Page last updated: 2024-08-25

efaroxan and phentolamine

efaroxan has been researched along with phentolamine in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (42.86)18.2507
2000's3 (42.86)29.6817
2010's1 (14.29)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Agbaba, D; Filipic, S; Nikolic, K1
Chan, SL; Morgan, NG; Stillings, MR1
Dunne, MJ; Hashmi, MN; Kane, C; Shepherd, RM; Squires, PE1
Ammälä, C; Chapman, JC; Cosgrove, KE; Dunne, MJ; Flatt, PR; Giesberts, AN; Hashmi, MN; McClenaghan, NH; Shepherd, RM; White, SJ1
Elliott, J; Morgan, NG; Mourtada, M; Smith, SA1
Fagerholm, V; Haaparanta, M; Scheinin, M1
Henquin, JC; Nenquin, M; Szollosi, A1

Other Studies

7 other study(ies) available for efaroxan and phentolamine

ArticleYear
QSAR study of imidazoline antihypertensive drugs.
    Bioorganic & medicinal chemistry, 2008, Aug-01, Volume: 16, Issue:15

    Topics: Antihypertensive Agents; Binding Sites; Imidazoline Receptors; Imidazolines; Ligands; Models, Molecular; Molecular Structure; Quantitative Structure-Activity Relationship

2008
Mechanisms involved in stimulation of insulin secretion by the hypoglycaemic alpha-adrenergic antagonist, DG-5128.
    Biochemical and biophysical research communications, 1991, May-15, Volume: 176, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Benzofurans; Diazoxide; Dioxanes; Dose-Response Relationship, Drug; Hypoglycemic Agents; Idazoxan; Imidazoles; In Vitro Techniques; Islets of Langerhans; Kinetics; Male; Phentolamine; Rats; Rats, Inbred Strains

1991
Elevation of cytosolic calcium by imidazolines in mouse islets of Langerhans: implications for stimulus-response coupling of insulin release.
    British journal of pharmacology, 1996, Volume: 119, Issue:5

    Topics: Adrenergic alpha-Antagonists; Agmatine; Animals; Benzofurans; Calcium; Cytosol; Down-Regulation; Glucose; Idazoxan; Imidazoles; Imidazoline Receptors; Insulin; Islets of Langerhans; Mice; Phentolamine; Receptors, Drug; Signal Transduction

1996
ATP-sensitive potassium channels and efaroxan-induced insulin release in the electrofusion-derived BRIN-BD11 beta-cell line.
    Diabetes, 1999, Volume: 48, Issue:12

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Adrenergic alpha-Antagonists; Animals; Benzofurans; Cell Fusion; Cell Line; Diazoxide; Glucose; Imidazoles; Insulin; Insulin Secretion; Insulinoma; Islets of Langerhans; Membrane Potentials; Pancreatic Neoplasms; Phentolamine; Pinacidil; Potassium Channels; Tolbutamide; Tumor Cells, Cultured

1999
Effects of imidazoline binding site ligands on the growth and viability of clonal pancreatic beta-cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 2000, Volume: 361, Issue:2

    Topics: Animals; Antazoline; Apoptosis; Benzofurans; Binding Sites; Cell Division; Cell Survival; Idazoxan; Imidazoles; Imidazoline Receptors; Insulin; Insulin Secretion; Islets of Langerhans; PC12 Cells; Phentolamine; Rats; Receptors, Drug

2000
alpha2A-adrenoceptor antagonism increases insulin secretion and synergistically augments the insulinotropic effect of glibenclamide in mice.
    British journal of pharmacology, 2008, Volume: 154, Issue:6

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Atropine Derivatives; Benzofurans; Blood Glucose; Drug Synergism; Fasting; Glyburide; Hypoglycemic Agents; Imidazoles; Insulin; Insulin Secretion; Isoquinolines; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscarinic Antagonists; Naphthyridines; Phentolamine; Propranolol; Receptors, Adrenergic, alpha-2

2008
Pharmacological stimulation and inhibition of insulin secretion in mouse islets lacking ATP-sensitive K+ channels.
    British journal of pharmacology, 2010, Feb-01, Volume: 159, Issue:3

    Topics: Animals; Benzofurans; Calcium; Cytosol; Diazoxide; Female; Imidazoles; Imidazolines; Insulin; Insulin Secretion; Insulin-Secreting Cells; KATP Channels; Mice; Mice, Knockout; Phentolamine; Pinacidil; Potassium Channels; Tolbutamide

2010