donepezil and rolipram

donepezil has been researched along with rolipram in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's8 (80.00)24.3611
2020's2 (20.00)2.80

Authors

AuthorsStudies
Huang, L; Li, W; Li, X; Wang, B; Wang, Y; Wang, Z1
An, B; Hu, J; Huang, L; Li, X; Li, Z; Pan, T1
Chen, Z; Gao, Y; Guo, L; He, X; Huang, L; Huang, YY; Li, Z; Liang, J; Liang, SH; Luo, HB; Wu, D; Wu, R; Yu, S; Zhou, Q1
Feng, KW; Liu, J; Liu, L; Wang, HT; Xu, JP; Zheng, L; Zhou, ZZ1
Wenger, GR; Whitney, KN1
Akkerman, S; Blokland, A; Prickaerts, J1
Akkerman, S; Blokland, A; Creemers, P; De Vry, J; Prickaerts, J; Sambeth, A; Uz, T; van Duinen, M; Vanmierlo, T1
Kumar, A; Singh, N1
Allouche, A; Almari, B; Fischer, N; Grayson, B; Harte, MK; Jackson, J; Koziel, V; McLean, SL; Neill, JC; Pillot, T; Watremez, W1
Graf, R; Hughes, ZA; Longo, JL1

Other Studies

10 other study(ies) available for donepezil and rolipram

ArticleYear
Design, Synthesis, and Evaluation of Orally Available Clioquinol-Moracin M Hybrids as Multitarget-Directed Ligands for Cognitive Improvement in a Rat Model of Neurodegeneration in Alzheimer's Disease.
    Journal of medicinal chemistry, 2015, Nov-12, Volume: 58, Issue:21

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Animals; Antioxidants; Benzofurans; Clioquinol; Cognition; Cyclic Nucleotide Phosphodiesterases, Type 4; Inflammation; Ligands; Male; Memory; Models, Molecular; Neurons; Neuroprotective Agents; Phosphodiesterase 4 Inhibitors; Protein Aggregates; Rats; Rats, Wistar; Resorcinols

2015
Synthesis and evaluation of clioquinol-rolipram/roflumilast hybrids as multitarget-directed ligands for the treatment of Alzheimer's disease.
    European journal of medicinal chemistry, 2019, Feb-01, Volume: 163

    Topics: Alzheimer Disease; Aminopyridines; Animals; Benzamides; Clioquinol; Cyclic Nucleotide Phosphodiesterases, Type 4; Cyclopropanes; Drug Design; Humans; Ligands; Mice; Rats; Rolipram

2019
Discovery and Optimization of α-Mangostin Derivatives as Novel PDE4 Inhibitors for the Treatment of Vascular Dementia.
    Journal of medicinal chemistry, 2020, 03-26, Volume: 63, Issue:6

    Topics: Aminopyridines; Animals; Benzamides; Cyclic Nucleotide Phosphodiesterases, Type 4; Cyclopropanes; Dementia, Vascular; Dogs; Drug Design; Humans; Male; Mice, Inbred C57BL; Molecular Structure; Phosphodiesterase 4 Inhibitors; Protein Binding; Rolipram; Structure-Activity Relationship; Vomiting; Xanthones

2020
Discovery of novel 2,3-dihydro-1H-inden-1-ones as dual PDE4/AChE inhibitors with more potency against neuroinflammation for the treatment of Alzheimer's disease.
    European journal of medicinal chemistry, 2022, Aug-05, Volume: 238

    Topics: Acetylcholinesterase; Alzheimer Disease; Animals; Cholinesterase Inhibitors; Donepezil; Drug Design; Indenes; Mice; Neuroinflammatory Diseases; Phosphodiesterase 4 Inhibitors; Structure-Activity Relationship

2022
Working memory in the aged Ts65Dn mouse, a model for Down syndrome.
    Behavioural brain research, 2012, Jun-15, Volume: 232, Issue:1

    Topics: Aging; Animals; Antidepressive Agents; Central Nervous System Stimulants; Cognition; Conditioning, Operant; Dextroamphetamine; Donepezil; Dose-Response Relationship, Drug; Down Syndrome; Indans; Longitudinal Studies; Male; Memantine; Memory, Short-Term; Mice; Mice, Neurologic Mutants; Nootropic Agents; Piperidines; Psychomotor Performance; Rolipram

2012
Possible overlapping time frames of acquisition and consolidation phases in object memory processes: a pharmacological approach.
    Learning & memory (Cold Spring Harbor, N.Y.), 2016, Volume: 23, Issue:1

    Topics: Animals; Cholinesterase Inhibitors; Discrimination, Psychological; Donepezil; Indans; Learning; Male; Memory; Phosphodiesterase 5 Inhibitors; Piperidines; Rats; Rats, Wistar; Recognition, Psychology; Rolipram; Scopolamine; Vardenafil Dihydrochloride

2016
The PDE4 inhibitor roflumilast improves memory in rodents at non-emetic doses.
    Behavioural brain research, 2016, Apr-15, Volume: 303

    Topics: Aminopyridines; Animals; Benzamides; Cyclopropanes; Donepezil; Indans; Male; Memory; Mice; Mice, Inbred C57BL; Nootropic Agents; Phosphodiesterase 4 Inhibitors; Piperidines; Rats, Wistar; Recognition, Psychology; Rolipram; Scopolamine; Spatial Memory; Vomiting

2016
Inhibitor of Phosphodiestearse-4 improves memory deficits, oxidative stress, neuroinflammation and neuropathological alterations in mouse models of dementia of Alzheimer's Type.
    Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie, 2017, Volume: 88

    Topics: Acetylcholinesterase; Aging; Alzheimer Disease; Animals; Antioxidants; Brain; Cholinesterase Inhibitors; Donepezil; Female; Indans; Inflammation; Learning; Male; Maze Learning; Memory Disorders; Mice; Neutrophil Infiltration; Oxidative Stress; Phosphodiesterase 4 Inhibitors; Piperidines; Plaque, Amyloid; Rolipram; Streptozocin

2017
Stabilized Low-n Amyloid-β Oligomers Induce Robust Novel Object Recognition Deficits Associated with Inflammatory, Synaptic, and GABAergic Dysfunction in the Rat.
    Journal of Alzheimer's disease : JAD, 2018, Volume: 62, Issue:1

    Topics: Amyloid beta-Peptides; Animals; Brain; Cognition; Disease Models, Animal; Donepezil; Female; gamma-Aminobutyric Acid; Inflammation; Male; Memory Disorders; Neurons; Nootropic Agents; Peptide Fragments; Random Allocation; Rats; Recognition, Psychology; Risperidone; Rolipram; Synapses

2018
The location discrimination reversal task in mice is sensitive to deficits in performance caused by aging, pharmacological and other challenges.
    Journal of psychopharmacology (Oxford, England), 2018, Volume: 32, Issue:9

    Topics: Aging; Animals; Conditioning, Operant; Discrimination, Psychological; Dizocilpine Maleate; Donepezil; Inflammation; Lipopolysaccharides; Male; Mice; Rolipram; Scopolamine; Space Perception

2018