eedq has been researched along with colforsin in 13 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 4 (30.77) | 18.7374 |
1990's | 8 (61.54) | 18.2507 |
2000's | 1 (7.69) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Iben, L; Meller, E; Yocca, FD | 1 |
Bohmaker, K; Chalfin, M; Meller, E | 1 |
Atkinson, BN; Minneman, KP | 1 |
Nishi, S; Yamada, S; Yokoo, H | 2 |
Bohmaker, K; Goldstein, M; Meller, E; Puza, T | 1 |
Norman, AB; Sanberg, PR; Wachendorf, TJ | 1 |
Battaglia, G; Creese, I; Hess, EJ; Norman, AB | 2 |
Adham, N; Branchek, T; Ellerbrock, B; Hartig, P; Weinshank, RL | 1 |
Aretha, CW; Galloway, MP | 1 |
Maullu, C; Olianas, MC; Onali, P | 1 |
Falardeau, P; Lévesque, D; Mercier, D | 1 |
13 other study(ies) available for eedq and colforsin
Article | Year |
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Lack of apparent receptor reserve at postsynaptic 5-hydroxytryptamine1A receptors negatively coupled to adenylyl cyclase activity in rat hippocampal membranes.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Adrenergic alpha-Antagonists; Animals; Colforsin; Hippocampus; Male; Membranes; Quinolines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Stimulation, Chemical; Substrate Specificity; Synapses; Tetrahydronaphthalenes; Tryptamines | 1992 |
Serotonin 5-HT1A receptor-mediated hypothermia in mice: absence of spare receptors and rapid induction of tolerance.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Body Temperature; Colforsin; Drug Tolerance; Fenclonine; Hypothermia; Male; Mice; Pindolol; Piperazines; Quinolines; Receptors, Serotonin; Serotonin | 1992 |
Occupancy-response relationships for beta- and alpha 2-adrenergic receptors exerting opposing effects on cAMP production.
Topics: Adrenergic alpha-Antagonists; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Isoproterenol; Kinetics; Neuroglia; Norepinephrine; Pindolol; Quinolines; Rats; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1992 |
[Regulation of (-)-sulpiride-induced increase in evoked dopamine release from striatal slices in rat].
Topics: Animals; Apomorphine; Benzazepines; Colforsin; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Electric Stimulation; Evoked Potentials; Male; Quinolines; Rats; Rats, Wistar; Sulpiride | 1992 |
Absence of spare autoreceptors regulating dopamine agonist inhibition of tyrosine hydroxylation in slices of rat striatum.
Topics: Animals; Colforsin; Corpus Striatum; Dopamine Agents; Dose-Response Relationship, Drug; In Vitro Techniques; Indoles; Male; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Tyrosine 3-Monooxygenase | 1989 |
Differential effect of N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ) on [3H]SCH23390 and [3H]forskolin binding in rat striatum.
Topics: Animals; Benzazepines; Binding Sites; Colforsin; Corpus Striatum; Guanylyl Imidodiphosphate; In Vitro Techniques; Magnesium; Magnesium Chloride; Male; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Second Messenger Systems; Sodium Fluoride | 1989 |
Functional recovery of D1 dopamine receptor-mediated stimulation of rat striatal adenylate cyclase activity following irreversible receptor modification by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ): evidence for spare receptors.
Topics: Adenylyl Cyclases; Animals; Colforsin; Corpus Striatum; Guanosine Triphosphate; Male; Neurons; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1 | 1986 |
Differential modification of striatal D1 dopamine receptors and effector moieties by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline in vivo and in vitro.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Benzazepines; Colforsin; Corpus Striatum; Dopamine; Enzyme Activation; GTP-Binding Proteins; Male; Quinolines; Rats; Receptors, Dopamine | 1987 |
Receptor reserve masks partial agonist activity of drugs in a cloned rat 5-hydroxytryptamine1B receptor expression system.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cell Line; Cloning, Molecular; Colforsin; Cyclic AMP; Iodocyanopindolol; Pindolol; Quinolines; Radioligand Assay; Rats; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Transfection; Virulence Factors, Bordetella | 1993 |
Modulation of (-)-sulpiride-induced increase in electrically-evoked release of dopamine from rat striatal slices.
Topics: Adrenergic alpha-Antagonists; Animals; Apomorphine; Benzazepines; Colforsin; Corpus Striatum; Dopamine; Dopamine Antagonists; Drug Interactions; Electric Stimulation; Kinetics; Male; Quinolines; Rats; Rats, Wistar; Sulpiride | 1993 |
Dopamine autoreceptor reserve in vitro: possible role of dopamine D3 receptors.
Topics: Adenylyl Cyclases; Alkylation; Animals; Colforsin; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Drug Interactions; Male; Olfactory Pathways; Potassium; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes | 1996 |
Effects of clozapine on rat striatal muscarinic receptors coupled to inhibition of adenylyl cyclase activity and on the human cloned m4 receptor.
Topics: Adenylyl Cyclases; Alkylation; Animals; Cell Membrane; CHO Cells; Clozapine; Colforsin; Corpus Striatum; Cricetinae; Cyclic AMP; Guanosine 5'-O-(3-Thiotriphosphate); Humans; In Vitro Techniques; Male; Muscarinic Antagonists; N-Methylscopolamine; Protein Binding; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Synaptosomes | 1997 |
Autoreceptor preference of dopamine D2 receptor agonists correlates with preferential coupling to cyclic AMP.
Topics: Adenylate Cyclase Toxin; Alkylating Agents; Animals; Autoreceptors; Brain; Cells, Cultured; Colforsin; Cyclic AMP; DNA, Complementary; Dopamine; Dopamine Agonists; Fibroblasts; Inositol 1,4,5-Trisphosphate; Linear Models; Mice; Movement; Neural Inhibition; Neurons; Quinolines; Receptors, Dopamine D2; Signal Transduction; Synaptic Transmission; Transfection; Virulence Factors, Bordetella | 2001 |