edrophonium and physostigmine

edrophonium has been researched along with physostigmine in 35 studies

Research

Studies (35)

TimeframeStudies, this research(%)All Research%
pre-199027 (77.14)18.7374
1990's4 (11.43)18.2507
2000's1 (2.86)29.6817
2010's2 (5.71)24.3611
2020's1 (2.86)2.80

Authors

AuthorsStudies
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Hecker, SE; Mitchelson, F1
DeFrance, JF; Kitai, ST; McCrea, RA; Yoshihara, H1
Kato, G; Robaire, B1
Artusio, JF; Okamoto, M; Riker, WF; Walewski, JL1
Giacobini, E; Ogane, N; Struble, R1
Kawashima, K; Kobayashi, N; Onishi, Y; Otsuka, M; Sakuma, M; Yanagisawa, M; Yoshioka, K1
Fiekers, JF1
Allen, CN; Carpenter, DO; Evans, ML; Hori, N; Oyama, Y1
Albuquerque, EX; Aracava, Y; Brossi, A; Cintra, WM; Deshpande, SS; Schönenberger, B1
Gandiha, A; Lord, JA; Marshall, IG1
Manganiello, VC; Stoner, JS; Vaughan, M1
Klawans, HL; Rubovits, R2
Flacke, W1
Hunter, AR; Pleuvry, BJ2
Schneider, R1
Brezenoff, HE1
Turner, P; Variava, DM1
Goodkin, P; Howard, BD1
Phillis, JW; York, DH1
Emson, PC; Kerkut, GA1
Kerkut, GA; Pitman, RM; Walker, RJ1
Tebecis, AK1
Kerkut, GA; Oliver, GW; Rick, JT; Walker, RJ1
Hein, GE; Powell, K1
Edge, ND1
Biggs, DF; Wasarab, DE1
Giovannini, E; Romani, R; Rosi, G; Talesa, V1
BOWMAN, WC1
VANMAANEN, EF1
Rakonczay, Z1
Kennedy, RT; Li, Q; Pei, J1
Barohn, RJ; Katz, NK1

Reviews

4 review(s) available for edrophonium and physostigmine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Structure-activity relationship of reversible cholinesterase inhibitors: activation, channel blockade and stereospecificity of the nicotinic acetylcholine receptor-ion channel complex.
    Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas, 1988, Volume: 21, Issue:6

    Topics: Animals; Binding Sites; Chemical Phenomena; Chemistry; Cholinesterase Inhibitors; Edrophonium; Muscle Contraction; Neostigmine; Organophosphate Poisoning; Physostigmine; Pyridostigmine Bromide; Rana pipiens; Receptors, Nicotinic; Sciatic Nerve; Structure-Activity Relationship

1988
Treatment of myasthenia gravis.
    The New England journal of medicine, 1973, Jan-04, Volume: 288, Issue:1

    Topics: Acetates; Adrenal Cortex Hormones; Adrenocorticotropic Hormone; Ambenonium Chloride; Aminophylline; Anesthetics, Local; Anti-Arrhythmia Agents; Anti-Bacterial Agents; Atropine; Bromides; Choline; Cholinesterase Inhibitors; Edrophonium; Hospitals, Special; Humans; Myasthenia Gravis; Neostigmine; Physostigmine; Phytotherapy; Plants, Medicinal; Plants, Toxic; Synaptic Transmission; United States; Veratrum

1973
The history of acetylcholinesterase inhibitors in the treatment of myasthenia gravis.
    Neuropharmacology, 2021, Volume: 182

    Topics: Acetylcholinesterase; Cholinesterase Inhibitors; Curare; Edrophonium; History, 19th Century; History, 20th Century; History, 21st Century; Humans; Myasthenia Gravis; Physicians; Physostigmine

2021

Trials

1 trial(s) available for edrophonium and physostigmine

ArticleYear
Pharmacological studies on a cholinergic inhibition in the cerebral cortex.
    Brain research, 1968, Volume: 10, Issue:3

    Topics: Acetylcholine; Atropine; Cerebral Cortex; Cholinesterase Inhibitors; Clinical Trials as Topic; Depression, Chemical; Edrophonium; Gallamine Triethiodide; Hypothalamus; Neostigmine; Neurons; Parasympathomimetics; Physostigmine; Pyramidal Tracts; Scopolamine; Sensory Receptor Cells; Strychnine; Time Factors; Tubocurarine

1968

Other Studies

30 other study(ies) available for edrophonium and physostigmine

ArticleYear
The effect of cholinesterase inhibitors on the antimuscarinic effect of hemicholinium-3 (HC-3) in the rat.
    The Journal of pharmacy and pharmacology, 1976, Volume: 28, Issue:5

    Topics: Animals; Benzenaminium, 4,4'-(3-oxo-1,5-pentanediyl)bis(N,N-dimethyl-N-2-propenyl-), Dibromide; Carbachol; Cholinesterase Inhibitors; Edrophonium; Hemicholinium 3; Ileum; Isoflurophate; Male; Parasympatholytics; Physostigmine; Rats; Receptors, Cholinergic; Urinary Bladder

1976
Pharmacology of the inhibiton in the lateral septal region.
    Experimental neurology, 1975, Volume: 48, Issue:3 Pt 1

    Topics: Acetylcholine; Animals; Atropine; Bicuculline; Cats; Depression, Chemical; Edrophonium; gamma-Aminobutyric Acid; Membrane Potentials; Neural Inhibition; Physostigmine; Septal Nuclei; Septum Pellucidum; Strychnine; Tubocurarine

1975
Effects of edrophonium, eserine, decamethonium, d-tubocurarine, and gallamine on the kinetics of membrane-bound and solubilized eel acetylcholinesterase.
    Molecular pharmacology, 1975, Volume: 11, Issue:6

    Topics: Acetylcholinesterase; Animals; Binding, Competitive; Centrifugation, Density Gradient; Decamethonium Compounds; Edrophonium; Electric Organ; Electrophorus; Gallamine Triethiodide; Kinetics; Membranes; Physostigmine; Protein Binding; Tubocurarine

1975
Neuromuscular pharmacology in rat neonates: development of responsiveness to prototypic blocking and reversal drugs.
    Anesthesia and analgesia, 1992, Volume: 75, Issue:3

    Topics: 4-Aminopyridine; Aging; Animals; Animals, Newborn; Cholinesterase Inhibitors; Curare; Dose-Response Relationship, Drug; Drug Synergism; Edrophonium; Fasciculation; Female; Male; Muscle Contraction; Neostigmine; Nerve Endings; Neuromuscular Blocking Agents; Neuromuscular Junction; Physostigmine; Rats; Rats, Inbred Strains; Succinylcholine; Synaptic Transmission; Tubocurarine

1992
Differential inhibition of acetylcholinesterase molecular forms in normal and Alzheimer disease brain.
    Brain research, 1992, Sep-04, Volume: 589, Issue:2

    Topics: Acetylcholinesterase; Aged; Alzheimer Disease; Brain; Centrifugation, Density Gradient; Cholinesterase Inhibitors; Edrophonium; Female; Humans; Male; Physostigmine; Protein Conformation; Sucrose

1992
Substance P-evoked release of acetylcholine from isolated spinal cord of the newborn rat.
    Neuroscience, 1991, Volume: 45, Issue:2

    Topics: Acetylcholine; Animals; Animals, Newborn; Calcium; Dihydro-beta-Erythroidine; Edrophonium; Neurokinin A; Neurokinin B; Peptide Fragments; Physostigmine; Potassium; Rats; Rats, Inbred Strains; Secretory Rate; Spinal Cord; Stimulation, Chemical; Substance P; Tetrodotoxin; Veratridine

1991
Interactions of edrophonium, physostigmine and methanesulfonyl fluoride with the snake end-plate acetylcholine receptor-channel complex.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 234, Issue:3

    Topics: Acetylcholine; Animals; Cholinesterase Inhibitors; Edrophonium; In Vitro Techniques; Ion Channels; Membrane Potentials; Motor Endplate; Neostigmine; Neuromuscular Junction; Physostigmine; Receptors, Cholinergic; Snakes; Sulfones

1985
Electrophysiological estimation of the actions of acetylcholinesterase inhibitors on acetylcholine receptor and cholinesterase in physically isolated Aplysia neurones.
    British journal of pharmacology, 1989, Volume: 96, Issue:3

    Topics: Animals; Aplysia; Cholinesterase Inhibitors; Cholinesterases; Edrophonium; Electrophysiology; In Vitro Techniques; Isoflurophate; Neurons; Physostigmine; Receptors, Cholinergic; Time Factors

1989
Further studies on the site of action of nicotinic blocking drugs.
    European journal of pharmacology, 1973, Volume: 23, Issue:2

    Topics: Acetylcholine; Animals; Binding Sites; Chickens; Choline; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Edrophonium; Electric Stimulation; Ganglionic Blockers; Hexamethonium Compounds; In Vitro Techniques; Muscles; Neuromuscular Junction; Physostigmine; Quaternary Ammonium Compounds; Tubocurarine

1973
Guanosine cyclic 3',5'-monophosphate and guanylate cyclase activity in guinea pig lung: effects of acetylcholine and cholinesterase inhibitors.
    Molecular pharmacology, 1974, Volume: 10, Issue:1

    Topics: Acetylcholine; Animals; Chromatography, DEAE-Cellulose; Cyclic AMP; Cyclic GMP; Edrophonium; Epinephrine; Female; Guanylate Cyclase; Guinea Pigs; Isoproterenol; Lung; Neostigmine; Phentolamine; Physostigmine; Propranolol; Prostaglandins; Serotonin; Theophylline; Time Factors; Tritium

1974
Central cholinergic-anticholinergic antagonism in Huntington's chorea.
    Neurology, 1972, Volume: 22, Issue:2

    Topics: Acetylcholine; Dopamine; Drug Antagonism; Edrophonium; Humans; Huntington Disease; Parasympatholytics; Physostigmine; Scopolamine; Tongue

1972
A quantitative comparison of the antagonism of tubocurarine and diallylnortoxiferine by four anticurare agents.
    The Journal of pharmacy and pharmacology, 1967, Volume: 19, Issue:11

    Topics: Ambenonium Chloride; Animals; Cholinesterase Inhibitors; Curare; Diaphragm; Drug Antagonism; Edrophonium; Electric Stimulation; Muscle Contraction; Neostigmine; Phrenic Nerve; Physostigmine; Rats; Toxiferine; Tubocurarine

1967
A test for the assessment of the duration of the action of neostigmine and of the relative potencies of various anticholinesterases using the pupil of the mouse.
    The Journal of pharmacy and pharmacology, 1970, Volume: 22, Issue:4

    Topics: Animals; Atropine; Cholinesterase Inhibitors; Edrophonium; Female; Male; Methods; Mice; Miotics; Neostigmine; Physostigmine; Pupil; Pyridostigmine Bromide; Time Factors

1970
Effect of cholinergic and anticholinergic agents on tardive dyskinesia.
    Journal of neurology, neurosurgery, and psychiatry, 1974, Volume: 37, Issue:8

    Topics: Adult; Aged; Anxiety Disorders; Edrophonium; Female; Humans; Male; Middle Aged; Movement Disorders; Neurocognitive Disorders; Physostigmine; Schizophrenia; Scopolamine; Tranquilizing Agents

1974
Cardiovascular responses to intrahypothalamic injections of carbachol and certain cholinesterase inhibitors.
    Neuropharmacology, 1972, Volume: 11, Issue:5

    Topics: Animals; Blood Pressure; Carbachol; Cholinesterase Inhibitors; Edrophonium; Electrocardiography; Heart Rate; Hemodynamics; Hypothalamus; Male; Microinjections; Neostigmine; Physostigmine; Rats

1972
Comparison of the potencies of edrophonium, neostigmine and eserine with a new anticholinesterase drug RX 67668 on human tissues.
    British journal of pharmacology, 1973, Volume: 47, Issue:3

    Topics: Cholinesterase Inhibitors; Colon; Cyclohexanes; Edrophonium; Humans; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Neostigmine; Physostigmine; Pyrrolidines; Stomach

1973
Studies on acetylcholinesterase of rat brain synaptosomal plasma membranes.
    Journal of neurochemistry, 1974, Volume: 22, Issue:1

    Topics: Acetylcholinesterase; Acridines; Allosteric Regulation; Animals; Brain; Cell Membrane; Centrifugation, Density Gradient; Cholinesterase Inhibitors; Chromatography, Affinity; Decamethonium Compounds; Edrophonium; Female; Gallamine Triethiodide; Hydrogen-Ion Concentration; Kinetics; Osmolar Concentration; Physostigmine; Pyridinium Compounds; Rats; Solubility; Spectrometry, Fluorescence; Surface-Active Agents; Synaptosomes; Tubocurarine

1974
Acetylcholinesterase in snail brain.
    Comparative biochemistry and physiology. B, Comparative biochemistry, 1971, Aug-15, Volume: 39, Issue:4

    Topics: Acetylcholine; Acetylcholinesterase; Acridines; Animals; Brain; Calcium Chloride; Carbachol; Cholinesterase Inhibitors; Detergents; Edrophonium; Electrophoresis, Disc; Enzyme Activation; Hydrogen-Ion Concentration; Kinetics; Magnesium; Molecular Weight; Physostigmine; Potassium Chloride; Snails; Sodium Chloride; Spectrophotometry; Subcellular Fractions; Sulfuric Acids; Tubocurarine; Urea

1971
Iontophoretic application of acetylcholine and GABA onto insect central neurones.
    Comparative biochemistry and physiology, 1969, Nov-15, Volume: 31, Issue:4

    Topics: Acetylcholine; Action Potentials; Aminobutyrates; Animals; Atropine; Carbachol; Central Nervous System; Chlorides; Dopamine; Edrophonium; Electrodes; Electrophoresis; Electrophysiology; Epinephrine; Glycine; Hydrogen-Ion Concentration; Insecta; Methacholine Compounds; Neostigmine; Neurons; Nicotine; Norepinephrine; Physostigmine; Pilocarpine; Potassium; Sodium; Synapses; Time Factors; Tubocurarine

1969
Properties of cholinoceptive neurones in the medial geniculate nucleus.
    British journal of pharmacology, 1970, Volume: 38, Issue:1

    Topics: Acetylcholine; Anesthesia, General; Animals; Cats; Depression, Chemical; Drug Synergism; Edrophonium; Evoked Potentials; Female; Geniculate Bodies; Glutamates; Male; Neostigmine; Parasympatholytics; Parasympathomimetics; Physostigmine; Stimulation, Chemical

1970
The effects of drugs on learning in a simple preparation.
    Comparative and general pharmacology, 1970, Volume: 1, Issue:4

    Topics: Amphetamine; Animals; Behavior, Animal; Carbon Isotopes; Chloramphenicol; Cholinesterases; Cockroaches; Congo Red; Cycloheximide; Dactinomycin; Dose-Response Relationship, Drug; Edrophonium; Ganglia; Learning; Leucine; Memory; Neostigmine; Pemoline; Physostigmine; RNA; Temperature; Time Factors; Uridine

1970
Antagonists to neuromuscular blocking agents. An experimental study.
    British journal of anaesthesia, 1968, Volume: 40, Issue:10

    Topics: Acetylcholine; Ambenonium Chloride; Animals; Anura; Curare; Diaphragm; Drug Synergism; Edrophonium; Heart; Heart Arrest; In Vitro Techniques; Mice; Muscles; Neostigmine; Physostigmine; Rabbits; Rats; Stimulation, Chemical; Toxiferine; Tubocurarine

1968
Evaluation of kinetic constants for mixed inhibitors of cholinesterase.
    Biochemical pharmacology, 1967, Volume: 16, Issue:3

    Topics: Animals; Bridged-Ring Compounds; Cattle; Cholinesterase Inhibitors; Cholinesterases; Edrophonium; Hallucinogens; Kinetics; Levallorphan; Lysergic Acid Diethylamide; Mathematics; Morphine; Nalorphine; Neostigmine; Phenazocine; Phenethylamines; Phenols; Physostigmine; Quaternary Ammonium Compounds

1967
pPy: a measure of potentiating activity.
    Nature, 1967, Dec-09, Volume: 216, Issue:5119

    Topics: Acetylcholine; Animals; Anura; Cholinesterase Inhibitors; Curare; Edrophonium; Isoflurophate; Muscle Contraction; Muscles; Neostigmine; Physostigmine

1967
Effects of drugs on miniature excitatory potentials in the adductor superficialis pectoralis muscle of the rainbow trout (Salmo gairdneri).
    Proceedings of the Western Pharmacology Society, 1980, Volume: 23

    Topics: Animals; Cations; Edrophonium; Electric Stimulation; Evoked Potentials; Membrane Potentials; Muscles; Nerve Endings; Physostigmine; Salmonidae; Trout

1980
Acetylcholinesterase in Dendrobaena veneta (Oligochaeta: Opisthopora) is present with forms sensitive and insensitive to phosphatidylinositol phospholipase C. Biochemical characterization and histochemical localization in the nervous system.
    European journal of biochemistry, 1996, Jun-01, Volume: 238, Issue:2

    Topics: Acetylcholinesterase; Animals; Centrifugation, Density Gradient; Cholinesterase Inhibitors; Chromatography, Gel; Disulfides; Edrophonium; Electrophoresis, Polyacrylamide Gel; Enzyme Inhibitors; Histocytochemistry; Kinetics; Molecular Weight; Nervous System; Oligochaeta; Phosphatidylinositol Diacylglycerol-Lyase; Phosphoric Diester Hydrolases; Physostigmine; Procainamide; Protein Conformation

1996
The neuromuscular blocking action of benzoquinonium chloride in the cat and in the hen.
    British journal of pharmacology and chemotherapy, 1958, Volume: 13, Issue:4

    Topics: Acetylcholine; Animals; Cats; Chickens; Cholinesterase Inhibitors; Cholinesterases; Edrophonium; Female; Muscle Relaxants, Central; Muscle, Skeletal; Neostigmine; Neuromuscular Blockade; Neuromuscular Diseases; Nicotinic Antagonists; Paralysis; Physostigmine; Quaternary Ammonium Compounds; Synaptic Transmission

1958
THE ANTI-TUBOCURARINE EFFECTS OF PHYSOSTIGMINE, NEOSTIGMINE, AND EDROPHONIUM IN THE RAT.
    Naunyn-Schmiedebergs Archiv fur experimentelle Pathologie und Pharmakologie, 1964, May-25, Volume: 248

    Topics: Acetylcholine; Cholinesterase Inhibitors; Edrophonium; Electric Stimulation; Neostigmine; Neuromuscular Junction; Neuromuscular Nondepolarizing Agents; Pharmacology; Physostigmine; Rats; Research; Tubocurarine

1964
Potencies and selectivities of inhibitors of acetylcholinesterase and its molecular forms in normal and Alzheimer's disease brain.
    Acta biologica Hungarica, 2003, Volume: 54, Issue:2

    Topics: Acetylcholinesterase; Alzheimer Disease; Benzazepines; Brain; Butyrylcholinesterase; Carbamates; Cerebral Cortex; Cholinesterase Inhibitors; Edrophonium; Humans; In Vitro Techniques; Phenylcarbamates; Physostigmine; Rivastigmine; Tacrine; Trichlorfon

2003
Rapid and label-free screening of enzyme inhibitors using segmented flow electrospray ionization mass spectrometry.
    Journal of the American Society for Mass Spectrometry, 2010, Volume: 21, Issue:7

    Topics: Acetylcholine; Acetylcholinesterase; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Edrophonium; Linear Models; Malathion; Neostigmine; Physostigmine; Spectrometry, Mass, Electrospray Ionization

2010