodotoxin) | Trials (tetrodotoxin) | Recent Studies (post-2010) (tetrodotoxin) |
---|---|---|---|---|---|
26 | 1 | 0 | 12,992 | 11 | 1,477 |
Protein | Taxonomy | em 523 (IC50) | tetrodotoxin (IC50) |
---|---|---|---|
Sodium channel protein type 9 subunit alpha | Homo sapiens (human) | 0.0186 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (50.00) | 18.2507 |
2000's | 1 (50.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Inatomi, N; Itoh, Z; Marui, S; Omura, S; Satoh, H; Satoh, T | 1 |
Itoh, Z; Koga, H; Omura, S; Ozaki, K; Takanashi, H; Yogo, K | 1 |
2 other study(ies) available for em 523 and tetrodotoxin
Article | Year |
---|---|
EM-523, an erythromycin derivative, and motilin show similar contractile activity in isolated rabbit intestine.
Topics: Acetylcholine; Animals; Atropine; Dinoprost; Drug Interactions; Erythromycin; Female; Guinea Pigs; Intestine, Small; Male; Motilin; Muscle Contraction; Muscle, Smooth; Rabbits; Rats; Rats, Inbred Strains; Species Specificity; Tetrodotoxin | 1990 |
In vitro pharmacological characterization of mitemcinal (GM-611), the first acid-resistant non-peptide motilin receptor agonist, in smooth muscle of rabbit small intestine.
Topics: Acetylcholine; Animals; Atropine; Binding, Competitive; Calcium Chloride; Diltiazem; Dose-Response Relationship, Drug; Erythromycin; Hexamethonium; Hydrogen-Ion Concentration; In Vitro Techniques; Indoles; Intestine, Small; Male; Molecular Structure; Muscle Contraction; Muscle, Smooth; Naloxone; Rabbits; Receptors, Gastrointestinal Hormone; Receptors, Neuropeptide; Tetrodotoxin; Tropisetron; Verapamil | 2007 |