Page last updated: 2024-09-04

docetaxel anhydrous and panobinostat

docetaxel anhydrous has been researched along with panobinostat in 4 studies

Compound Research Comparison

Studies
(docetaxel anhydrous)
Trials
(docetaxel anhydrous)
Recent Studies (post-2010)
(docetaxel anhydrous)
Studies
(panobinostat)
Trials
(panobinostat)
Recent Studies (post-2010) (panobinostat)
12,1103,2166,92067895593

Protein Interaction Comparison

ProteinTaxonomydocetaxel anhydrous (IC50)panobinostat (IC50)
Histone deacetylase 8Schistosoma mansoni0.45
Histone deacetylase 3Homo sapiens (human)0.2031
Bromodomain-containing protein 4Homo sapiens (human)0.005
Cytochrome P450 3A5Homo sapiens (human)0.0033
Histone deacetylase 4Homo sapiens (human)0.3792
Histone deacetylase 1Homo sapiens (human)0.181
Histone deacetylase 7Homo sapiens (human)0.9434
Histone deacetylase 2Homo sapiens (human)0.2527
Polyamine deacetylase HDAC10Homo sapiens (human)0.007
Histone deacetylase 11 Homo sapiens (human)0.8396
Histone deacetylase 8Homo sapiens (human)0.46
Histone deacetylase 6Homo sapiens (human)0.2307
Histone deacetylase 9Homo sapiens (human)0.5825
Histone deacetylase 5Homo sapiens (human)0.3424
Histone deacetylase Plasmodium falciparum (malaria parasite P. falciparum)0.0025
Nuclear receptor corepressor 2Homo sapiens (human)0.002

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (75.00)24.3611
2020's1 (25.00)2.80

Authors

AuthorsStudies
Asquith, CRM; Crona, DJ; Koutentis, PA; Koyioni, M; Maffuid, KA; Mewada, HK; Murphy, WA; Torrice, CD1
Anand, A; Dzik-Jurasz, A; Hu, J; Rathkopf, D; Ross, RW; Scher, HI; Tanaka, E; Wong, BY; Woo, MM; Yang, W1
Chang, L; Chao, H; Graham, PH; Hao, J; Kearsley, JH; Li, Y; Ni, J; Wang, L1
Budman, DR; Calabro, A; Lesser, M; Rosen, L1

Trials

1 trial(s) available for docetaxel anhydrous and panobinostat

ArticleYear
A phase I study of oral panobinostat alone and in combination with docetaxel in patients with castration-resistant prostate cancer.
    Cancer chemotherapy and pharmacology, 2010, Volume: 66, Issue:1

    Topics: Acetylation; Administration, Oral; Aged; Aged, 80 and over; Antineoplastic Combined Chemotherapy Protocols; Docetaxel; Drug Resistance, Neoplasm; Fluorodeoxyglucose F18; Histone Deacetylase Inhibitors; Histones; Humans; Hydroxamic Acids; Indoles; Male; Maximum Tolerated Dose; Middle Aged; Neoplasm Metastasis; Neoplastic Cells, Circulating; Panobinostat; Positron-Emission Tomography; Prostate-Specific Antigen; Prostatic Neoplasms; Taxoids; Treatment Outcome

2010

Other Studies

3 other study(ies) available for docetaxel anhydrous and panobinostat

ArticleYear
Design and evaluation of 1,2,3-dithiazoles and fused 1,2,4-dithiazines as anti-cancer agents.
    Bioorganic & medicinal chemistry letters, 2021, 07-01, Volume: 43

    Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Design; Drug Screening Assays, Antitumor; Humans; Molecular Structure; Structure-Activity Relationship; Thiazoles

2021
Low dose histone deacetylase inhibitor, LBH589, potentiates anticancer effect of docetaxel in epithelial ovarian cancer via PI3K/Akt pathway in vitro.
    Cancer letters, 2013, Feb-01, Volume: 329, Issue:1

    Topics: Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Carcinoma, Ovarian Epithelial; Caspase 3; Cell Line, Tumor; Cell Proliferation; DNA Repair; Docetaxel; Dose-Response Relationship, Drug; Female; Histone Deacetylase Inhibitors; Histones; Humans; Hydroxamic Acids; Indoles; Neoplasms, Glandular and Epithelial; Ovarian Neoplasms; Panobinostat; Phosphatidylinositol 3-Kinases; Proto-Oncogene Proteins c-akt; Signal Transduction; Taxoids

2013
Identification of unique synergistic drug combinations associated with downexpression of survivin in a preclinical breast cancer model system.
    Anti-cancer drugs, 2012, Volume: 23, Issue:3

    Topics: Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Carboplatin; Caspase 3; Cell Line, Tumor; Deoxycytidine; Docetaxel; Down-Regulation; Doxorubicin; Drug Screening Assays, Antitumor; Fatty Acids, Monounsaturated; Female; Fluvastatin; Gemcitabine; Humans; Hydroxamic Acids; Indoles; Inhibitor of Apoptosis Proteins; Panobinostat; Receptor, ErbB-2; Survivin; Taxoids

2012