elacridar has been researched along with incb-018424 in 1 studies
Studies (elacridar) | Trials (elacridar) | Recent Studies (post-2010) (elacridar) | Studies (incb-018424) | Trials (incb-018424) | Recent Studies (post-2010) (incb-018424) |
---|---|---|---|---|---|
284 | 8 | 119 | 1,487 | 185 | 1,451 |
Protein | Taxonomy | elacridar (IC50) | incb-018424 (IC50) |
---|---|---|---|
Cyclin-G-associated kinase | Homo sapiens (human) | 0.12 | |
Tyrosine-protein kinase JAK2 | Homo sapiens (human) | 0.0573 | |
Cytochrome P450 1A2 | Homo sapiens (human) | 0.0001 | |
Tyrosine-protein kinase JAK1 | Homo sapiens (human) | 0.0327 | |
Non-receptor tyrosine-protein kinase TYK2 | Homo sapiens (human) | 0.0962 | |
Tyrosine-protein kinase JAK3 | Homo sapiens (human) | 0.3547 | |
AP2-associated protein kinase 1 | Homo sapiens (human) | 0.1 | |
Histone deacetylase 6 | Homo sapiens (human) | 0.015 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 1 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ | 1 |
1 other study(ies) available for elacridar and incb-018424
Article | Year |
---|---|
Identification of potent Yes1 kinase inhibitors using a library screening approach.
Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship | 2013 |