efaroxan has been researched along with diazoxide in 11 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 7 (63.64) | 18.2507 |
2000's | 2 (18.18) | 29.6817 |
2010's | 2 (18.18) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Chan, SL; Morgan, NG; Stillings, MR | 1 |
Chan, SL; Dunne, MJ; Morgan, NG; Stillings, MR | 1 |
Chan, SL; Morgan, NG | 1 |
Haque, M; Kulkarni, RN; MacDermot, J; Olmos, G | 1 |
Brown, CA; Morgan, NG | 1 |
Martín-Ruiz, R; Pineda, J; Ruiz-Ortega, JA; Ugedo, L | 1 |
Ammälä, C; Chapman, JC; Cosgrove, KE; Dunne, MJ; Flatt, PR; Giesberts, AN; Hashmi, MN; McClenaghan, NH; Shepherd, RM; White, SJ | 1 |
Chan, SL; Morgan, NG; Mourtada, M | 1 |
Cooper, EJ; Hills, CE; Hudson, AL; Morgan, NG; Parker, CA; Squires, PE | 1 |
Henquin, JC; Nenquin, M; Szollosi, A | 1 |
Adorjan, I; Bauer, L; Belz, M; Brunmair, B; de Cillia, VA; Fenzl, A; Frobel, K; Fürnsinn, C; Gruber, D; Lehner, Z; Luger, A; Rustenbeck, I; Stadlbauer, K | 1 |
11 other study(ies) available for efaroxan and diazoxide
Article | Year |
---|---|
Mechanisms involved in stimulation of insulin secretion by the hypoglycaemic alpha-adrenergic antagonist, DG-5128.
Topics: Adrenergic alpha-Antagonists; Animals; Benzofurans; Diazoxide; Dioxanes; Dose-Response Relationship, Drug; Hypoglycemic Agents; Idazoxan; Imidazoles; In Vitro Techniques; Islets of Langerhans; Kinetics; Male; Phentolamine; Rats; Rats, Inbred Strains | 1991 |
The alpha 2-adrenoceptor antagonist efaroxan modulates K+ATP channels in insulin-secreting cells.
Topics: Adenosine Triphosphate; Adrenergic alpha-Antagonists; Animals; Benzofurans; Diazoxide; Drug Interactions; Imidazoles; Insulin; Insulin Secretion; Islets of Langerhans; Male; Potassium Channels; Rats; Rats, Inbred Strains | 1991 |
Stimulation of insulin secretion by efaroxan may involve interaction with potassium channels.
Topics: Animals; Benzofurans; Diazoxide; Glucose; Hypoglycemic Agents; Imidazoles; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Potassium Channels; Rats; Rats, Inbred Strains | 1990 |
Imidazolines stimulate release of insulin from RIN-5AH cells independently from imidazoline I1 and I2 receptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Affinity Labels; Animals; Benzofurans; Binding, Competitive; Clonidine; Clorgyline; Diazoxide; Dioxanes; Guanidines; Idazoxan; Imidazoles; Imidazoline Receptors; Insulin; Insulinoma; Ligands; Pancreatic Neoplasms; Potassium Channels; Rats; Receptors, Drug; Regression Analysis; Software; Tumor Cells, Cultured | 1994 |
Control of insulin secretion by imidazolines in rat pancreatic islets.
Topics: Animals; Benzofurans; Diazoxide; Dioxanes; Idazoxan; Imidazoles; Insulin; Insulin Secretion; Islets of Langerhans; Rats | 1993 |
Stimulation of locus coeruleus neurons by non-I1/I2-type imidazoline receptors: an in vivo and in vitro electrophysiological study.
Topics: Adenosine Triphosphate; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Benzofurans; Diazoxide; Electrophysiology; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Ligands; Locus Coeruleus; Male; Neurons; Potassium Channels; Rats; Receptors, Adrenergic, alpha-2; Receptors, Drug; Vasodilator Agents | 1998 |
ATP-sensitive potassium channels and efaroxan-induced insulin release in the electrofusion-derived BRIN-BD11 beta-cell line.
Topics: Adenosine Diphosphate; Adenosine Triphosphate; Adrenergic alpha-Antagonists; Animals; Benzofurans; Cell Fusion; Cell Line; Diazoxide; Glucose; Imidazoles; Insulin; Insulin Secretion; Insulinoma; Islets of Langerhans; Membrane Potentials; Pancreatic Neoplasms; Phentolamine; Pinacidil; Potassium Channels; Tolbutamide; Tumor Cells, Cultured | 1999 |
Characterization of a KATP channel-independent pathway involved in potentiation of insulin secretion by efaroxan.
Topics: 1-Methyl-3-isobutylxanthine; Adenosine Triphosphate; Animals; Benzofurans; Bucladesine; Cyclic AMP; Diazoxide; Glucose; Imidazoles; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Permeability; Phosphodiesterase Inhibitors; Potassium Channels; Rats; Rats, Wistar | 2001 |
Comparative effects of efaroxan and beta-carbolines on the secretory activity of rodent and human beta cells.
Topics: Adrenergic alpha-Antagonists; Animals; Benzofurans; Binding Sites; Calcium; Carbolines; Cells, Cultured; Diazoxide; Glucose; Humans; Imidazoles; Insulin; Insulin Secretion; Islets of Langerhans; Ligands; Male; Rats; Rats, Wistar | 2003 |
Pharmacological stimulation and inhibition of insulin secretion in mouse islets lacking ATP-sensitive K+ channels.
Topics: Animals; Benzofurans; Calcium; Cytosol; Diazoxide; Female; Imidazoles; Imidazolines; Insulin; Insulin Secretion; Insulin-Secreting Cells; KATP Channels; Mice; Mice, Knockout; Phentolamine; Pinacidil; Potassium Channels; Tolbutamide | 2010 |
Mechanisms of antihyperglycaemic action of efaroxan in mice: time for reappraisal of α2A-adrenergic antagonism in the treatment of type 2 diabetes?
Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzofurans; Brimonidine Tartrate; Calcium; Cells, Cultured; Diabetes Mellitus, Type 2; Diazoxide; Female; Hyperglycemia; Imidazoles; Insulin; Insulin-Secreting Cells; KATP Channels; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Patch-Clamp Techniques; Quinoxalines; Yohimbine | 2012 |