Page last updated: 2024-08-23

eedq and colforsin

eedq has been researched along with colforsin in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19904 (30.77)18.7374
1990's8 (61.54)18.2507
2000's1 (7.69)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Iben, L; Meller, E; Yocca, FD1
Bohmaker, K; Chalfin, M; Meller, E1
Atkinson, BN; Minneman, KP1
Nishi, S; Yamada, S; Yokoo, H2
Bohmaker, K; Goldstein, M; Meller, E; Puza, T1
Norman, AB; Sanberg, PR; Wachendorf, TJ1
Battaglia, G; Creese, I; Hess, EJ; Norman, AB2
Adham, N; Branchek, T; Ellerbrock, B; Hartig, P; Weinshank, RL1
Aretha, CW; Galloway, MP1
Maullu, C; Olianas, MC; Onali, P1
Falardeau, P; Lévesque, D; Mercier, D1

Other Studies

13 other study(ies) available for eedq and colforsin

ArticleYear
Lack of apparent receptor reserve at postsynaptic 5-hydroxytryptamine1A receptors negatively coupled to adenylyl cyclase activity in rat hippocampal membranes.
    Molecular pharmacology, 1992, Volume: 41, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Adrenergic alpha-Antagonists; Animals; Colforsin; Hippocampus; Male; Membranes; Quinolines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Stimulation, Chemical; Substrate Specificity; Synapses; Tetrahydronaphthalenes; Tryptamines

1992
Serotonin 5-HT1A receptor-mediated hypothermia in mice: absence of spare receptors and rapid induction of tolerance.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 43, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Body Temperature; Colforsin; Drug Tolerance; Fenclonine; Hypothermia; Male; Mice; Pindolol; Piperazines; Quinolines; Receptors, Serotonin; Serotonin

1992
Occupancy-response relationships for beta- and alpha 2-adrenergic receptors exerting opposing effects on cAMP production.
    Receptor, 1992,Fall, Volume: 2, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Isoproterenol; Kinetics; Neuroglia; Norepinephrine; Pindolol; Quinolines; Rats; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1992
[Regulation of (-)-sulpiride-induced increase in evoked dopamine release from striatal slices in rat].
    Yakubutsu, seishin, kodo = Japanese journal of psychopharmacology, 1992, Volume: 12, Issue:4

    Topics: Animals; Apomorphine; Benzazepines; Colforsin; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Electric Stimulation; Evoked Potentials; Male; Quinolines; Rats; Rats, Wistar; Sulpiride

1992
Absence of spare autoreceptors regulating dopamine agonist inhibition of tyrosine hydroxylation in slices of rat striatum.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:1

    Topics: Animals; Colforsin; Corpus Striatum; Dopamine Agents; Dose-Response Relationship, Drug; In Vitro Techniques; Indoles; Male; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Tyrosine 3-Monooxygenase

1989
Differential effect of N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ) on [3H]SCH23390 and [3H]forskolin binding in rat striatum.
    Life sciences, 1989, Volume: 44, Issue:13

    Topics: Animals; Benzazepines; Binding Sites; Colforsin; Corpus Striatum; Guanylyl Imidodiphosphate; In Vitro Techniques; Magnesium; Magnesium Chloride; Male; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Second Messenger Systems; Sodium Fluoride

1989
Functional recovery of D1 dopamine receptor-mediated stimulation of rat striatal adenylate cyclase activity following irreversible receptor modification by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ): evidence for spare receptors.
    Neuroscience letters, 1986, Sep-12, Volume: 69, Issue:3

    Topics: Adenylyl Cyclases; Animals; Colforsin; Corpus Striatum; Guanosine Triphosphate; Male; Neurons; Quinolines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1

1986
Differential modification of striatal D1 dopamine receptors and effector moieties by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline in vivo and in vitro.
    Molecular pharmacology, 1987, Volume: 31, Issue:1

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Benzazepines; Colforsin; Corpus Striatum; Dopamine; Enzyme Activation; GTP-Binding Proteins; Male; Quinolines; Rats; Receptors, Dopamine

1987
Receptor reserve masks partial agonist activity of drugs in a cloned rat 5-hydroxytryptamine1B receptor expression system.
    Molecular pharmacology, 1993, Volume: 43, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cell Line; Cloning, Molecular; Colforsin; Cyclic AMP; Iodocyanopindolol; Pindolol; Quinolines; Radioligand Assay; Rats; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Transfection; Virulence Factors, Bordetella

1993
Modulation of (-)-sulpiride-induced increase in electrically-evoked release of dopamine from rat striatal slices.
    The Journal of pharmacy and pharmacology, 1993, Volume: 45, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Apomorphine; Benzazepines; Colforsin; Corpus Striatum; Dopamine; Dopamine Antagonists; Drug Interactions; Electric Stimulation; Kinetics; Male; Quinolines; Rats; Rats, Wistar; Sulpiride

1993
Dopamine autoreceptor reserve in vitro: possible role of dopamine D3 receptors.
    European journal of pharmacology, 1996, Jun-03, Volume: 305, Issue:1-3

    Topics: Adenylyl Cyclases; Alkylation; Animals; Colforsin; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Drug Interactions; Male; Olfactory Pathways; Potassium; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes

1996
Effects of clozapine on rat striatal muscarinic receptors coupled to inhibition of adenylyl cyclase activity and on the human cloned m4 receptor.
    British journal of pharmacology, 1997, Volume: 122, Issue:3

    Topics: Adenylyl Cyclases; Alkylation; Animals; Cell Membrane; CHO Cells; Clozapine; Colforsin; Corpus Striatum; Cricetinae; Cyclic AMP; Guanosine 5'-O-(3-Thiotriphosphate); Humans; In Vitro Techniques; Male; Muscarinic Antagonists; N-Methylscopolamine; Protein Binding; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Synaptosomes

1997
Autoreceptor preference of dopamine D2 receptor agonists correlates with preferential coupling to cyclic AMP.
    Neuroreport, 2001, May-25, Volume: 12, Issue:7

    Topics: Adenylate Cyclase Toxin; Alkylating Agents; Animals; Autoreceptors; Brain; Cells, Cultured; Colforsin; Cyclic AMP; DNA, Complementary; Dopamine; Dopamine Agonists; Fibroblasts; Inositol 1,4,5-Trisphosphate; Linear Models; Mice; Movement; Neural Inhibition; Neurons; Quinolines; Receptors, Dopamine D2; Signal Transduction; Synaptic Transmission; Transfection; Virulence Factors, Bordetella

2001