efavirenz and dpc 961

efavirenz has been researched along with dpc 961 in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's7 (87.50)29.6817
2010's1 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Corbett, JW; Cordova, BC; Erickson-Viitanen, SK; Gearhart, LA; Klabe, RM; Ko, SS; Rodgers, JD1
Anderson, PS; Bacheler, LT; Corbett, JW; Cordova, BC; Diamond, S; Erickson-Viitanen, SK; Garber, S; Gearhart, LA; Jeffrey, S; Klabe, RM; Ko, SS; Logue, K; Magnus, NA; Rodgers, JD; Trainor, GL1
Corbett, JW; Cordova, BC; Erickson-Viitanen, SK; Garber, S; Klabe, RM; Markwalder, JA; Pan, S; Rodgers, JD1
Corbett, JW; Cordova, BC; Erickson-Viitanen, SK; Klabe, RM; Kresge, KJ; Pan, S; Rodgers, JD1
Bacheler, LT; Chidester, DR; Cocuzza, AJ; Cordova, BC; Diamond, S; Erickson-Viitanen, SK; Jeffrey, S; Klabe, RM; Ko, SS; Rodgers, JD; Weigelt, CA1
Kang, X; Kollman, PA; Kuntz, ID; Wang, J1
Bastos, MM; Bezerra, TC; Boechat, N; Costa, CCP; da Silva, FC1
Caballero, J; Castro, EA; Duchowicz, PR; Fernández, FM; Fernández, M1

Reviews

1 review(s) available for efavirenz and dpc 961

ArticleYear
Efavirenz a nonnucleoside reverse transcriptase inhibitor of first-generation: Approaches based on its medicinal chemistry.
    European journal of medicinal chemistry, 2016, Jan-27, Volume: 108

    Topics: Alkynes; Anti-HIV Agents; Benzoxazines; Chemistry, Pharmaceutical; Cyclopropanes; HIV Reverse Transcriptase; HIV-1; Humans; Molecular Conformation; Reverse Transcriptase Inhibitors; Structure-Activity Relationship

2016

Other Studies

7 other study(ies) available for efavirenz and dpc 961

ArticleYear
Novel 2,2-dioxide-4,4-disubstituted-1,3-H-2,1,3-benzothiadiazines as non-nucleoside reverse transcriptase inhibitors.
    Bioorganic & medicinal chemistry letters, 2000, Jan-17, Volume: 10, Issue:2

    Topics: Benzothiadiazines; HIV-1; Humans; Molecular Structure; Reverse Transcriptase Inhibitors

2000
Inhibition of clinically relevant mutant variants of HIV-1 by quinazolinone non-nucleoside reverse transcriptase inhibitors.
    Journal of medicinal chemistry, 2000, May-18, Volume: 43, Issue:10

    Topics: Alkynes; Anti-HIV Agents; Benzoxazines; Blood Proteins; Cyclopropanes; HIV Reverse Transcriptase; HIV-1; Humans; Molecular Structure; Mutation; Oxazines; Protein Binding; Quinazolines; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Virus Replication

2000
3,3a-Dihydropyrano[4,3,2-de]quinazolin-2(1H)-ones are potent non-nucleoside reverse transcriptase inhibitors.
    Bioorganic & medicinal chemistry letters, 2001, Jan-22, Volume: 11, Issue:2

    Topics: Binding Sites; Combinatorial Chemistry Techniques; Drug Resistance; Heterocyclic Compounds, 2-Ring; Heterocyclic Compounds, 3-Ring; HIV Reverse Transcriptase; Humans; Inhibitory Concentration 50; Models, Molecular; Point Mutation; Pyrans; Quinazolines; Reverse Transcriptase Inhibitors; Structure-Activity Relationship

2001
Trifluoromethyl-containing 3-alkoxymethyl- and 3-aryloxymethyl-2-pyridinones are potent inhibitors of HIV-1 non-nucleoside reverse transcriptase.
    Bioorganic & medicinal chemistry letters, 2001, Feb-12, Volume: 11, Issue:3

    Topics: Anti-HIV Agents; Combinatorial Chemistry Techniques; Cytopathogenic Effect, Viral; Enzyme Inhibitors; Fluorine; HIV Reverse Transcriptase; HIV-1; Inhibitory Concentration 50; Mutation; Pyridones; Structure-Activity Relationship

2001
4,1-Benzoxazepinone analogues of efavirenz (Sustiva) as HIV-1 reverse transcriptase inhibitors.
    Bioorganic & medicinal chemistry letters, 2001, Jun-04, Volume: 11, Issue:11

    Topics: Alkynes; Animals; Benzoxazines; Cyclopropanes; HIV Reverse Transcriptase; Humans; Macaca mulatta; Oxazines; Protein Binding; Quinazolines; Quinazolinones; Reverse Transcriptase Inhibitors; Structure-Activity Relationship

2001
Hierarchical database screenings for HIV-1 reverse transcriptase using a pharmacophore model, rigid docking, solvation docking, and MM-PB/SA.
    Journal of medicinal chemistry, 2005, Apr-07, Volume: 48, Issue:7

    Topics: Allosteric Site; Anti-HIV Agents; Crystallography, X-Ray; Databases, Factual; Drug Design; HIV Reverse Transcriptase; Models, Molecular; Molecular Conformation; Molecular Structure; Protein Binding; Quantitative Structure-Activity Relationship; Reverse Transcriptase Inhibitors; Statistics as Topic; Thermodynamics

2005
QSAR for non-nucleoside inhibitors of HIV-1 reverse transcriptase.
    Bioorganic & medicinal chemistry, 2006, Sep-01, Volume: 14, Issue:17

    Topics: Alkynes; Benzoxazines; Combinatorial Chemistry Techniques; Cyclopropanes; HIV Reverse Transcriptase; HIV-1; Molecular Structure; Mutation; Oxazines; Quantitative Structure-Activity Relationship; Quinazolines; Quinazolinones; Reverse Transcriptase Inhibitors

2006
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