ebselen and glutaminase

ebselen has been researched along with glutaminase in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's4 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Auld, DS; Boxer, MB; Ferraris, DV; Rojas, C; Shen, M; Simeonov, A; Slusher, BS; Tanega, C; Thomas, AG; Tsukamoto, T1
Chen, Z; Fang, J; Hou, W; Ruan, BH; Ruan, JJ; Su, W; Xie, J; Yang, G; Yu, Y; Zhang, J; Zhang, Z; Zhu, M1
Ji, X; Jin, Y; Li, D; Lu, S; Ruan, BH; Ruan, H; Yu, Y; Zhang, Y; Zhao, H; Zhou, J1
Behar, KL; Chowdhury, GMI; Kosten, L; Mingote, S; Rayport, S; Rothman, DL; Staelens, S1

Other Studies

4 other study(ies) available for ebselen and glutaminase

ArticleYear
Kinetic characterization of ebselen, chelerythrine and apomorphine as glutaminase inhibitors.
    Biochemical and biophysical research communications, 2013, Aug-23, Volume: 438, Issue:2

    Topics: AIDS Dementia Complex; Apomorphine; Azoles; Benzophenanthridines; Cell Proliferation; Dose-Response Relationship, Drug; Drug Design; Drug Evaluation, Preclinical; Glutaminase; Humans; Inhibitory Concentration 50; Isoindoles; Neoplasms; Organoselenium Compounds; RNA, Small Interfering; Sensitivity and Specificity

2013
Biomolecular Interaction Assays Identified Dual Inhibitors of Glutaminase and Glutamate Dehydrogenase That Disrupt Mitochondrial Function and Prevent Growth of Cancer Cells.
    Analytical chemistry, 2017, 02-07, Volume: 89, Issue:3

    Topics: Allosteric Site; Azoles; Cell Line, Tumor; Cell Proliferation; Chromatography, High Pressure Liquid; Enzyme Assays; Enzyme Inhibitors; Glutamate Dehydrogenase; Glutaminase; Humans; Isoindoles; Kinetics; Membrane Potential, Mitochondrial; Mitochondria; Organoselenium Compounds; Recombinant Proteins; Structure-Activity Relationship

2017
Ebselen: Mechanisms of Glutamate Dehydrogenase and Glutaminase Enzyme Inhibition.
    ACS chemical biology, 2017, 12-15, Volume: 12, Issue:12

    Topics: Amino Acid Sequence; Azoles; Cloning, Molecular; Escherichia coli; Glutamate Dehydrogenase; Glutaminase; Isoindoles; Models, Molecular; Organoselenium Compounds; Protein Conformation; Proteomics; Thioredoxin-Disulfide Reductase

2017
Glutaminase activity in GLS1 Het mouse brain compared to putative pharmacological inhibition by ebselen using ex vivo MRS.
    Neurochemistry international, 2019, Volume: 129

    Topics: Amino Acids; Animals; Azoles; Brain; Brain Chemistry; Female; gamma-Aminobutyric Acid; Glutaminase; Heterozygote; Hippocampus; Isoindoles; Male; Mice; Nerve Tissue Proteins; Nuclear Magnetic Resonance, Biomolecular; Organoselenium Compounds; Sequence Deletion

2019