Page last updated: 2024-08-23

du-21220 and isoproterenol

du-21220 has been researched along with isoproterenol in 24 studies

Research

Studies (24)

TimeframeStudies, this research(%)All Research%
pre-199013 (54.17)18.7374
1990's8 (33.33)18.2507
2000's3 (12.50)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Akahane, M; Akahane, S; Hirabayashi, A; Miyata, H; Mukaiyama, H; Muranaka, H; Tamai, T; Tanaka, N1
Lombardo, F; Obach, RS; Waters, NJ1
Larsen, JJ1
Schulman, H1
Berg-Johnsen, P1
Brooks, J; Casper, RF; Dayes, BA; Freitag, CL; Lye, SJ1
Colbert, WE; Williams, GD; Williams, PD; Wilson, BF1
Colbert, WE; Williams, GD; Williams, PD1
Caritis, SN; Chiao, JP; Kridgen, P1
Brikas, P; Buéno, L; Fioramonti, J1
Casper, RF; Lye, SJ1
Aureggi, G; Bianchetti, A; Boigegrain, R; Cecchi, R; Croci, T; Manara, L; Tarantino, A1
Broadley, KJ; Grassby, PF1
Arch, JR; Broadley, KJ; Grassby, PF; Wilson, C1
Dubyak, GR; Moore, JJ; Moore, RM; Vander Kooy, D1
Ikeda, S; Tamaoki, H1
Izumi, H; Kishikawa, T1
Akahane, M; Ikeda, S; Nebashi, Y; Tamaoki, H1
Akahane, M; Ikeda, S; Nebashi, Y1
Cosentino, M; Costa, A; Crema, A; D'Angelo, L; De Ponti, F; Frigo, G; Gibelli, G; Girani, M1
De Ridder, WJ; Higashino, M; Kinoshita, H; Meulemans, AL; Schuurkes, JA; Tokuhara, T1
Collins, PL; Maguire, ME; Moore, JJ; Moore, RM; Roberts, JM; Zink, E1
Asano, M; Azuma, H; Hashimoto, S; Ito, Y; Kato, H; Morikawa, K; Ohashi, T1

Other Studies

24 other study(ies) available for du-21220 and isoproterenol

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Discovery of novel N-phenylglycine derivatives as potent and selective beta(3)-adrenoceptor agonists for the treatment of frequent urination and urinary incontinence.
    Journal of medicinal chemistry, 2001, Apr-26, Volume: 44, Issue:9

    Topics: Adrenergic beta-Agonists; Animals; Blood Pressure; Female; Ferrets; Glycine; Heart Rate; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Pregnancy; Pressure; Rats; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Structure-Activity Relationship; Urinary Bladder; Urinary Incontinence; Urination; Uterus

2001
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Beta-adrenoceptors in the pregnant and non-pregnant myometrium of the goat and cow.
    Acta pharmacologica et toxicologica, 1979, Volume: 44, Issue:2

    Topics: Albuterol; Animals; Butoxamine; Cattle; Dose-Response Relationship, Drug; Female; Goats; Isoproterenol; Myometrium; Practolol; Pregnancy; Pregnancy, Animal; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta; Ritodrine; Uterine Contraction; Uterus

1979
The comparative actions of uterine inhibiting drugs.
    American journal of obstetrics and gynecology, 1978, Mar-15, Volume: 130, Issue:6

    Topics: Animals; Depression, Chemical; Electric Stimulation; Female; Humans; Isoproterenol; Isoxsuprine; Myometrium; Norepinephrine; Pregnancy; Propanolamines; Propranolol; Rabbits; Ritodrine; Uterine Contraction

1978
Action of isoprenaline, isoxsuprine and ritodrine in the human non-pregnant myometrium.
    Acta pharmacologica et toxicologica, 1976, Volume: 39, Issue:2

    Topics: Drug Interactions; Female; Humans; In Vitro Techniques; Isoproterenol; Isoxsuprine; Myometrium; Propanolamines; Propranolol; Ritodrine; Uterine Contraction; Uterus

1976
Failure of ritodrine to prevent preterm labor in the sheep.
    American journal of obstetrics and gynecology, 1992, Volume: 167, Issue:5

    Topics: Animals; Cyclic AMP; Depression, Chemical; Down-Regulation; Female; Fetal Movement; Heart Rate; Heart Rate, Fetal; Isoproterenol; Myometrium; Obstetric Labor, Premature; Pregnancy; Prostaglandins; Receptors, Adrenergic, beta; Respiration; Ritodrine; Sheep; Uterine Contraction

1992
Relationship between in vitro relaxation of the costo-uterine smooth muscle and mesovarial leiomyoma formation in vivo by beta-receptor agonists.
    Archives of toxicology, 1991, Volume: 65, Issue:7

    Topics: Adrenergic beta-Agonists; Albuterol; Animals; Female; Guinea Pigs; Isoproterenol; Leiomyoma; Male; Myometrium; Norepinephrine; Rats; Rats, Inbred Strains; Ritodrine; Terbutaline; Uterine Contraction; Uterine Neoplasms

1991
Beta-adrenoceptor profile of ractopamine HCl in isolated smooth and cardiac muscle tissues of rat and guinea-pig.
    The Journal of pharmacy and pharmacology, 1991, Volume: 43, Issue:12

    Topics: Adrenergic beta-Agonists; Albuterol; Animals; Female; Guinea Pigs; Heart; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Phenethylamines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Ritodrine

1991
Comparison of pulsatile and continuous ritodrine administration: effects on uterine contractility and beta-adrenergic receptor cascade.
    American journal of obstetrics and gynecology, 1991, Volume: 164, Issue:4

    Topics: Adenylyl Cyclases; Animals; Enzyme Activation; Female; Isoproterenol; Myometrium; Osmolar Concentration; Oxytocin; Pulsatile Flow; Receptors, Adrenergic, beta; Ritodrine; Sheep; Uterine Contraction

1991
Central and peripheral beta-adrenergic influences on reticulo-rumen and upper-gut myoelectrical activity in sheep.
    Journal of veterinary pharmacology and therapeutics, 1989, Volume: 12, Issue:4

    Topics: Acebutolol; Animals; Dobutamine; Duodenum; Electromyography; Female; Gastrointestinal Motility; Intestine, Small; Isoproterenol; Jejunum; Propranolol; Receptors, Adrenergic, beta; Reticulum; Ritodrine; Rumen; Sheep

1989
Myometrial desensitization to continuous but not to intermittent beta-adrenergic agonist infusion in the sheep.
    American journal of obstetrics and gynecology, 1986, Volume: 154, Issue:2

    Topics: Adrenergic beta-Agonists; Animals; Electromyography; Female; Half-Life; Isoproterenol; Myometrium; Obstetric Labor, Premature; Pregnancy; Pressure; Ritodrine; Sheep; Time Factors; Uterine Contraction; Uterus

1986
Inhibition of rat colon motility by stimulation of atypical beta-adrenoceptors with new gut-specific agents.
    Pharmacological research communications, 1988, Volume: 20, Issue:2

    Topics: Adrenergic beta-Agonists; Albuterol; Animals; Colon; Ethanolamines; Gastrointestinal Motility; In Vitro Techniques; Isoproterenol; Male; Rats; Rats, Inbred Strains; Ritodrine

1988
Responses mediated via beta-1 adrenoceptors but not beta-2 adrenoceptors exhibit supersensitivity after chronic reserpine pretreatment.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:3

    Topics: Animals; Blood Vessels; Carbachol; Dose-Response Relationship, Drug; Female; Guinea Pigs; Heart Rate; Ileum; In Vitro Techniques; Isoproterenol; Lung; Male; Myocardial Contraction; Norepinephrine; Practolol; Prenalterol; Receptors, Adrenergic, beta; Reserpine; Ritodrine; Trachea; Vas Deferens; Vasoconstriction

1986
Beta-adrenoceptor sensitivity of brown and white adipocytes after chronic pretreatment of rats with reserpine.
    Biochemical pharmacology, 1987, Jan-01, Volume: 36, Issue:1

    Topics: Adipose Tissue; Adipose Tissue, Brown; Animals; Body Weight; Dose-Response Relationship, Drug; Heart Atria; Isoproterenol; Lipolysis; Male; Oxyfedrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Reserpine; Ritodrine; Vas Deferens

1987
Oxytocin activates the inositol-phospholipid-protein kinase-C system and stimulates prostaglandin production in human amnion cells.
    Endocrinology, 1988, Volume: 123, Issue:4

    Topics: Amnion; Calcium; Cells, Cultured; Colforsin; Dinoprostone; Egtazic Acid; Epithelium; Humans; Inositol Phosphates; Isoproterenol; Oxytocin; Prostaglandins E; Protein Kinase C; Reference Values; Ritodrine; Sugar Phosphates; Tetradecanoylphorbol Acetate; Type C Phospholipases

1988
Pharmacological investigation of ritodrine hydrochloride, a beta 2-adrenoceptor stimulant.
    Japanese journal of pharmacology, 1984, Volume: 36, Issue:4

    Topics: Adrenergic beta-Agonists; Animals; Calcium; Carbachol; Cyclic AMP; Female; Guinea Pigs; Heart Rate; In Vitro Techniques; Isoproterenol; Isoxsuprine; Myocardium; Pregnancy; Propanolamines; Rats; Rats, Inbred Strains; Ritodrine; Uterine Contraction; Uterus; Verapamil

1984
Effects of ritodrine, a beta 2-adrenoceptor agonist, on smooth muscle cells of the myometrium of pregnant rats.
    British journal of pharmacology, 1982, Volume: 76, Issue:3

    Topics: Animals; Calcium; Cyclic AMP; Female; Isoproterenol; Membrane Potentials; Myometrium; Pregnancy; Pregnancy, Animal; Propanolamines; Rats; Rats, Inbred Strains; Ritodrine; Uterine Contraction; Uterus

1982
Effects of ritodrine hydrochloride, a beta 2-adrenoceptor stimulant, on uterine motilities in late pregnancy.
    Japanese journal of pharmacology, 1984, Volume: 35, Issue:3

    Topics: Anesthesia; Animals; Blood Pressure; Female; Heart Rate; Isoproterenol; Isoxsuprine; Oxytocin; Pregnancy; Propanolamines; Rabbits; Rats; Rats, Inbred Strains; Ritodrine; Species Specificity; Uterine Contraction

1984
[Effects of a beta 2-stimulant, ritodrine hydrochloride, on the fetuses and dams in the late stage of pregnancy: an experimental study using rabbits].
    Nihon Sanka Fujinka Gakkai zasshi, 1983, Volume: 35, Issue:11

    Topics: Animals; Blood Pressure; Female; Fetal Heart; Fetus; Heart Rate; Isoproterenol; Isoxsuprine; Placenta; Pregnancy; Pregnancy, Animal; Propanolamines; Prostaglandins F; Rabbits; Regional Blood Flow; Ritodrine; Uterine Contraction

1983
Inhibitory effects of SR 58611A on canine colonic motility: evidence for a role of beta 3-adrenoceptors.
    British journal of pharmacology, 1995, Volume: 114, Issue:7

    Topics: Adrenergic beta-Agonists; Alprenolol; Animals; Atropine; Colon; Dogs; Dose-Response Relationship, Drug; Female; Gastrointestinal Motility; Heart Rate; Isoproterenol; Receptors, Adrenergic, beta; Ritodrine; Tetrahydronaphthalenes

1995
Effect of adrenoceptor agonists on striated muscle strips of the canine oesophagus.
    British journal of pharmacology, 1993, Volume: 110, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dogs; Esophagus; Female; In Vitro Techniques; Isometric Contraction; Isoproterenol; Male; Muscle, Smooth; Norepinephrine; Phenylephrine; Prazosin; Propanolamines; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Ritodrine

1993
Ritodrine: a beta-adrenergic receptor antagonist in human amnion.
    American journal of obstetrics and gynecology, 1993, Volume: 168, Issue:1 Pt 1

    Topics: Amnion; Binding, Competitive; Cyclic AMP; Dinoprostone; Epinephrine; Humans; Isoproterenol; Norepinephrine; Pindolol; Receptors, Adrenergic, beta; Ritodrine

1993
Potent inhibition of spontaneous rhythmic contraction by a novel beta 2-adrenoceptor agonist, HSR-81, in pregnant rat uterus.
    European journal of pharmacology, 1996, Jul-04, Volume: 307, Issue:3

    Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atenolol; Benzyl Alcohols; Binding, Competitive; Colforsin; Diestrus; Female; Gestational Age; In Vitro Techniques; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Isotope Labeling; Kinetics; Pindolol; Pregnancy; Propanolamines; Protein Binding; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, beta-2; Ritodrine; Uterine Contraction

1996