Page last updated: 2024-09-03

e 5324 and pd 128042

e 5324 has been researched along with pd 128042 in 3 studies

Compound Research Comparison

Studies
(e 5324)
Trials
(e 5324)
Recent Studies (post-2010)
(e 5324)
Studies
(pd 128042)
Trials
(pd 128042)
Recent Studies (post-2010) (pd 128042)
70066014

Protein Interaction Comparison

ProteinTaxonomye 5324 (IC50)pd 128042 (IC50)
Sterol O-acyltransferase 1Rattus norvegicus (Norway rat)2.1277
Adenosine receptor A1Rattus norvegicus (Norway rat)0.14
Sterol O-acyltransferase 1Homo sapiens (human)1.7444
Sterol O-acyltransferase 1Mus musculus (house mouse)0.31
Acyl-CoA:cholesterol acyltransferase Oryctolagus cuniculus (rabbit)0.1487

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fujimori, T; Hayashi, K; Hiyoshi, H; Kimura, T; Kobayashi, H; Kogushi, M; Ohtsuka, I; Saeki, T; Tanaka, H; Yamada, T1
Hakamata, H; Horiuchi, S; Kawasaki, T; Matsuda, H; Miyazaki, A1
Azuma, Y; Kawasaki, T; Nobuhara, Y; Ohno, K; Seto, J; Yamada, T; Yamasaki, M1

Other Studies

3 other study(ies) available for e 5324 and pd 128042

ArticleYear
Effect of the acyl-CoA:cholesterol acyltransferase inhibitor, E5324, on experimental atherosclerosis in rabbits.
    Atherosclerosis, 1994, Volume: 107, Issue:2

    Topics: Anilides; Animals; Aorta, Thoracic; Arteriosclerosis; Cholestyramine Resin; Dose-Response Relationship, Drug; Lipid Metabolism; Liver; Male; Phenylurea Compounds; Probucol; Rabbits; Sterol O-Acyltransferase; Tunica Intima; Tunica Media

1994
Biochemical evidence for oligomerization of rat adrenal acyl-coenzyme A:cholesterol acyltransferase.
    Biochemical and biophysical research communications, 1998, Mar-17, Volume: 244, Issue:2

    Topics: Adrenal Glands; Anilides; Aniline Compounds; Animals; Cross-Linking Reagents; Cyclohexanes; Enzyme Inhibitors; Humans; Immunoblotting; Macromolecular Substances; Male; Microsomes; Microsomes, Liver; Molecular Weight; Phenylurea Compounds; Protein Conformation; Rats; Rats, Wistar; Sterol O-Acyltransferase; Tissue Distribution

1998
Effects of NTE-122, a novel acyl-CoA:cholesterol acyltransferase inhibitor, on cholesterol esterification and secretions of apolipoprotein B-containing lipoprotein and bile acids in HepG2.
    Japanese journal of pharmacology, 1999, Volume: 79, Issue:2

    Topics: Acetates; Anilides; Aniline Compounds; Apolipoproteins B; Bile Acids and Salts; Carcinoma, Hepatocellular; Cholesterol; Cyclohexanes; Drug Interactions; Enzyme Inhibitors; Humans; Hydroxycholesterols; Lipoproteins; Oleic Acid; Phenylurea Compounds; Phospholipids; Sterol O-Acyltransferase; Triglycerides; Tumor Cells, Cultured

1999