Page last updated: 2024-09-04

ds 4574 and cimetidine

ds 4574 has been researched along with cimetidine in 2 studies

Compound Research Comparison

Studies
(ds 4574)
Trials
(ds 4574)
Recent Studies (post-2010)
(ds 4574)
Studies
(cimetidine)
Trials
(cimetidine)
Recent Studies (post-2010) (cimetidine)
13209,4731,687377

Protein Interaction Comparison

ProteinTaxonomyds 4574 (IC50)cimetidine (IC50)
Solute carrier family 22 member 1Mus musculus (house mouse)0.59
Solute carrier family 22 member 2Mus musculus (house mouse)8
Potassium-transporting ATPase alpha chain 1Homo sapiens (human)0.82
Histamine H2 receptorHomo sapiens (human)1.1742
Histamine H2 receptorCavia porcellus (domestic guinea pig)1.02
Potassium-transporting ATPase subunit betaHomo sapiens (human)0.82
Multidrug and toxin extrusion protein 1Homo sapiens (human)3.0333

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kurebayashi, Y; Tabuchi, Y1
Furuhama, K; Kawarabayashi, K; Tabuchi, Y1

Other Studies

2 other study(ies) available for ds 4574 and cimetidine

ArticleYear
Effect of DS-4574, a novel peptidoleukotriene antagonist with mast cell stabilizing action, on acute gastric lesions and gastric secretion in rats.
    Japanese journal of pharmacology, 1992, Volume: 60, Issue:4

    Topics: Animals; Anti-Ulcer Agents; Aspirin; Cimetidine; Dose-Response Relationship, Drug; Ethanol; Gastric Acid; Gastric Mucosa; Hydrochloric Acid; Immersion; Leukotriene Antagonists; Male; Mast Cells; Pylorus; Pyrimidines; Rats; Rats, Sprague-Dawley; Restraint, Physical; Stomach Ulcer; Triazoles

1992
Inhibitory effect of DS-4574, a peptidoleukotriene antagonist with mast cell stabilizing action, on compound 48/80-induced gastric mucosal lesions in rats.
    Agents and actions, 1994, Volume: 41, Issue:1-2

    Topics: Acetophenones; Administration, Oral; Animals; Cimetidine; Cromolyn Sodium; Gastric Mucosa; Histamine; Histamine Release; Injections, Intraperitoneal; Injections, Subcutaneous; Leukotriene Antagonists; Male; Mast Cells; p-Methoxy-N-methylphenethylamine; Pyrimidines; Rats; Rats, Sprague-Dawley; Tetrazoles; Triazoles

1994