Page last updated: 2024-09-04

ds 4574 and histamine

ds 4574 has been researched along with histamine in 4 studies

Compound Research Comparison

Studies
(ds 4574)
Trials
(ds 4574)
Recent Studies (post-2010)
(ds 4574)
Studies
(histamine)
Trials
(histamine)
Recent Studies (post-2010) (histamine)
132037,7181,3723,457

Protein Interaction Comparison

ProteinTaxonomyds 4574 (IC50)histamine (IC50)
Histamine H1 receptorRattus norvegicus (Norway rat)0.1585
Histamine H1 receptorHomo sapiens (human)0.1585

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Aibara, S; Iwamoto, T; Mori, M; Tsubokawa, M; Tsukada, W1
Furuhama, K; Kawarabayashi, K; Tabuchi, Y1
Furuhama, K; Tabuchi, Y1
Kokue, E; Tabuchi, Y; Yamashika, Y1

Other Studies

4 other study(ies) available for ds 4574 and histamine

ArticleYear
Antiallergic activity of 6-(2-cyclohexylethyl)-[1,3,4]thiadiazolo- [3,2-a]-1,2,3-triazolo-[4,5-d]pyrimidin-9(3H)-one (DS-4574) in rats.
    International archives of allergy and immunology, 1992, Volume: 98, Issue:2

    Topics: Adrenalectomy; Anaphylaxis; Animals; Capillary Permeability; Histamine; Histamine Release; Hypersensitivity; Leukotriene Antagonists; Lung; Male; Passive Cutaneous Anaphylaxis; Peritoneal Cavity; Pyrimidines; Rats; Rats, Inbred Strains; Serotonin; Time Factors; Triazoles

1992
Inhibitory effect of DS-4574, a peptidoleukotriene antagonist with mast cell stabilizing action, on compound 48/80-induced gastric mucosal lesions in rats.
    Agents and actions, 1994, Volume: 41, Issue:1-2

    Topics: Acetophenones; Administration, Oral; Animals; Cimetidine; Cromolyn Sodium; Gastric Mucosa; Histamine; Histamine Release; Injections, Intraperitoneal; Injections, Subcutaneous; Leukotriene Antagonists; Male; Mast Cells; p-Methoxy-N-methylphenethylamine; Pyrimidines; Rats; Rats, Sprague-Dawley; Tetrazoles; Triazoles

1994
Inhibitory effect of DS-4574, a mast cell stabilizer with peptidoleukotriene receptor antagonism, on gastric acid secretion in rats.
    European journal of pharmacology, 1994, Apr-01, Volume: 255, Issue:1-3

    Topics: Animals; Bucladesine; Carbachol; Fistula; Gastric Acid; H(+)-K(+)-Exchanging ATPase; Histamine; Leukotriene Antagonists; Male; Mast Cells; Pentagastrin; Pyrimidines; Rats; Rats, Sprague-Dawley; Stomach; Triazoles

1994
Antisecretory effect of DS-4574, a mast cell stabilizer with peptidoleukotriene antagonism, on gastric acid secretion in the pig.
    Agents and actions, 1994, Volume: 41, Issue:1-2

    Topics: Adenosine Triphosphatases; Animals; Carbachol; Cation Transport Proteins; Female; Gastric Acid; Gastric Mucosa; Histamine; In Vitro Techniques; Injections, Intramuscular; Leukotriene Antagonists; Male; Pyrimidines; Swine; Swine, Miniature; Tetragastrin; Triazoles

1994