draflazine has been researched along with thioinosine in 12 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 6 (50.00) | 18.2507 |
| 2000's | 6 (50.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| IJzerman, AP; Janssen, C; Kruidering, M; van Belle, H; van Weert, A | 1 |
| Van Belle, H; Ver Donck, K; Wynants, J | 1 |
| Böhm, D; Böhm, M; Erdmann, E; Müller-Ehmsen, J; Reichart, B; Reichenspurner, H; Schwinger, RH; Weinhold, C | 1 |
| Beukers, MW; IJzerman, AP; Kerkhof, CJ; Soudijn, W | 1 |
| Hammond, JR; Jones, KW | 1 |
| Deussen, A; Kelm, M; Schäfer, S; Stappert, M | 1 |
| Hammond, JR | 1 |
| Baldwin, SA; Cass, CE; Hyde, RJ; McConkey, GA; McRobert, L; Parker, MD; Yao, SY; Young, JD | 1 |
| Archer, RG; Hammond, JR; McConnell, K; Stolk, M | 1 |
| Archer, RG; Hammond, JR; Pitelka, V | 1 |
| Bone, DB; Hammond, JR | 1 |
| Baldwin, SA; Cass, CE; Damaraju, V; Paproski, RJ; Tackaberry, T; Visser, F; Young, JD; Zhang, J | 1 |
12 other study(ies) available for draflazine and thioinosine
| Article | Year |
|---|---|
[3H]R75231--a new radioligand for the nitrobenzylthioinosine sensitive nucleoside transport proteins. Characterization of (+/-)-[3H]R75231 binding to calf lung membranes, stereospecificity of its two stereoisomers, and comparison with [3H]nitrobenzylthioi
Topics: Affinity Labels; Animals; Cattle; In Vitro Techniques; Lung; Membranes; Piperazines; Radioligand Assay; Stereoisomerism; Thioinosine; Tritium | 1992 |
Comparison of the existing nucleoside transport inhibitors: in vitro and in vivo data.
Topics: Animals; Biological Transport; Dilazep; Dipyridamole; Epinephrine; Erythrocytes; Humans; In Vitro Techniques; Nucleosides; Phosphates; Piperazines; Rabbits; Thioinosine | 1991 |
Studies of the nucleoside transporter inhibitor, draflazine, in the human myocardium.
Topics: Adult; Affinity Labels; Aged; Carbachol; Cardiac Pacing, Artificial; Carrier Proteins; Dipyridamole; Erythrocyte Membrane; Female; Heart; Humans; In Vitro Techniques; Male; Membrane Proteins; Middle Aged; Myocardial Contraction; Myocardium; Nucleoside Transport Proteins; Phenylisopropyladenosine; Piperazines; Radioligand Assay; Thioinosine | 1994 |
Nucleoside transport inhibition and platelet aggregation in human blood: R75231 and its enantiomers, draflazine and R88016.
Topics: Adenosine; Adenosine Diphosphate; Binding Sites; Biological Transport; Blood Platelets; Erythrocytes; Humans; Piperazines; Platelet Aggregation; Platelet Aggregation Inhibitors; Radioligand Assay; Stereoisomerism; Thioinosine | 1994 |
Interaction of the mioflazine derivative R75231 with the nucleoside transporter: evidence for positive cooperativity.
Topics: Adenosine; Animals; Binding, Competitive; Carrier Proteins; Cerebral Cortex; Erythrocyte Membrane; Half-Life; Humans; In Vitro Techniques; Kinetics; Membrane Proteins; Nucleoside Transport Proteins; Piperazines; Rabbits; Synaptosomes; Thioinosine; Uridine | 1993 |
Quantification of extracellular and intracellular adenosine production: understanding the transmembranous concentration gradient.
Topics: Adenine; Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Animals; Biological Transport; Bradykinin; Coronary Circulation; Cytosol; Depression, Chemical; Dipyridamole; Drug Synergism; Enzyme Inhibitors; Extracellular Space; Guinea Pigs; Heart; Models, Biological; Myocardium; Osmolar Concentration; Oxygen; Oxygen Consumption; Piperazines; Thioinosine; Tubercidin | 1999 |
Interaction of a series of draflazine analogues with equilibrative nucleoside transporters: species differences and transporter subtype selectivity.
Topics: Animals; Carcinoma, Ehrlich Tumor; Carrier Proteins; Cell Membrane; Equilibrative Nucleoside Transporter 1; Equilibrative-Nucleoside Transporter 2; Erythrocytes; Humans; In Vitro Techniques; Membrane Proteins; Mice; Piperazines; Radioligand Assay; Species Specificity; Thioinosine; Tumor Cells, Cultured; Uridine | 2000 |
Identification of a nucleoside/nucleobase transporter from Plasmodium falciparum, a novel target for anti-malarial chemotherapy.
Topics: Adenine; Amino Acid Sequence; Animals; Antimalarials; Biological Transport; Blotting, Southern; Carrier Proteins; Cations; Cell Membrane; Cloning, Molecular; Dilazep; Dipyridamole; Dose-Response Relationship, Drug; Hydrogen-Ion Concentration; Kinetics; Molecular Sequence Data; Nucleobase, Nucleoside, Nucleotide, and Nucleic Acid Transport Proteins; Nucleosides; Phylogeny; Piperazines; Plasmodium falciparum; Platelet Aggregation Inhibitors; Protein Structure, Secondary; Protozoan Proteins; Sequence Homology, Amino Acid; Substrate Specificity; Thioinosine; Time Factors; Uridine; Vasodilator Agents; Xenopus | 2000 |
Pharmacological analysis and molecular cloning of the canine equilibrative nucleoside transporter 1.
Topics: Amino Acid Sequence; Animals; Binding, Competitive; Carrier Proteins; Cell Line; Cloning, Molecular; Dilazep; Dipyridamole; DNA, Complementary; Dogs; Dose-Response Relationship, Drug; Equilibrative Nucleoside Transporter 1; Formycins; Kinetics; Molecular Sequence Data; Piperazines; Protein Binding; Protein Conformation; Radioligand Assay; Sequence Alignment; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Structure-Activity Relationship; Thioinosine; Tritium | 2004 |
Nucleoside transporter subtype expression and function in rat skeletal muscle microvascular endothelial cells.
Topics: Animals; Capillaries; Cell Separation; Cells, Cultured; Dilazep; Dipyridamole; DNA Primers; Endothelial Cells; Formycins; Muscle, Skeletal; Nucleoside Transport Proteins; Piperazines; Radioligand Assay; Rats; Reverse Transcriptase Polymerase Chain Reaction; Thioinosine; Vasodilator Agents | 2004 |
Nucleoside and nucleobase transporters of primary human cardiac microvascular endothelial cells: characterization of a novel nucleobase transporter.
Topics: 2-Chloroadenosine; Animals; Cell Culture Techniques; Cell Line; Cells, Cultured; Child, Preschool; Coronary Vessels; Dilazep; Dipyridamole; Dogs; Endothelial Cells; Equilibrative Nucleoside Transporter 1; Equilibrative-Nucleoside Transporter 2; Female; Humans; Hypoxanthine; Kinetics; Microcirculation; Nucleobase Transport Proteins; Piperazines; Protein Binding; Purines; Rats; Swine; Thioinosine; Transfection; Tritium | 2007 |
Mutation of Trp29 of human equilibrative nucleoside transporter 1 alters affinity for coronary vasodilator drugs and nucleoside selectivity.
Topics: Adenosine; Biological Transport; Dilazep; Dipyridamole; Enzyme Activation; Equilibrative Nucleoside Transporter 1; Humans; Kinetics; Models, Biological; Mutation; Nucleosides; Piperazines; Protein Binding; Thioinosine; Tryptophan; Vasodilator Agents | 2008 |