Page last updated: 2024-08-24

draflazine and dipyridamole

draflazine has been researched along with dipyridamole in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (33.33)18.2507
2000's6 (50.00)29.6817
2010's1 (8.33)24.3611
2020's1 (8.33)2.80

Authors

AuthorsStudies
Heitman, LH; IJzerman, AP; Vlachodimou, A1
Van Belle, H; Ver Donck, K; Wynants, J1
Van Belle, H; Ver Donck, KL; Verheyen, WJ1
Böhm, D; Böhm, M; Erdmann, E; Müller-Ehmsen, J; Reichart, B; Reichenspurner, H; Schwinger, RH; Weinhold, C1
Deussen, A; Kelm, M; Schäfer, S; Stappert, M1
Baldwin, SA; Cass, CE; Hyde, RJ; McConkey, GA; McRobert, L; Parker, MD; Yao, SY; Young, JD1
Karasawa, A; Katagiri, C; Kusaka, H; Mizutani, M; Nan-ya, K; Nishikawa, S; Noji, T; Sano, J1
Archer, RG; Hammond, JR; McConnell, K; Stolk, M1
Archer, RG; Hammond, JR; Pitelka, V1
Bone, DB; Hammond, JR1
Baldwin, SA; Cass, CE; Damaraju, V; Paproski, RJ; Tackaberry, T; Visser, F; Young, JD; Zhang, J1
Heitman, LH; IJzerman, AP; Konstantinopoulou, K; Vlachodimou, A1

Other Studies

12 other study(ies) available for draflazine and dipyridamole

ArticleYear
Label-free detection of transporter activity via GPCR signalling in living cells: A case for SLC29A1, the equilibrative nucleoside transporter 1.
    Scientific reports, 2019, 09-24, Volume: 9, Issue:1

    Topics: Cell Line, Tumor; Equilibrative Nucleoside Transporter 1; Humans; Ligands; Membrane Transport Proteins; Osteosarcoma; Receptors, G-Protein-Coupled; Receptors, Purinergic P1; Signal Transduction

2019
Comparison of the existing nucleoside transport inhibitors: in vitro and in vivo data.
    Advances in experimental medicine and biology, 1991, Volume: 309A

    Topics: Animals; Biological Transport; Dilazep; Dipyridamole; Epinephrine; Erythrocytes; Humans; In Vitro Techniques; Nucleosides; Phosphates; Piperazines; Rabbits; Thioinosine

1991
Nucleoside transport inhibition and fMLP-stimulated whole blood luminescence.
    Journal of molecular and cellular cardiology, 1991, Volume: 23, Issue:7

    Topics: Adenosine; Biological Transport; Dilazep; Dipyridamole; Humans; Luminescent Measurements; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Piperazines; Respiratory Burst

1991
Studies of the nucleoside transporter inhibitor, draflazine, in the human myocardium.
    British journal of pharmacology, 1994, Volume: 112, Issue:1

    Topics: Adult; Affinity Labels; Aged; Carbachol; Cardiac Pacing, Artificial; Carrier Proteins; Dipyridamole; Erythrocyte Membrane; Female; Heart; Humans; In Vitro Techniques; Male; Membrane Proteins; Middle Aged; Myocardial Contraction; Myocardium; Nucleoside Transport Proteins; Phenylisopropyladenosine; Piperazines; Radioligand Assay; Thioinosine

1994
Quantification of extracellular and intracellular adenosine production: understanding the transmembranous concentration gradient.
    Circulation, 1999, Apr-20, Volume: 99, Issue:15

    Topics: Adenine; Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Animals; Biological Transport; Bradykinin; Coronary Circulation; Cytosol; Depression, Chemical; Dipyridamole; Drug Synergism; Enzyme Inhibitors; Extracellular Space; Guinea Pigs; Heart; Models, Biological; Myocardium; Osmolar Concentration; Oxygen; Oxygen Consumption; Piperazines; Thioinosine; Tubercidin

1999
Identification of a nucleoside/nucleobase transporter from Plasmodium falciparum, a novel target for anti-malarial chemotherapy.
    The Biochemical journal, 2000, Jul-01, Volume: 349, Issue:Pt 1

    Topics: Adenine; Amino Acid Sequence; Animals; Antimalarials; Biological Transport; Blotting, Southern; Carrier Proteins; Cations; Cell Membrane; Cloning, Molecular; Dilazep; Dipyridamole; Dose-Response Relationship, Drug; Hydrogen-Ion Concentration; Kinetics; Molecular Sequence Data; Nucleobase, Nucleoside, Nucleotide, and Nucleic Acid Transport Proteins; Nucleosides; Phylogeny; Piperazines; Plasmodium falciparum; Platelet Aggregation Inhibitors; Protein Structure, Secondary; Protozoan Proteins; Sequence Homology, Amino Acid; Substrate Specificity; Thioinosine; Time Factors; Uridine; Vasodilator Agents; Xenopus

2000
Adenosine uptake inhibition ameliorates cerulein-induced acute pancreatitis in mice.
    Pancreas, 2002, Volume: 25, Issue:4

    Topics: Acute Disease; Adenosine; Amylases; Animals; Biological Transport; Ceruletide; Dipyridamole; Female; Lipase; Mice; Mice, Inbred BALB C; Models, Chemical; Pancreatitis; Piperazines; Pyrimidinones; Quinazolines; Theophylline

2002
Pharmacological analysis and molecular cloning of the canine equilibrative nucleoside transporter 1.
    European journal of pharmacology, 2004, Apr-26, Volume: 491, Issue:1

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; Carrier Proteins; Cell Line; Cloning, Molecular; Dilazep; Dipyridamole; DNA, Complementary; Dogs; Dose-Response Relationship, Drug; Equilibrative Nucleoside Transporter 1; Formycins; Kinetics; Molecular Sequence Data; Piperazines; Protein Binding; Protein Conformation; Radioligand Assay; Sequence Alignment; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Structure-Activity Relationship; Thioinosine; Tritium

2004
Nucleoside transporter subtype expression and function in rat skeletal muscle microvascular endothelial cells.
    British journal of pharmacology, 2004, Volume: 143, Issue:1

    Topics: Animals; Capillaries; Cell Separation; Cells, Cultured; Dilazep; Dipyridamole; DNA Primers; Endothelial Cells; Formycins; Muscle, Skeletal; Nucleoside Transport Proteins; Piperazines; Radioligand Assay; Rats; Reverse Transcriptase Polymerase Chain Reaction; Thioinosine; Vasodilator Agents

2004
Nucleoside and nucleobase transporters of primary human cardiac microvascular endothelial cells: characterization of a novel nucleobase transporter.
    American journal of physiology. Heart and circulatory physiology, 2007, Volume: 293, Issue:6

    Topics: 2-Chloroadenosine; Animals; Cell Culture Techniques; Cell Line; Cells, Cultured; Child, Preschool; Coronary Vessels; Dilazep; Dipyridamole; Dogs; Endothelial Cells; Equilibrative Nucleoside Transporter 1; Equilibrative-Nucleoside Transporter 2; Female; Humans; Hypoxanthine; Kinetics; Microcirculation; Nucleobase Transport Proteins; Piperazines; Protein Binding; Purines; Rats; Swine; Thioinosine; Transfection; Tritium

2007
Mutation of Trp29 of human equilibrative nucleoside transporter 1 alters affinity for coronary vasodilator drugs and nucleoside selectivity.
    The Biochemical journal, 2008, Sep-01, Volume: 414, Issue:2

    Topics: Adenosine; Biological Transport; Dilazep; Dipyridamole; Enzyme Activation; Equilibrative Nucleoside Transporter 1; Humans; Kinetics; Models, Biological; Mutation; Nucleosides; Piperazines; Protein Binding; Thioinosine; Tryptophan; Vasodilator Agents

2008
Affinity, binding kinetics and functional characterization of draflazine analogues for human equilibrative nucleoside transporter 1 (SLC29A1).
    Biochemical pharmacology, 2020, Volume: 172

    Topics: Cardiotonic Agents; Cell Line, Tumor; Dilazep; Dipyridamole; Equilibrative Nucleoside Transporter 1; Humans; Molecular Structure; Piperazines; Protein Binding; Radioligand Assay; Structure-Activity Relationship

2020