Page last updated: 2024-09-03

efonidipine and nitrendipine

efonidipine has been researched along with nitrendipine in 3 studies

Compound Research Comparison

Studies
(efonidipine)
Trials
(efonidipine)
Recent Studies (post-2010)
(efonidipine)
Studies
(nitrendipine)
Trials
(nitrendipine)
Recent Studies (post-2010) (nitrendipine)
12918302,17037883

Protein Interaction Comparison

ProteinTaxonomyefonidipine (IC50)nitrendipine (IC50)
G-protein coupled receptor 55Homo sapiens (human)1.4652
Voltage-dependent L-type calcium channel subunit alpha-1FHomo sapiens (human)0.0152
Cytochrome P450 2C9 Homo sapiens (human)0.3
Voltage-dependent L-type calcium channel subunit alpha-1CRattus norvegicus (Norway rat)0.0013
Voltage-dependent L-type calcium channel subunit alpha-1DRattus norvegicus (Norway rat)0.0013
Cytochrome P450 2C19Homo sapiens (human)3
Voltage-dependent L-type calcium channel subunit alpha-1D Homo sapiens (human)0.0152
Voltage-dependent L-type calcium channel subunit alpha-1SRattus norvegicus (Norway rat)0.0013
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)10
Voltage-dependent L-type calcium channel subunit alpha-1SHomo sapiens (human)0.0152
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)0.0152
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1CHomo sapiens (human)1.85

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (33.33)18.2507
2000's2 (66.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Horinouchi, M; Komada, F; Nishiguchi, K; Ohmoto, N; Ohnishi, N; Okumura, K; Sakaeda, T; Takara, K; Tanigawara, Y; Yokoyama, T1
Kasuya, Y; Masuda, Y; Sakai, T; Tanaka, S; Yamashita, T1
Arai, Y; Fujiwara, M; Harada, M; Kinoshita, H; Kuwabara, Y; Kuwahara, K; Murakami, M; Nakagawa, Y; Nakanishi, M; Nakao, K; Takano, M; Ueshima, K; Yasuno, S1

Other Studies

3 other study(ies) available for efonidipine and nitrendipine

ArticleYear
Effects of 12 Ca2+ antagonists on multidrug resistance, MDR1-mediated transport and MDR1 mRNA expression.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2002, Volume: 16, Issue:3

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Calcium Channel Blockers; Cell Line; Digoxin; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Gene Expression; Humans; Nifedipine; Paclitaxel; RNA, Messenger; Swine; Tritium; Tumor Cells, Cultured; Verapamil; Vinblastine

2002
NZ-105, a new 1,4-dihydropyridine derivative: correlation between dihydropyridine receptor binding and inhibition of calcium uptake in rabbit aorta.
    Japanese journal of pharmacology, 1991, Volume: 57, Issue:3

    Topics: Animals; Antihypertensive Agents; Aorta; Binding, Competitive; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Radioisotopes; Dihydropyridines; In Vitro Techniques; Kinetics; Male; Membranes; Microsomes; Muscle, Smooth, Vascular; Nitrendipine; Nitrophenols; Organophosphorus Compounds; Rabbits; Receptors, Nicotinic; Time Factors; Tritium

1991
T-type Ca2+ channel blockade prevents sudden death in mice with heart failure.
    Circulation, 2009, Sep-01, Volume: 120, Issue:9

    Topics: Animals; Arrhythmias, Cardiac; Autonomic Nervous System; Blood Pressure; Body Weight; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Channels, T-Type; Cardiomyopathy, Dilated; Death, Sudden, Cardiac; Dihydropyridines; Disease Models, Animal; Female; Mibefradil; Mice; Mice, Inbred C57BL; Mice, Transgenic; Myocardial Infarction; Myocytes, Cardiac; Nitrendipine; Nitrophenols; Organophosphorus Compounds; Patch-Clamp Techniques

2009