Page last updated: 2024-09-03

elacridar and pepstatin

elacridar has been researched along with pepstatin in 2 studies

Compound Research Comparison

Studies
(elacridar)
Trials
(elacridar)
Recent Studies (post-2010)
(elacridar)
Studies
(pepstatin)
Trials
(pepstatin)
Recent Studies (post-2010) (pepstatin)
28481196960125

Protein Interaction Comparison

ProteinTaxonomyelacridar (IC50)pepstatin (IC50)
Pepsin ASus scrofa (pig)0.011
ReninHomo sapiens (human)1.9333
Cathepsin DHomo sapiens (human)0.3597
Procathepsin LHomo sapiens (human)0.8
Cathepsin BHomo sapiens (human)4.26
Candidapepsin-2Candida albicans0.09
Pepsin A-5Homo sapiens (human)0.059
Cathepsin EHomo sapiens (human)0.5558
Plasmepsin-1Plasmodium falciparum (malaria parasite P. falciparum)0.0009
Plasmepsin-2Plasmodium falciparum (malaria parasite P. falciparum)0.0005
Cathepsin D Bos taurus (cattle)0.0235
Disintegrin and metalloproteinase domain-containing protein 9Homo sapiens (human)0.0563
Plasmepsin 4 Plasmodium falciparum (malaria parasite P. falciparum)0.0003
Cysteine proteaseLeishmania donovani0.16
Protease Human immunodeficiency virus 10.947

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (50.00)24.3611
2020's1 (50.00)2.80

Authors

AuthorsStudies
Adler, P; Falson, P; Gimenez, AS; Gros, G; Hasserodt, J; Martinez, L; Maurin, P; Wolkowicz, R1
Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M1

Other Studies

2 other study(ies) available for elacridar and pepstatin

ArticleYear
Modular construction of quaternary hemiaminal-based inhibitor candidates and their in cellulo assessment with HIV-1 protease.
    Bioorganic & medicinal chemistry, 2013, Sep-01, Volume: 21, Issue:17

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Cell Line; Cell Survival; HEK293 Cells; HIV Protease; HIV Protease Inhibitors; HIV-1; Humans; Mice; Neoplasm Proteins; NIH 3T3 Cells; Urea

2013
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
    Disease models & mechanisms, 2023, 03-01, Volume: 16, Issue:3

    Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries

2023