Page last updated: 2024-09-05

em 523 and tetrodotoxin

em 523 has been researched along with tetrodotoxin in 2 studies

Compound Research Comparison

Studies
(em 523)
Trials
(em 523)
Recent Studies (post-2010)
(em 523)
Studies
(tetrodotoxin)
Trials
(tetrodotoxin)
Recent Studies (post-2010) (tetrodotoxin)
261012,992111,477

Protein Interaction Comparison

ProteinTaxonomyem 523 (IC50)tetrodotoxin (IC50)
Sodium channel protein type 9 subunit alphaHomo sapiens (human)0.0186

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Inatomi, N; Itoh, Z; Marui, S; Omura, S; Satoh, H; Satoh, T1
Itoh, Z; Koga, H; Omura, S; Ozaki, K; Takanashi, H; Yogo, K1

Other Studies

2 other study(ies) available for em 523 and tetrodotoxin

ArticleYear
EM-523, an erythromycin derivative, and motilin show similar contractile activity in isolated rabbit intestine.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:3

    Topics: Acetylcholine; Animals; Atropine; Dinoprost; Drug Interactions; Erythromycin; Female; Guinea Pigs; Intestine, Small; Male; Motilin; Muscle Contraction; Muscle, Smooth; Rabbits; Rats; Rats, Inbred Strains; Species Specificity; Tetrodotoxin

1990
In vitro pharmacological characterization of mitemcinal (GM-611), the first acid-resistant non-peptide motilin receptor agonist, in smooth muscle of rabbit small intestine.
    Pharmacology, 2007, Volume: 79, Issue:3

    Topics: Acetylcholine; Animals; Atropine; Binding, Competitive; Calcium Chloride; Diltiazem; Dose-Response Relationship, Drug; Erythromycin; Hexamethonium; Hydrogen-Ion Concentration; In Vitro Techniques; Indoles; Intestine, Small; Male; Molecular Structure; Muscle Contraction; Muscle, Smooth; Naloxone; Rabbits; Receptors, Gastrointestinal Hormone; Receptors, Neuropeptide; Tetrodotoxin; Tropisetron; Verapamil

2007