Page last updated: 2024-09-02

ecopipam and raclopride

ecopipam has been researched along with raclopride in 15 studies

Compound Research Comparison

Studies
(ecopipam)
Trials
(ecopipam)
Recent Studies (post-2010)
(ecopipam)
Studies
(raclopride)
Trials
(raclopride)
Recent Studies (post-2010) (raclopride)
14718341,802132419

Protein Interaction Comparison

ProteinTaxonomyecopipam (IC50)raclopride (IC50)
D(2) dopamine receptorHomo sapiens (human)0.052
D(2) dopamine receptorMus musculus (house mouse)0.032
D(2) dopamine receptorRattus norvegicus (Norway rat)0.0279

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (53.33)18.2507
2000's4 (26.67)29.6817
2010's2 (13.33)24.3611
2020's1 (6.67)2.80

Authors

AuthorsStudies
Goldman-Rakic, PS; Sawaguchi, T2
Balster, RL; Jortani, SA; Mansbach, RS1
Cools, AR; Ellenbroek, BA; Prinssen, EP; Stamatovic, B1
Chausmer, AL; Ettenberg, A1
Hicks, PB; Richter, TJ; Trompler, RA; Wadenberg, ML; Young, KA; Zavodny, RA1
Gold, LH; Weed, MR1
Handley, SL; McCreary, AC1
Bassareo, V; Di Chiara, G; Fenu, S1
Goldman-Rakic, PS; Vijayraghavan, S; Wang, M1
Di Chiara, G; Fenu, S; Rivas, E2
Li, Y; Liu, X; Mishra, PK; Patel, KP; Zheng, H1
Enomoto, T; Ikeda, K; Konoike, N; Nakamura, K; Takemoto, A1
Hashimoto, H; Hayashida, M; Hirato, Y; Kasai, A; Niu, M; Seiriki, K; Tanuma, M; Yokoyama, R1

Other Studies

15 other study(ies) available for ecopipam and raclopride

ArticleYear
D1 dopamine receptors in prefrontal cortex: involvement in working memory.
    Science (New York, N.Y.), 1991, Feb-22, Volume: 251, Issue:4996

    Topics: Animals; Benzazepines; Cerebral Cortex; Dopamine Antagonists; Macaca mulatta; Memory; Raclopride; Receptors, Dopamine; Receptors, Dopamine D1; Salicylamides; Visual Perception

1991
Discriminative stimulus effects of esteratic local anesthetics in squirrel monkeys.
    European journal of pharmacology, 1995, Feb-14, Volume: 274, Issue:1-3

    Topics: Aminobenzoates; Anesthetics, Local; Animals; Benzazepines; Binding, Competitive; Carrier Proteins; Cocaine; Dopamine; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Propanolamines; Raclopride; Regression Analysis; Saimiri; Salicylamides; Substance-Related Disorders

1995
The role of D1-dopamine receptor in working memory: local injections of dopamine antagonists into the prefrontal cortex of rhesus monkeys performing an oculomotor delayed-response task.
    Journal of neurophysiology, 1994, Volume: 71, Issue:2

    Topics: Animals; Antipsychotic Agents; Appetitive Behavior; Attention; Benzazepines; Dominance, Cerebral; Dopamine; Dopamine Antagonists; Eye Movements; Fixation, Ocular; Haloperidol; Injections; Ketanserin; Macaca mulatta; Male; Mental Recall; Orientation; Prefrontal Cortex; Raclopride; Reaction Time; Receptors, Dopamine D1; Saccades; Salicylamides; Sulpiride

1994
The effects of haloperidol and raclopride in the paw test are influenced similarly by SCH 39166.
    European journal of pharmacology, 1993, Feb-09, Volume: 231, Issue:2

    Topics: Animals; Antipsychotic Agents; Basal Ganglia Diseases; Behavior, Animal; Benzazepines; Dopamine D2 Receptor Antagonists; Drug Interactions; Forelimb; Haloperidol; Hindlimb; Male; Raclopride; Rats; Rats, Wistar; Reaction Time; Receptors, Dopamine D1; Salicylamides

1993
A role for D2, but not D1, dopamine receptors in the response-reinstating effects of food reinforcement.
    Pharmacology, biochemistry, and behavior, 1997, Volume: 57, Issue:4

    Topics: Animals; Benzazepines; Conditioning, Operant; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Food; Male; Motor Activity; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Reinforcement, Psychology; Reward; Salicylamides

1997
A novel computer-controlled conditioned avoidance apparatus for rats.
    Journal of pharmacological and toxicological methods, 1997, Volume: 38, Issue:4

    Topics: Amphetamines; Animals; Antipsychotic Agents; Avoidance Learning; Benzazepines; Clozapine; Computers; Cross-Over Studies; Dopamine Antagonists; Fluorobenzenes; Haloperidol; Male; Physical Conditioning, Animal; Piperidines; Raclopride; Rats; Rats, Sprague-Dawley; Salicylamides; Serotonin Antagonists; Serotonin Receptor Agonists

1997
The effects of dopaminergic agents on reaction time in rhesus monkeys.
    Psychopharmacology, 1998, Volume: 137, Issue:1

    Topics: Animals; Benzazepines; Dextroamphetamine; Dopamine Agents; Dose-Response Relationship, Drug; Macaca mulatta; Male; Motor Activity; Raclopride; Reaction Time; Salicylamides

1998
The thyrotrophin-releasing hormone analogue MK771 induces tic-like behaviours: the effects of dopamine D1 and D2 receptor antagonists.
    European journal of pharmacology, 1999, Mar-12, Volume: 369, Issue:1

    Topics: Animals; Antidepressive Agents; Behavior, Animal; Behavioral Symptoms; Benzazepines; Blinking; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Male; Mice; Raclopride; Receptors, Dopamine D1; Salicylamides; Sulpiride; Thiazolidines; Thyrotropin-Releasing Hormone; Tic Disorders

1999
A role for dopamine D1 receptors of the nucleus accumbens shell in conditioned taste aversion learning.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2001, Sep-01, Volume: 21, Issue:17

    Topics: Animals; Avoidance Learning; Benzazepines; Cacao; Conditioning, Classical; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Administration Routes; Lithium Chloride; Male; Microinjections; Nucleus Accumbens; Raclopride; Rats; Receptors, Dopamine D1; Saccharin; Sucrose; Taste; Time Factors

2001
Selective D2 receptor actions on the functional circuitry of working memory.
    Science (New York, N.Y.), 2004, Feb-06, Volume: 303, Issue:5659

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Cues; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Electrophysiology; Macaca mulatta; Male; Memory; Neurons; Prefrontal Cortex; Psychomotor Performance; Quinpirole; Raclopride; Receptors, Dopamine D1; Receptors, Dopamine D2; Reward; Saccades; Salicylamides

2004
Differential role of dopamine in drug- and lithium-conditioned saccharin avoidance.
    Physiology & behavior, 2005, May-19, Volume: 85, Issue:1

    Topics: Analysis of Variance; Animals; Avoidance Learning; Benzazepines; Conditioning, Operant; Dopamine; Dopamine Antagonists; Drug Interactions; Eating; Lithium Chloride; Male; Nicotine; Nicotinic Agonists; Raclopride; Rats; Rats, Sprague-Dawley; Saccharin

2005
Differential involvement of dopamine D1 receptors in morphine- and lithium-conditioned saccharin avoidance.
    Physiology & behavior, 2009, Jan-08, Volume: 96, Issue:1

    Topics: Animals; Avoidance Learning; Benzazepines; Conditioning, Operant; Dopamine Antagonists; Food Preferences; Lithium Chloride; Male; Morphine; Narcotics; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Saccharin; Time Factors; Water Deprivation

2009
Attenuated dopaminergic tone in the paraventricular nucleus contributing to sympathoexcitation in rats with Type 2 diabetes.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2014, Jan-15, Volume: 306, Issue:2

    Topics: Animals; Benzazepines; Blood Glucose; Diabetes Mellitus, Type 2; Dopamine; Dopamine Antagonists; Gene Expression Regulation; Paraventricular Hypothalamic Nucleus; Raclopride; Rats; Receptors, Dopamine; Sympathetic Nervous System

2014
Blockade of dopamine D₁ receptors, but not D₂ receptors, decreases motivation in a novel effort-discounting paradigm in common marmosets.
    Behavioral neuroscience, 2018, Volume: 132, Issue:6

    Topics: Animals; Benzazepines; Callithrix; Decision Making; Dopamine Antagonists; Dose-Response Relationship, Drug; Female; Male; Motivation; Motor Activity; Physical Exertion; Psychological Tests; Psychotropic Drugs; Raclopride; Receptors, Dopamine D1; Receptors, Dopamine D2; Reward

2018
Altered Functional Connectivity of the Orbital Cortex and Striatum Associated with Catalepsy Induced by Dopamine D1 and D2 Antagonists.
    Biological & pharmaceutical bulletin, 2021, Volume: 44, Issue:3

    Topics: Animals; Benzazepines; Catalepsy; Corpus Striatum; Dopamine Antagonists; Mice, Inbred C57BL; Mice, Transgenic; Prefrontal Cortex; Raclopride; Receptors, Dopamine D1; Receptors, Dopamine D2

2021