egtazic acid has been researched along with bisindolylmaleimide i in 45 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 10 (22.22) | 18.2507 |
2000's | 33 (73.33) | 29.6817 |
2010's | 2 (4.44) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Bekker, OB; Danilenko, VN; Elizarov, SM; Kubbutat, MH; Lakatosh, SA; Luzikov, YN; Preobrazhenskaya, MN; Printsevskaya, SS; Reznikova, MI; Schächtele, C; Shtil, AA; Simonov, AY; Totzke, F | 1 |
Brugge, JS; Cunningham, M; Ginsberg, MH; Haimovich, B; Lipfert, L; Parsons, JT; Shattil, SJ | 1 |
Haimovich, B; Ji, P; Kaneshiki, N | 1 |
Artemenko, IP; Hokin, LE; Los, GV | 1 |
Petryniak, MA; Slack, BE; Wurtman, RJ | 1 |
Breu, J; Muchnicki, L; Slack, BE; Wurtman, RJ | 1 |
Del Valle, J; Nagahara, A; Todisco, A; Wang, L | 1 |
Blank, U; David, B; Guérin-Marchand, C; Iannascoli, B; Marchand, F; Pelletier, C; Weyer, A | 1 |
Bae, YS; Baek, SH; Ju, SA; Kim, BS; Kim, JY; Kwak, JY; Ryu, SH; Seo, JK; Suh, PG | 1 |
Goracci, G; Gresele, P; Macchioni, L; Nardicchi, V; Nenci, GG; Nucciarelli, F; Porcellati, S | 1 |
Akiba, S; Hayama, M; Kume, K; Mizunaga, S; Sato, T | 1 |
Han, B; Logsdon, CD | 1 |
Abbott, KL; Berts, A; Lee, D; Minneman, KP; Murphy, TJ; Zhong, H | 1 |
Boland, R; Buitrago, C; de Boland, AR; Morelli, S | 1 |
Chien, CS; Chiu, CT; Hsiao, LD; Lin, CC; Shyr, MH; Wang, CC; Yang, CM | 1 |
Chang, LC; Wang, JP | 1 |
Drew, AE; Werling, LL | 1 |
Inanami, O; Kuwabara, M; Tsuji, M | 1 |
Crow, T; Neary, JT; Siddiqi, V; Xue-Bian, JJ | 1 |
Nakajima, Y; Nakanishi, S; Shinohara, Y | 1 |
Låg, M; Refsnes, M; Schwarze, PE; Thoresen, GH; Thrane, EV | 1 |
Juang, YT; Kiang, JG; Kiang, SC; Tsokos, GC | 1 |
Hörsch, D; Trümper, A; Trümper, K | 1 |
Bazan, NG; Bernatchez, PN; Gélinas, DS; Rollin, S; Sirois, MG | 1 |
Barak, V; Moroz, C; Traub, L; Zahalka, MA | 1 |
Bhugra, P; Dhalla, NS; Rathi, S; Xu, YJ | 1 |
Calixto, JB; El Sayah, M | 1 |
Abbey-Hosch, SE; Cody, AN; Potter, LR | 1 |
Choi, JW; Donowitz, M; Jeon, ES; Kang, YJ; Kawano, K; Kim, HS; Kim, JH; Lee-Kwon, W; Suh, PG | 1 |
Ramamoorthy, S; Stepan, V; Todisco, A | 1 |
Camden, JM; Camden, RE; Erb, L; González, FA; Schrader, AM; Seye, CI; Weisman, GA | 1 |
Cameron, P; Kanke, T; Macfarlane, SR; McKenzie, RC; Plevin, R; Sloss, CM | 1 |
Fu, WM; Tang, CH; Yang, RS | 1 |
Chang, Q; Soper, BD; Tepperman, BL | 1 |
Kobayashi, D; Nakahata, N; Ohkubo, S; Yoshida, H | 1 |
Horie, T; Ito, K; Sekine, S | 1 |
Aguilar, R; Bellido, C; Garrido-Gracia, JC; Sánchez-Criado, JE | 1 |
Chang, HC; Chen, IS; Cheng, HH; Chi, CC; Chu, ST; Ho, CM; Hsu, SS; Huang, CJ; Huang, JK; Jan, CR; Liu, SI; Lu, YC; Su, HH; Wang, JL | 1 |
Burgos, RA; Carretta, D; Hancke, JL; Hidalgo, MA; Sandoval, A; Sanhueza, A; Triviños, F | 1 |
Goode, GD; Johnson, AL; Mtshali, C; Myles, EL; Washington, B | 1 |
Bastián, Y; Mújica, A; Uribe, S; Zepeda-Bastida, A | 1 |
Cai, L; Hertz, L; Li, B; Nu, W; Peng, L; Zhang, H; Zhang, S | 1 |
Alrefai, WA; Annaba, F; Dwivedi, A; Gill, RK; Saksena, S; Sarwar, Z | 1 |
Baxter, RC; Bolitho, C; Marsh, DJ; Mertens-Walker, I | 1 |
Chang, HT; Chou, CT; Jan, CR; Kuo, DH; Liang, WZ; Shieh, P | 1 |
45 other study(ies) available for egtazic acid and bisindolylmaleimide i
Article | Year |
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Search for inhibitors of bacterial and human protein kinases among derivatives of diazepines[1,4] annelated with maleimide and indole cycles.
Topics: Chemistry, Pharmaceutical; Humans; Indoles; Inhibitory Concentration 50; Maleimides; Models, Chemical; Molecular Conformation; Phosphorylation; Protein Kinase Inhibitors; Protein Kinases; Recombinant Proteins; Serine; Streptomyces lividans; Thiourea; Threonine | 2008 |
Tyrosine phosphorylation of pp125FAK in platelets requires coordinated signaling through integrin and agonist receptors.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Actins; Alprostadil; Apyrase; Blood Platelets; Calcium; Cell Adhesion Molecules; Cytoplasm; Egtazic Acid; Epinephrine; Fibrinogen; Focal Adhesion Kinase 1; Focal Adhesion Protein-Tyrosine Kinases; Humans; Immunoglobulin Fab Fragments; In Vitro Techniques; Indoles; Indomethacin; Maleimides; Models, Biological; Phosphorylation; Phosphotyrosine; Platelet Membrane Glycoproteins; Prostaglandin Endoperoxides, Synthetic; Protein Kinase C; Protein-Tyrosine Kinases; Signal Transduction; Thromboxane A2; Tyrosine; Vasodilator Agents | 1994 |
Protein kinase C regulates tyrosine phosphorylation of pp125FAK in platelets adherent to fibrinogen.
Topics: Adenosine Diphosphate; Apyrase; Blood Platelets; Calcium; Cell Adhesion Molecules; Cell Size; Egtazic Acid; Enzyme Inhibitors; Fibrinogen; Focal Adhesion Kinase 1; Focal Adhesion Protein-Tyrosine Kinases; Humans; Indoles; Maleimides; Phosphoproteins; Phosphorylation; Platelet Adhesiveness; Platelet Glycoprotein GPIIb-IIIa Complex; Protein Kinase C; Protein Processing, Post-Translational; Protein-Tyrosine Kinases; Signal Transduction; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin; Tyrosine | 1996 |
Phosphoinositide signalling in human neuroblastoma cells: biphasic effect of Li+ on the level of the inositolphosphate second messengers.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetylcholine; Atropine; Calcium; Egtazic Acid; Enzyme Inhibitors; Humans; Indoles; Inositol 1,4,5-Trisphosphate; Inositol Phosphates; Lithium; Maleimides; Neuroblastoma; Nickel; Phosphatidylinositols; Protein Kinase Inhibitors; Signal Transduction; Staurosporine; Tumor Cells, Cultured | 1996 |
Elevated intracellular calcium concentration increases secretory processing of the amyloid precursor protein by a tyrosine phosphorylation-dependent mechanism.
Topics: Amyloid beta-Protein Precursor; Blotting, Western; Calcium; Carbachol; Cells, Cultured; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Genistein; Humans; Indoles; Ionomycin; Isoflavones; Kidney; Maleimides; Phosphorylation; Phosphotyrosine; Protein Kinase C; Receptors, Muscarinic; Signal Transduction; Tyrosine | 1996 |
Rapid stimulation of amyloid precursor protein release by epidermal growth factor: role of protein kinase C.
Topics: Amyloid beta-Protein Precursor; Amyloid Precursor Protein Secretases; Androstadienes; Aspartic Acid Endopeptidases; Egtazic Acid; Electrophoresis, Polyacrylamide Gel; Endopeptidases; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; ErbB Receptors; Humans; Indoles; Inositol; Inositol Phosphates; Maleimides; Nitriles; Phosphatidylinositols; Phosphotyrosine; Protein Kinase C; Quinazolines; Tumor Cells, Cultured; Tyrphostins; Wortmannin | 1997 |
Regulation of c-Jun NH2-terminal kinases in isolated canine gastric parietal cells.
Topics: Animals; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Cells, Cultured; Chelating Agents; Dogs; Egtazic Acid; Enzyme Induction; Enzyme Inhibitors; Epidermal Growth Factor; Gastric Fundus; Gene Expression Regulation, Enzymologic; Genes, jun; Histamine; Indoles; JNK Mitogen-Activated Protein Kinases; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 9; Mitogen-Activated Protein Kinases; Parietal Cells, Gastric; Protein Kinase C; Protein Kinases; Proto-Oncogene Proteins c-jun; Recombinant Proteins; RNA, Messenger; Thapsigargin; Transcription, Genetic; Transfection | 1998 |
Specific signaling pathways in the regulation of TNF-alpha mRNA synthesis and TNF-alpha secretion in RBL-2H3 mast cells stimulated through the high affinity IgE receptor.
Topics: Androstadienes; Animals; beta-N-Acetylhexosaminidases; Egtazic Acid; Enzyme Inhibitors; Gene Expression; Indoles; Leukemia, Basophilic, Acute; Maleimides; Mast Cells; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Rats; Receptors, IgE; Reverse Transcriptase Polymerase Chain Reaction; Ribonucleases; RNA, Messenger; Signal Transduction; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha; Wortmannin | 1998 |
Trp-Lys-Tyr-Met-Val-D-Met stimulates superoxide generation and killing of Staphylococcus aureus via phospholipase D activation in human monocytes.
Topics: Calcium; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Humans; Indoles; Maleimides; Monocytes; Oligopeptides; Phospholipase D; Receptors, Cell Surface; Staphylococcus aureus; Superoxides; Type C Phospholipases | 1999 |
Evidence that cytosolic phospholipase A2 is down-regulated by protein kinase C in intact human platelets stimulated with fluoroaluminate.
Topics: Aluminum; Arachidonic Acid; Arachidonic Acids; Blood Platelets; Calcium; Cytosol; Down-Regulation; Egtazic Acid; Enzyme Inhibitors; Fluorine; Humans; Indoles; Maleimides; Phospholipases A; Phospholipases A2; Protein Kinase C | 1999 |
Involvement of group VI Ca2+-independent phospholipase A2 in protein kinase C-dependent arachidonic acid liberation in zymosan-stimulated macrophage-like P388D1 cells.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Calcium; Diglycerides; Egtazic Acid; Group VI Phospholipases A2; Indoles; Leukemia P388; Maleimides; Mice; Naphthalenes; Oligonucleotides, Antisense; Organophosphonates; Phospholipases A; Phospholipases A2; Protein Kinase C; Pyrones; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Zymosan | 1999 |
CCK stimulates mob-1 expression and NF-kappaB activation via protein kinase C and intracellular Ca(2+).
Topics: Animals; Biological Transport; Calcium; Carcinogens; Cell Nucleus; Chelating Agents; Chemokine CXCL10; Chemokines, CXC; Cholecystokinin; Cytokines; DNA-Binding Proteins; Egtazic Acid; Enzyme Inhibitors; Gene Expression; In Vitro Techniques; Indoles; Ionomycin; Ionophores; Male; Maleimides; NF-kappa B; Pancreas; Phosphorylation; Protein Kinase C; Rats; Rats, Wistar; RNA, Messenger; Tetradecanoylphorbol Acetate | 2000 |
Transcriptional responses to growth factor and G protein-coupled receptors in PC12 cells: comparison of alpha(1)-adrenergic receptor subtypes.
Topics: Animals; Cell Differentiation; Chelating Agents; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; DNA-Binding Proteins; Dose-Response Relationship, Drug; Egtazic Acid; Enzyme Inhibitors; Epidermal Growth Factor; Flavonoids; Gene Expression; Genes, Reporter; GTP-Binding Proteins; Humans; Imidazoles; Indoles; Luciferases; Maleimides; Mitogen-Activated Protein Kinases; Nerve Growth Factors; Neurons; NF-kappa B; NFATC Transcription Factors; Norepinephrine; Nuclear Proteins; p38 Mitogen-Activated Protein Kinases; PC12 Cells; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Pyridines; Rats; Receptors, Adrenergic, alpha-1; Sympathomimetics; Transcription Factors; Transcriptional Activation; Transfection | 2000 |
The stimulation of MAP kinase by 1,25(OH)(2)-vitamin D(3) in skeletal muscle cells is mediated by protein kinase C and calcium.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calcitriol; Calcium; Calmodulin; Chick Embryo; Egtazic Acid; Enzyme Activation; Fluphenazine; Indoles; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Muscle, Skeletal; Naphthalenes; Neomycin; Phosphorylation; Protein Kinase C; Tetradecanoylphorbol Acetate; Thapsigargin; Type C Phospholipases; Verapamil | 2001 |
Mechanisms of thrombin-induced MAPK activation associated with cell proliferation in human cultured tracheal smooth muscle cells.
Topics: Androstadienes; Benzoquinones; Blotting, Western; Cell Division; Cells, Cultured; Chelating Agents; Chromones; Dose-Response Relationship, Drug; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Estrenes; Flavonoids; Genistein; Humans; Indoles; Lactams, Macrocyclic; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Morpholines; Muscle, Smooth; Pertussis Toxin; Phosphatidylinositol 3-Kinases; Phosphorylation; Plasmids; Protein Isoforms; Protein Kinase C; Proto-Oncogene Proteins c-raf; Pyrrolidinones; Quinones; ras Proteins; Rifabutin; Thrombin; Time Factors; Trachea; Transfection; Virulence Factors, Bordetella; Wortmannin | 2001 |
Signal transduction pathways for activation of extracellular signal-regulated kinase by arachidonic acid in rat neutrophils.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Androstadienes; Animals; Arachidonic Acid; Arachidonic Acids; Butadienes; Calcium; Carbazoles; Chelating Agents; Chromones; Cyclooxygenase Inhibitors; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Estrenes; Flavonoids; GTP-Binding Protein alpha Subunits, Gi-Go; Heterotrimeric GTP-Binding Proteins; Indoles; Lipoxygenase Inhibitors; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Morpholines; Neutrophils; Nitriles; Pertussis Toxin; Phosphatidylinositol Diacylglycerol-Lyase; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Processing, Post-Translational; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Type C Phospholipases; Virulence Factors, Bordetella; Wortmannin | 2001 |
Protein kinase C regulation of dopamine transporter initiated by nicotinic receptor activation in slices of rat prefrontal cortex.
Topics: Alkaloids; Amphetamine; Animals; Benzophenanthridines; Calcium; Calcium Channel Blockers; Carrier Proteins; Dopamine; Dopamine Plasma Membrane Transport Proteins; Egtazic Acid; Enzyme Inhibitors; Indoles; Male; Maleimides; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Nicotine; omega-Conotoxin GVIA; Phenanthridines; Potassium; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Second Messenger Systems; Sodium Channels; Staurosporine; Tetrodotoxin; Tritium; Veratridine | 2001 |
Induction of neurite outgrowth in PC12 cells by alpha -phenyl-N-tert-butylnitron through activation of protein kinase C and the Ras-extracellular signal-regulated kinase pathway.
Topics: Acetylcysteine; Androstadienes; Animals; Cyclic N-Oxides; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Free Radical Scavengers; Indoles; Isoquinolines; Kinetics; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Neurites; Neuroprotective Agents; Nitrogen Oxides; p38 Mitogen-Activated Protein Kinases; PC12 Cells; Protein Kinase C; ras Proteins; Rats; Recombinant Proteins; Signal Transduction; Sulfonamides; Transfection; Wortmannin | 2001 |
Serotonin activation of the ERK pathway in Hermissenda: contribution of calcium-dependent protein kinase C.
Topics: Animals; Calcium; Carbazoles; Chelating Agents; Conditioning, Classical; Egtazic Acid; Enzyme Inhibitors; Indoles; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Mollusca; Phosphorylation; Serotonin; Tetradecanoylphorbol Acetate | 2001 |
Glutamate induces focal adhesion kinase tyrosine phosphorylation and actin rearrangement in heterologous mGluR1-expressing CHO cells via calcium/calmodulin signaling.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Actins; Animals; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; CHO Cells; Cricetinae; Cytoskeleton; Edetic Acid; Egtazic Acid; Enzyme Inhibitors; Estrenes; Focal Adhesion Protein-Tyrosine Kinases; Focal Adhesions; Glutamic Acid; Indoles; Kinetics; Maleimides; Phosphorylation; Protein-Tyrosine Kinases; Pyrrolidinones; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Recombinant Proteins; Transfection; Type C Phospholipases | 2001 |
Mechanisms in fluoride-induced interleukin-8 synthesis in human lung epithelial cells.
Topics: Androstadienes; Benzylamines; Cell Line; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Egtazic Acid; Epithelial Cells; Flavonoids; Genistein; Humans; Indoles; Interleukin-8; Isoquinolines; Lung; Maleimides; Okadaic Acid; Pertussis Toxin; Protein Kinase C; Signal Transduction; Sodium Fluoride; Sulfonamides; Tetradecanoylphorbol Acetate; Vanadates; Virulence Factors, Bordetella; Wortmannin | 2001 |
N(omega)-nitro-L-arginine inhibits inducible HSP-70 via Ca(2+), PKC, and PKA in human intestinal epithelial T84 cells.
Topics: Calcium; Cell Nucleus; Chelating Agents; Colonic Neoplasms; Cyclic AMP-Dependent Protein Kinases; Cycloheximide; Cytosol; Dactinomycin; DNA-Binding Proteins; Egtazic Acid; Enzyme Inhibitors; Guanidines; Heat Shock Transcription Factors; Hot Temperature; HSP70 Heat-Shock Proteins; Humans; Indoles; Intestinal Mucosa; Intestines; Isoquinolines; Maleimides; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Protein Kinase C; Protein Kinases; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sulfonamides; Transcription Factors; Tumor Cells, Cultured | 2002 |
Mechanisms of mitogenic and anti-apoptotic signaling by glucose-dependent insulinotropic polypeptide in beta(INS-1)-cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alloxan; Androstadienes; Apoptosis; Arginase; B-Lymphocytes; Benzylamines; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Chelating Agents; Cyclic AMP-Dependent Protein Kinases; Deoxyglucose; Egtazic Acid; Enzyme Inhibitors; Flavonoids; Gastric Inhibitory Polypeptide; Genistein; Glucokinase; Glucose; Humans; Indoles; Isoquinolines; Maleimides; MAP Kinase Kinase 1; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase Kinases; Mitosis; Phosphoinositide-3 Kinase Inhibitors; Plasmids; Protein Kinase C; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Signal Transduction; Sulfonamides; Wortmannin | 2002 |
Immediate and delayed VEGF-mediated NO synthesis in endothelial cells: role of PI3K, PKC and PLC pathways.
Topics: 1-Methyl-3-isobutylxanthine; Androstadienes; Animals; Calcimycin; Calcium; Cattle; Cells, Cultured; Chelating Agents; Chromones; Cyclic GMP; Diterpenes; Dose-Response Relationship, Drug; Egtazic Acid; Endothelial Growth Factors; Endothelium, Vascular; Enzyme Inhibitors; Ginkgolides; Indoles; Intercellular Signaling Peptides and Proteins; Ionophores; Lactones; Lymphokines; Maleimides; Morpholines; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Nitroprusside; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Platelet Activating Factor; Platelet Membrane Glycoproteins; Protein Kinase C; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Serine; Signal Transduction; Time Factors; Type C Phospholipases; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors; Wortmannin | 2002 |
PLIF induces IL-10 production in monocytes: a calmodulin-p38 mitogen-activated protein kinase-dependent pathway.
Topics: Binding Sites; Calcium; Calmodulin; Coculture Techniques; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Ferritins; Humans; Indoles; Interleukin-10; Isoquinolines; Leukocytes, Mononuclear; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Monocytes; Oxidoreductases; p38 Mitogen-Activated Protein Kinases; Peptide Fragments; Pregnancy Proteins; Recombinant Proteins; Sulfonamides; T-Lymphocytes | 2003 |
Modification of intracellular free calcium in cultured A10 vascular smooth muscle cells by exogenous phosphatidic acid.
Topics: Animals; Boron Compounds; Calcium; Carbamates; Cells, Cultured; Diltiazem; Drug Interactions; Egtazic Acid; Indoles; Macrocyclic Compounds; Maleimides; Muscle, Smooth, Vascular; Oxazoles; Pertussis Toxin; Phenylcarbamates; Phosphatidic Acids; Rats; Tetradecanoylphorbol Acetate; Thapsigargin; Verapamil | 2003 |
New evidence on the mechanisms underlying bradykinin-mediated contraction of the pig iris sphincter in vitro.
Topics: Animals; Benzamides; Bradykinin; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Calcium; Calcium Channels; Capsaicin; Carbazoles; Conotoxins; Dipeptides; Dose-Response Relationship, Drug; Egtazic Acid; In Vitro Techniques; Indoles; Iris; Maleimides; Muscle Contraction; Nicardipine; omega-Agatoxin IVA; Peptide Fragments; Piperidines; Protein Kinase Inhibitors; Protein Kinases; Pyrroles; Receptors, Calcitonin Gene-Related Peptide; Receptors, Drug; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Swine; Tachykinins | 2003 |
Sphingosine-1-phosphate inhibits C-type natriuretic peptide activation of guanylyl cyclase B (GC-B/NPR-B).
Topics: Animals; Cell Division; Cyclic GMP; Dose-Response Relationship, Drug; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Fibroblasts; Guanylate Cyclase; Indoles; Inhibitory Concentration 50; Ionomycin; Maleimides; Mice; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Natriuretic Peptide, C-Type; NIH 3T3 Cells; Organ Specificity; Rats; Receptors, Cell Surface; Signal Transduction; Sphingosine | 2004 |
Lysophosphatidic acid induces exocytic trafficking of Na(+)/H(+) exchanger 3 by E3KARP-dependent activation of phospholipase C.
Topics: Animals; Calcium; Cell Membrane; Cells, Cultured; Chelating Agents; CHO Cells; Cricetinae; Cytoskeletal Proteins; Egtazic Acid; Enzyme Inhibitors; Exocytosis; Indoles; Kidney Tubules, Proximal; Lysophospholipids; Maleimides; Opossums; Protein Kinase C; Protein Transport; Signal Transduction; Sodium-Hydrogen Exchanger 3; Sodium-Hydrogen Exchangers; Type C Phospholipases | 2004 |
Intracellular mechanisms mediating the anti-apoptotic action of gastrin.
Topics: Animals; Apoptosis; bcl-Associated Death Protein; Blotting, Western; Calcium; Carrier Proteins; Cell Line; Chelating Agents; DNA-Binding Proteins; Egtazic Acid; Enzyme Inhibitors; Forkhead Transcription Factors; Gastrins; Genes, Reporter; Genetic Vectors; Immunoprecipitation; Indoles; Luciferases; Maleimides; Nerve Tissue Proteins; Phosphorylation; Plasmids; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Rats; Recombinant Proteins; Transcription Factors; Transcription, Genetic; Transfection | 2004 |
P2Y2 nucleotide receptors enhance alpha-secretase-dependent amyloid precursor protein processing.
Topics: ADAM Proteins; ADAM17 Protein; Amino Acid Chloromethyl Ketones; Amyloid beta-Protein Precursor; Amyloid Precursor Protein Secretases; Aspartic Acid Endopeptidases; Blotting, Western; Butadienes; Calcium; Cell Line, Tumor; Central Nervous System; Chelating Agents; Dose-Response Relationship, Drug; Down-Regulation; Egtazic Acid; Endopeptidases; Furin; Humans; Indoles; Maleimides; MAP Kinase Signaling System; Metalloendopeptidases; Nitriles; Phorbol Esters; Protein Kinase C; Protein Structure, Tertiary; Receptors, Purinergic P2; Receptors, Purinergic P2Y2; RNA, Small Interfering; Tetradecanoylphorbol Acetate; Time Factors; Transfection; Uridine Triphosphate | 2005 |
The role of intracellular Ca2+ in the regulation of proteinase-activated receptor-2 mediated nuclear factor kappa B signalling in keratinocytes.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcium; Cell Line; Chelating Agents; Egtazic Acid; Enzyme Inhibitors; Estrenes; Humans; I-kappa B Kinase; Indoles; Keratinocytes; Maleimides; Mitogen-Activated Protein Kinases; NF-kappa B; Oligonucleotides; Phosphodiesterase Inhibitors; Protein Binding; Protein Kinase C; Protein Serine-Threonine Kinases; Pyrrolidinones; Receptor, PAR-2; Signal Transduction; Tacrolimus; Tetradecanoylphorbol Acetate; Trypsin; Type C Phospholipases | 2005 |
Prostaglandin E2 stimulates fibronectin expression through EP1 receptor, phospholipase C, protein kinase Calpha, and c-Src pathway in primary cultured rat osteoblasts.
Topics: Animals; Blotting, Western; Bone and Bones; Bone Density; Calcium; Cell Membrane; Cells, Cultured; Chelating Agents; Cyclic AMP-Dependent Protein Kinases; Dinoprostone; Egtazic Acid; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Estrenes; Fibronectins; Genes, Dominant; Genes, Reporter; Immunoblotting; Immunohistochemistry; Immunoprecipitation; Indoles; Integrin alpha5; Integrin beta1; Integrins; Maleimides; Microscopy, Fluorescence; Mutation; Oligonucleotides; Oligonucleotides, Antisense; Osteoblasts; Promoter Regions, Genetic; Protein Isoforms; Protein Kinase C; Pyrimidines; Pyrrolidinones; Rats; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP1 Subtype; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; src-Family Kinases; Transfection; Type C Phospholipases; Up-Regulation | 2005 |
Effect of protein kinase C activation on intracellular Ca2+ signaling and integrity of intestinal epithelial cells.
Topics: Acetophenones; Animals; Benzopyrans; Calcium; Calcium Channel Blockers; Calcium Signaling; Carbazoles; Cell Line; Cell Survival; Chelating Agents; Dose-Response Relationship, Drug; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Epithelial Cells; Indoles; Intestinal Mucosa; Intracellular Space; Maleimides; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-delta; Protein Kinase C-epsilon; Tetradecanoylphorbol Acetate; Verapamil | 2005 |
ATP stimulates interleukin-6 production via P2Y receptors in human HaCaT keratinocytes.
Topics: Adenosine Triphosphate; Calcium; Cell Line; Dactinomycin; Dose-Response Relationship, Drug; Egtazic Acid; Enzyme-Linked Immunosorbent Assay; Gene Expression; Humans; Indoles; Interleukin-6; Keratinocytes; Maleimides; Purinergic P2 Receptor Agonists; Receptors, Purinergic P2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Stress, Mechanical; Suramin; Time Factors; Uridine Triphosphate | 2006 |
Oxidative stress and Mrp2 internalization.
Topics: Animals; ATP-Binding Cassette Transporters; Bile Canaliculi; Calcium; Cell Nucleus; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Egtazic Acid; Enzyme Activation; Ethacrynic Acid; Glutathione; Hepatocytes; In Vitro Techniques; Indoles; Isoenzymes; Liver; Male; Maleimides; Nitric Oxide; Oxidative Stress; Protein Kinase C; Protein Kinase Inhibitors; Protein Transport; Rats; Rats, Sprague-Dawley | 2006 |
Protein kinase C cross-talk with gonadotrope progesterone receptor is involved in GnRH-induced LH secretion.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Bodily Secretions; Cells, Cultured; Chelating Agents; Colforsin; Egtazic Acid; Enzyme Inhibitors; Female; Gonadotropin-Releasing Hormone; Imines; Indoles; Ionomycin; Luteinizing Hormone; Maleimides; Mifepristone; Nifedipine; Pituitary Gland, Anterior; Protein Kinase C; Rats; Rats, Wistar; Receptors, Progesterone; Signal Transduction; Tetradecanoylphorbol Acetate | 2006 |
Phospholipase A2-independent Ca2+ entry and subsequent apoptosis induced by melittin in human MG63 osteosarcoma cells.
Topics: Apoptosis; Calcium; Calcium Channels, L-Type; Cell Line, Tumor; Cell Survival; Egtazic Acid; Enzyme Inhibitors; Fluorescent Dyes; Fura-2; Humans; Indoles; Maleimides; Melitten; Osteoblasts; Osteosarcoma; Phospholipases A; Phospholipases A2; Tetradecanoylphorbol Acetate | 2007 |
Propionate induces pH(i) changes through calcium flux, ERK1/2, p38, and PKC in bovine neutrophils.
Topics: Animals; Butadienes; Calcium; Cattle; Chelating Agents; Chromones; Egtazic Acid; Extracellular Signal-Regulated MAP Kinases; Female; Hydrogen-Ion Concentration; Imidazoles; Indoles; Ionomycin; Maleimides; Morpholines; Neutrophils; Nitriles; p38 Mitogen-Activated Protein Kinases; Propionates; Protein Kinase C; Protein Kinase Inhibitors; Pyridines; Sodium-Hydrogen Exchangers; Spectrometry, Fluorescence | 2007 |
Protein Kinase C- alpha/betaII, delta, and zeta/lambda involvement in ethanol-induced MAPK expression in vascular smooth muscle cells.
Topics: Animals; Cells, Cultured; Egtazic Acid; Ethanol; Indoles; Isoenzymes; Maleimides; Mitogen-Activated Protein Kinase Kinases; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-alpha; Protein Kinase C-delta; Rats; Time Factors; Up-Regulation | 2007 |
In spermatozoa, Stat1 is activated during capacitation and the acrosomal reaction.
Topics: Acrosome Reaction; Animals; Biological Transport; Blotting, Western; Calcium; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Cytoplasm; Egtazic Acid; Electrophoresis, Polyacrylamide Gel; Genistein; Guinea Pigs; Indoles; Isoflavones; Isoquinolines; Male; Maleimides; Phosphorylation; Protein Kinase C; Protein-Tyrosine Kinases; Sperm Capacitation; Sperm Tail; Spermatozoa; STAT1 Transcription Factor; STAT4 Transcription Factor; Sulfonamides; Transcriptional Activation | 2007 |
Fluoxetine-mediated 5-HT2B receptor stimulation in astrocytes causes EGF receptor transactivation and ERK phosphorylation.
Topics: Aminopyridines; Animals; Antidepressive Agents, Second-Generation; Astrocytes; Butadienes; Calcium; Cells, Cultured; Chelating Agents; Dipeptides; Dose-Response Relationship, Drug; Egtazic Acid; ErbB Receptors; Extracellular Signal-Regulated MAP Kinases; Fluorobenzenes; Fluoxetine; Gene Expression; Indoles; Maleimides; Mice; Nitriles; Phosphorylation; Piperidines; Protein Kinase C; Proto-Oncogene Proteins c-fos; Quinazolines; Receptor, Serotonin, 5-HT2B; RNA, Messenger; Signal Transduction; Substrate Specificity; Transcriptional Activation; Tyrphostins; Up-Regulation; Urea | 2008 |
Modulation of ileal apical Na+-dependent bile acid transporter ASBT by protein kinase C.
Topics: Bile Acids and Salts; Caco-2 Cells; Calcium; Cell Membrane; Chelating Agents; Chromones; Egtazic Acid; Enzyme Activators; Humans; Ileum; Indoles; Intestinal Mucosa; Kinetics; Maleimides; Morpholines; Organic Anion Transporters, Sodium-Dependent; Peptides; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Protein Kinase Inhibitors; Protein Processing, Post-Translational; Symporters; Tetradecanoylphorbol Acetate; Transfection | 2009 |
Gonadotropin-induced ovarian cancer cell migration and proliferation require extracellular signal-regulated kinase 1/2 activation regulated by calcium and protein kinase C{delta}.
Topics: Acetophenones; Benzopyrans; Calcium; Calcium Channels, L-Type; Cell Line, Tumor; Cell Movement; Cell Proliferation; Dantrolene; Egtazic Acid; Female; Flavonoids; Follicle Stimulating Hormone; Humans; Indoles; Luteinizing Hormone; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Ovarian Neoplasms; Protein Kinase C-delta; RNA, Small Interfering; Signal Transduction; Verapamil | 2010 |
The Mechanism of Ca(2+) Movement in the Involvement of Baicalein-Induced Cytotoxicity in ZR-75-1 Human Breast Cancer Cells.
Topics: Acetylcysteine; Animals; Apoptosis; Boron Compounds; Breast Neoplasms; Calcium; Caspase 3; Caspase 9; Cytosol; Egtazic Acid; Endoplasmic Reticulum; Female; Flavanones; Humans; Indoles; Maleimides; Molecular Structure; Reactive Oxygen Species; Thapsigargin; Type C Phospholipases | 2015 |