Page last updated: 2024-09-02

dodecyl-beta-d-maltoside and tariquidar

dodecyl-beta-d-maltoside has been researched along with tariquidar in 2 studies

Compound Research Comparison

Studies
(dodecyl-beta-d-maltoside)
Trials
(dodecyl-beta-d-maltoside)
Recent Studies (post-2010)
(dodecyl-beta-d-maltoside)
Studies
(tariquidar)
Trials
(tariquidar)
Recent Studies (post-2010) (tariquidar)
319010421016138

Protein Interaction Comparison

ProteinTaxonomydodecyl-beta-d-maltoside (IC50)tariquidar (IC50)
ATP-dependent translocase ABCB1Mus musculus (house mouse)0.0643
ATP-dependent translocase ABCB1Homo sapiens (human)1.0841
Cytochrome P450 2C9 Homo sapiens (human)7.1
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)1.2363

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Abel, B; Ambudkar, SV; Chufan, EE; Shukla, S1
Clarke, DM; Loo, TW1

Other Studies

2 other study(ies) available for dodecyl-beta-d-maltoside and tariquidar

ArticleYear
Effects of a detergent micelle environment on P-glycoprotein (ABCB1)-ligand interactions.
    The Journal of biological chemistry, 2017, 04-28, Volume: 292, Issue:17

    Topics: Acridines; Adenosine Triphosphate; Animals; ATP Binding Cassette Transporter, Subfamily B; Baculoviridae; Binding Sites; Detergents; Dibenzocycloheptenes; Drug Delivery Systems; Drug Evaluation, Preclinical; Glucosides; Humans; Hydrolysis; Inhibitory Concentration 50; Insecta; Ligands; Mice; Micelles; Peptides, Cyclic; Protein Binding; Quinolines; Tetrahydroisoquinolines; Verapamil

2017
Thiol-reactive drug substrates of human P-glycoprotein label the same sites to activate ATPase activity in membranes or dodecyl maltoside detergent micelles.
    Biochemical and biophysical research communications, 2017, 07-08, Volume: 488, Issue:4

    Topics: Adenosine Triphosphatases; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Cell Membrane; Detergents; Enzyme Activation; Glucosides; Humans; Micelles; Quinolines; Rhodamines; Verapamil

2017